PL2010498T3 - Sposób otrzymywania acyloaminoalkilenoamidów użytecznych jako antagoniści substancji P - Google Patents
Sposób otrzymywania acyloaminoalkilenoamidów użytecznych jako antagoniści substancji PInfo
- Publication number
- PL2010498T3 PL2010498T3 PL07724154T PL07724154T PL2010498T3 PL 2010498 T3 PL2010498 T3 PL 2010498T3 PL 07724154 T PL07724154 T PL 07724154T PL 07724154 T PL07724154 T PL 07724154T PL 2010498 T3 PL2010498 T3 PL 2010498T3
- Authority
- PL
- Poland
- Prior art keywords
- acylaminoalkenylene
- antagonists
- synthesis
- substance
- amides useful
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D223/12—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Neurology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0607532A GB0607532D0 (en) | 2006-04-13 | 2006-04-13 | Organic compounds |
GB0610244A GB0610244D0 (en) | 2006-05-23 | 2006-05-23 | Organic compounds |
EP07724154A EP2010498B1 (en) | 2006-04-13 | 2007-04-11 | Synthesis of acylaminoalkenylene amides useful as substance p antagonists |
PCT/EP2007/003213 WO2007118651A1 (en) | 2006-04-13 | 2007-04-11 | Synthesis of acylaminoalkenylene amides useful as substance p antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
PL2010498T3 true PL2010498T3 (pl) | 2011-04-29 |
Family
ID=38324102
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL07724154T PL2010498T3 (pl) | 2006-04-13 | 2007-04-11 | Sposób otrzymywania acyloaminoalkilenoamidów użytecznych jako antagoniści substancji P |
Country Status (29)
Country | Link |
---|---|
US (2) | US8008479B2 (pl) |
EP (1) | EP2010498B1 (pl) |
JP (1) | JP5208917B2 (pl) |
KR (1) | KR20080108291A (pl) |
AR (1) | AR060506A1 (pl) |
AT (1) | ATE486853T1 (pl) |
AU (1) | AU2007237482B2 (pl) |
CA (1) | CA2645362C (pl) |
CL (1) | CL2007001040A1 (pl) |
CY (1) | CY1111294T1 (pl) |
DE (1) | DE602007010269D1 (pl) |
DK (1) | DK2010498T3 (pl) |
EC (1) | ECSP088820A (pl) |
GT (1) | GT200800209A (pl) |
HK (1) | HK1125640A1 (pl) |
HR (1) | HRP20110045T1 (pl) |
JO (1) | JO2630B1 (pl) |
MA (1) | MA30394B1 (pl) |
MX (1) | MX2008013117A (pl) |
MY (1) | MY145069A (pl) |
NO (1) | NO20084783L (pl) |
NZ (1) | NZ571142A (pl) |
PE (1) | PE20071223A1 (pl) |
PL (1) | PL2010498T3 (pl) |
PT (1) | PT2010498E (pl) |
RU (1) | RU2433122C2 (pl) |
SI (1) | SI2010498T1 (pl) |
TW (1) | TW200815358A (pl) |
WO (1) | WO2007118651A1 (pl) |
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ES2356334T3 (es) | 2007-06-12 | 2011-04-07 | Concert Pharmaceuticals, Inc. | Derivados de azapéptidos como inhibidores de la proteasa vih. |
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US8809521B2 (en) | 2007-08-28 | 2014-08-19 | Fmc Biopolymer As | Delayed self-gelling alginate systems and uses thereof |
WO2009035662A1 (en) | 2007-09-12 | 2009-03-19 | Concert Pharmaceuticals, Inc. | Deuterated 4 -oxoquinoline derivatives for the treatment of hiv infection |
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US8410124B2 (en) | 2007-10-18 | 2013-04-02 | Concert Pharmaceuticals Inc. | Deuterated etravirine |
US8592487B2 (en) | 2007-10-26 | 2013-11-26 | Concert Pharmaceuticals, Inc. | Deuterated darunavir |
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US8609673B2 (en) | 2008-01-22 | 2013-12-17 | Concert Pharmaceuticals, Inc. | Vandetanib derivatives |
WO2009094216A1 (en) | 2008-01-22 | 2009-07-30 | Concert Pharmaceuticals Inc. | Derivatives of gefitinib |
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WO2009154754A2 (en) | 2008-06-17 | 2009-12-23 | Concert Pharmaceuticals, Inc. | Synthesis of deuterated morpholine derivatives |
JP5183808B2 (ja) | 2008-08-29 | 2013-04-17 | コンサート ファーマシューティカルズ インコーポレイテッド | 置換トリアゾロ−ピリダジン誘導体 |
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US9045453B2 (en) | 2008-11-14 | 2015-06-02 | Concert Pharmaceuticals, Inc. | Substituted dioxopiperidinyl phthalimide derivatives |
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US9260432B2 (en) | 2009-09-02 | 2016-02-16 | Concert Pharmaceuticals, Inc. | Substituted derivatives of bicyclic [4.3.0] heteroaryl compounds |
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US8278460B2 (en) | 2009-10-15 | 2012-10-02 | Concert Pharmaceuticals, Inc. | Substituted benzimidazoles |
US8471034B2 (en) | 2009-11-18 | 2013-06-25 | Concert Pharmaceuticals, Inc. | Niacin prodrugs and deuterated versions thereof |
DE102010001040A1 (de) | 2010-01-20 | 2011-07-21 | Evonik RohMax Additives GmbH, 64293 | (Meth)acrylat-Polymere zur Verbesserung des Viskositätsindexes |
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US8759394B2 (en) | 2011-02-14 | 2014-06-24 | Concert Pharmaceuticals, Inc. | 4-hydroxybutyric acid analogs |
US9145390B2 (en) | 2011-03-03 | 2015-09-29 | Concert Pharmaceuticals, Inc. | Derivatives of pyrazole-substituted amino-heteroaryl compounds |
WO2012122028A2 (en) | 2011-03-04 | 2012-09-13 | Concert Pharmaceuticals Inc. | Pyrazinoisoquinoline compounds |
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US9328113B2 (en) | 2012-04-13 | 2016-05-03 | Concert Pharmaceuticals, Inc. | Substituted xanthine derivatives |
US9249093B2 (en) | 2012-04-20 | 2016-02-02 | Concert Pharmaceuticals, Inc. | Deuterated rigosertib |
US20150197525A1 (en) | 2012-06-15 | 2015-07-16 | Concert Pharmaceuticals, Inc. | Deuterated derivatives of ruxolitinib |
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US10017445B2 (en) | 2012-07-12 | 2018-07-10 | Concert Pharmaceuticals, Inc. | Deuterated idebenone |
KR20150038486A (ko) | 2012-07-30 | 2015-04-08 | 콘서트 파마슈티컬즈, 인크. | 중수소화된 아이브루티닙 |
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JP2015534989A (ja) | 2012-10-22 | 2015-12-07 | コンサート ファーマシューティカルズ インコーポレイテッド | {s−3−(4−アミノ−1−オキソ−イソインドリン−2−イル)(ピペリジン−3,4,4,5,5−d5)−2,6−ジオン}の固体形態 |
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US8906951B1 (en) | 2013-06-24 | 2014-12-09 | Tigercat Pharma, Inc. | Use of NK-1 receptor antagonists in pruritus |
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CN106459056A (zh) | 2014-02-10 | 2017-02-22 | 康塞特医药品公司 | 经取代的三唑苯二氮卓 |
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AU2016327603B2 (en) | 2015-09-25 | 2021-04-22 | Vertex Pharmaceuticals (Europe) Limited | Deuterated CFTR potentiators |
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US10442761B2 (en) | 2016-02-16 | 2019-10-15 | Concert Pharmaceuticals, Inc. | Deuterated GFT-505 |
CN111491629A (zh) | 2017-11-22 | 2020-08-04 | 康塞特医药品公司 | D-丝氨酸的氘化类似物及其用途 |
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Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HU226562B1 (en) * | 1995-02-22 | 2009-04-28 | Novartis Ag | 1-aryl-2-acylamino-ethane compounds as neurokinin, especially neurokinin-1 antagonists, and medicaments containing the said compounds. |
MY132550A (en) * | 1996-08-22 | 2007-10-31 | Novartis Ag | Acylaminoalkenylene-amide derivatives as nk1 and nk2 antogonists |
GB0010958D0 (en) * | 2000-05-05 | 2000-06-28 | Novartis Ag | Organic compounds |
-
2007
- 2007-04-10 JO JO2007129A patent/JO2630B1/en active
- 2007-04-11 WO PCT/EP2007/003213 patent/WO2007118651A1/en active Application Filing
- 2007-04-11 KR KR1020087024839A patent/KR20080108291A/ko not_active Application Discontinuation
- 2007-04-11 PE PE2007000444A patent/PE20071223A1/es not_active Application Discontinuation
- 2007-04-11 AR ARP070101533A patent/AR060506A1/es not_active Application Discontinuation
- 2007-04-11 DE DE602007010269T patent/DE602007010269D1/de active Active
- 2007-04-11 AT AT07724154T patent/ATE486853T1/de active
- 2007-04-11 PT PT07724154T patent/PT2010498E/pt unknown
- 2007-04-11 CA CA2645362A patent/CA2645362C/en not_active Expired - Fee Related
- 2007-04-11 JP JP2009504637A patent/JP5208917B2/ja not_active Expired - Fee Related
- 2007-04-11 NZ NZ571142A patent/NZ571142A/en not_active IP Right Cessation
- 2007-04-11 DK DK07724154.5T patent/DK2010498T3/da active
- 2007-04-11 MX MX2008013117A patent/MX2008013117A/es active IP Right Grant
- 2007-04-11 AU AU2007237482A patent/AU2007237482B2/en not_active Ceased
- 2007-04-11 PL PL07724154T patent/PL2010498T3/pl unknown
- 2007-04-11 US US12/296,969 patent/US8008479B2/en not_active Expired - Fee Related
- 2007-04-11 RU RU2008145102/04A patent/RU2433122C2/ru not_active IP Right Cessation
- 2007-04-11 SI SI200730483T patent/SI2010498T1/sl unknown
- 2007-04-11 EP EP07724154A patent/EP2010498B1/en active Active
- 2007-04-12 TW TW096112886A patent/TW200815358A/zh unknown
- 2007-04-12 CL CL200701040A patent/CL2007001040A1/es unknown
-
2008
- 2008-10-08 MY MYPI20083997A patent/MY145069A/en unknown
- 2008-10-10 GT GT200800209A patent/GT200800209A/es unknown
- 2008-10-13 EC EC2008008820A patent/ECSP088820A/es unknown
- 2008-11-03 MA MA31347A patent/MA30394B1/fr unknown
- 2008-11-12 NO NO20084783A patent/NO20084783L/no not_active Application Discontinuation
-
2009
- 2009-05-15 HK HK09104457.9A patent/HK1125640A1/xx not_active IP Right Cessation
-
2011
- 2011-01-21 HR HR20110045T patent/HRP20110045T1/hr unknown
- 2011-01-26 CY CY20111100082T patent/CY1111294T1/el unknown
- 2011-07-22 US US13/188,795 patent/US20110282053A1/en not_active Abandoned
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