PL1809624T3 - Pochodne pirymidynosulfonoamidu jako modulatory receptora chemokinowego - Google Patents
Pochodne pirymidynosulfonoamidu jako modulatory receptora chemokinowegoInfo
- Publication number
- PL1809624T3 PL1809624T3 PL05773278T PL05773278T PL1809624T3 PL 1809624 T3 PL1809624 T3 PL 1809624T3 PL 05773278 T PL05773278 T PL 05773278T PL 05773278 T PL05773278 T PL 05773278T PL 1809624 T3 PL1809624 T3 PL 1809624T3
- Authority
- PL
- Poland
- Prior art keywords
- chemokine receptor
- receptor modulators
- sulphonamide derivatives
- pyrimidine sulphonamide
- pyrimidine
- Prior art date
Links
- 102000009410 Chemokine receptor Human genes 0.000 title 1
- 108050000299 Chemokine receptor Proteins 0.000 title 1
- WJJBIYLGJUVNJX-UHFFFAOYSA-N pyrimidine-2-sulfonamide Chemical class NS(=O)(=O)C1=NC=CC=N1 WJJBIYLGJUVNJX-UHFFFAOYSA-N 0.000 title 1
Classifications
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- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0419235A GB0419235D0 (en) | 2004-08-28 | 2004-08-28 | Compounds |
| GB0502544A GB0502544D0 (en) | 2005-02-08 | 2005-02-08 | Compounds |
| PCT/GB2005/003257 WO2006024823A1 (en) | 2004-08-28 | 2005-08-23 | Pyrimidine sulphonamide derivatives as chemokine receptor modulators |
| EP05773278.6A EP1809624B1 (en) | 2004-08-28 | 2005-08-23 | Pyrimidine sulphonamide derivatives as chemokine receptor modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL1809624T3 true PL1809624T3 (pl) | 2014-03-31 |
Family
ID=35549576
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL05773278T PL1809624T3 (pl) | 2004-08-28 | 2005-08-23 | Pochodne pirymidynosulfonoamidu jako modulatory receptora chemokinowego |
Country Status (27)
| Country | Link |
|---|---|
| US (5) | US7838675B2 (pl) |
| EP (3) | EP2311827A1 (pl) |
| JP (3) | JP4795352B2 (pl) |
| KR (1) | KR101280095B1 (pl) |
| CN (1) | CN102796081B (pl) |
| AR (1) | AR050617A1 (pl) |
| AU (1) | AU2005279045B2 (pl) |
| BR (1) | BRPI0514735B8 (pl) |
| CA (1) | CA2578441C (pl) |
| CY (1) | CY1114803T1 (pl) |
| DK (1) | DK1809624T3 (pl) |
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| HR (1) | HRP20140023T1 (pl) |
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| ME (1) | ME01620B (pl) |
| MX (1) | MX2007002240A (pl) |
| MY (1) | MY148125A (pl) |
| NO (1) | NO338749B1 (pl) |
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| PT (1) | PT1809624E (pl) |
| RS (1) | RS53145B (pl) |
| RU (1) | RU2408587C2 (pl) |
| SI (1) | SI1809624T1 (pl) |
| TW (1) | TWI369983B (pl) |
| UY (1) | UY29085A1 (pl) |
| WO (1) | WO2006024823A1 (pl) |
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| JPS6262286A (ja) * | 1985-09-13 | 1987-03-18 | 株式会社東芝 | 沸騰水型原子炉炉心 |
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| RU2395503C2 (ru) | 2004-05-19 | 2010-07-27 | Зольвай Фармасьютиклз Гмбх | Лекарственные средства, содержащие n-сульфамоил-n'-арилпиперазины, предназначенные для профилактики или лечения ожирения и связанных с ним состояний |
| RU2408587C2 (ru) | 2004-08-24 | 2011-01-10 | Астразенека Аб | Производные пиримидинсульфонамида в качестве модуляторов рецепторов хемокинов |
| JP2008540539A (ja) | 2005-05-10 | 2008-11-20 | バーテックス ファーマシューティカルズ インコーポレイテッド | イオンチャンネルの調節因子としての二環系誘導体 |
| EP2099444A4 (en) | 2006-12-14 | 2012-11-07 | Nps Pharma Inc | USE OF D-SERIN DERIVATIVES FOR THE TREATMENT OF ANTIBODIES |
| US20100137398A1 (en) * | 2007-05-04 | 2010-06-03 | Novartis Ag | Use of hdac inhibitors for the treatment of gastrointestinal cancers |
| WO2009151910A2 (en) * | 2008-05-25 | 2009-12-17 | Wyeth | Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer |
| KR20110031462A (ko) * | 2008-07-16 | 2011-03-28 | 아스트라제네카 아베 | 피리미딜 술폰아미드 유도체 및 케모카인 매개 질환의 치료를 위한 그의 용도 |
| CA2762680C (en) | 2009-05-21 | 2018-04-17 | Chlorion Pharma, Inc. | Methyl sulfanyl pyrmidmes useful as antiinflammatories, analgesics, and antiepileptics |
| AR080375A1 (es) | 2010-03-05 | 2012-04-04 | Sanofi Aventis | Procedimiento para la preparacion de 2-(cicloheximetil)-n-{2-[(2s)-1-metilpirrolidin-2-il] etil}-1,2,3,4-tetrahidroisoquinolina- 7-sulfonamida |
| WO2012007748A1 (en) * | 2010-07-13 | 2012-01-19 | Astrazeneca Ab | New crystalline forms of n-[2-[[(2,3-difluoropheny)methyl)thio]-6-{[(1r,2s)-2,3-dihydroxy-1- methylpropyl]oxy}-4-pyrimidinyl]-1-azetidinesulfonamide |
| MX342874B (es) | 2011-07-12 | 2016-10-17 | Astrazeneca Ab | N-(6-((2r,3s)-3,4-dihidroxibutan-2-iloxi)-2-(4-fluorobenciltio)pi rimidin-4-il)-3-metilacetidina-1-sulfonamida como modulador del receptor de quimiocina. |
| TW201512171A (zh) | 2013-04-19 | 2015-04-01 | Pfizer Ltd | 化學化合物 |
| PT3263133T (pt) | 2015-02-27 | 2020-05-21 | Univ Kyushu Nat Univ Corp | Composto de piridinona e a sua utilização |
| EP3426253A4 (en) * | 2016-03-11 | 2019-11-06 | Ardea Biosciences, Inc. | CXCR-2 INHIBITORS FOR THE TREATMENT OF CRYSTALARTHROPATHIES |
| US10660909B2 (en) | 2016-11-17 | 2020-05-26 | Syntrix Biosystems Inc. | Method for treating cancer using chemokine antagonists |
| WO2019165315A1 (en) | 2018-02-23 | 2019-08-29 | Syntrix Biosystems Inc. | Method for treating cancer using chemokine antagonists alone or in combination |
| WO2023028077A1 (en) | 2021-08-24 | 2023-03-02 | Genentech, Inc. | Sodium channel inhibitors and methods of designing same |
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2005
- 2005-08-23 RU RU2007106037/04A patent/RU2408587C2/ru active
- 2005-08-23 ME MEP-2014-3A patent/ME01620B/me unknown
- 2005-08-23 WO PCT/GB2005/003257 patent/WO2006024823A1/en not_active Ceased
- 2005-08-23 DK DK05773278.6T patent/DK1809624T3/da active
- 2005-08-23 NZ NZ553335A patent/NZ553335A/en not_active IP Right Cessation
- 2005-08-23 EP EP10194614A patent/EP2311827A1/en not_active Withdrawn
- 2005-08-23 MX MX2007002240A patent/MX2007002240A/es active IP Right Grant
- 2005-08-23 EP EP05773278.6A patent/EP1809624B1/en not_active Expired - Lifetime
- 2005-08-23 AU AU2005279045A patent/AU2005279045B2/en not_active Expired
- 2005-08-23 HR HRP20140023TT patent/HRP20140023T1/hr unknown
- 2005-08-23 PL PL05773278T patent/PL1809624T3/pl unknown
- 2005-08-23 CN CN201210247005.5A patent/CN102796081B/zh not_active Expired - Lifetime
- 2005-08-23 US US11/574,340 patent/US7838675B2/en active Active
- 2005-08-23 JP JP2007528961A patent/JP4795352B2/ja not_active Expired - Lifetime
- 2005-08-23 EP EP10194616A patent/EP2301933A1/en not_active Withdrawn
- 2005-08-23 CA CA2578441A patent/CA2578441C/en not_active Expired - Lifetime
- 2005-08-23 KR KR1020077004736A patent/KR101280095B1/ko not_active Expired - Lifetime
- 2005-08-23 ES ES05773278.6T patent/ES2442678T3/es not_active Expired - Lifetime
- 2005-08-23 SI SI200531819T patent/SI1809624T1/sl unknown
- 2005-08-23 RS RS20140015A patent/RS53145B/sr unknown
- 2005-08-23 BR BRPI0514735A patent/BRPI0514735B8/pt active IP Right Grant
- 2005-08-23 PT PT5773278T patent/PT1809624E/pt unknown
- 2005-08-25 MY MYPI20054004A patent/MY148125A/en unknown
- 2005-08-26 TW TW094129379A patent/TWI369983B/zh not_active IP Right Cessation
- 2005-08-26 AR ARP050103584A patent/AR050617A1/es active IP Right Grant
- 2005-08-26 UY UY29085A patent/UY29085A1/es not_active Application Discontinuation
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2007
- 2007-02-08 IL IL181241A patent/IL181241A0/en active IP Right Grant
- 2007-03-27 NO NO20071594A patent/NO338749B1/no unknown
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2010
- 2010-11-17 US US12/947,916 patent/US8269002B2/en not_active Expired - Lifetime
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2011
- 2011-01-26 JP JP2011013745A patent/JP5364735B2/ja not_active Expired - Lifetime
- 2011-12-23 US US13/336,269 patent/US8410123B2/en not_active Expired - Lifetime
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2012
- 2012-09-14 US US13/620,075 patent/US20130012490A1/en not_active Abandoned
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2013
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