PH26678A - 4-(aroylamino) piperidine butanamide derivatives - Google Patents

4-(aroylamino) piperidine butanamide derivatives Download PDF

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Publication number
PH26678A
PH26678A PH35495A PH35495A PH26678A PH 26678 A PH26678 A PH 26678A PH 35495 A PH35495 A PH 35495A PH 35495 A PH35495 A PH 35495A PH 26678 A PH26678 A PH 26678A
Authority
PH
Philippines
Prior art keywords
parts
amino
alkyl
hydrogen
formula
Prior art date
Application number
PH35495A
Other languages
English (en)
Inventor
George Van Daele
Freddy Vlaeminck
Francois Sommen
Michel De Cleyn
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PH26678A publication Critical patent/PH26678A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PH35495A 1986-07-03 1987-07-03 4-(aroylamino) piperidine butanamide derivatives PH26678A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US88206786A 1986-07-03 1986-07-03

Publications (1)

Publication Number Publication Date
PH26678A true PH26678A (en) 1992-09-15

Family

ID=25379820

Family Applications (1)

Application Number Title Priority Date Filing Date
PH35495A PH26678A (en) 1986-07-03 1987-07-03 4-(aroylamino) piperidine butanamide derivatives

Country Status (25)

Country Link
EP (1) EP0251417B1 (ru)
JP (1) JP2512755B2 (ru)
KR (1) KR960009422B1 (ru)
CN (1) CN87104641A (ru)
AT (1) ATE88181T1 (ru)
AU (1) AU593660B2 (ru)
BG (1) BG80406A (ru)
CA (1) CA1311755C (ru)
DE (1) DE3785393T2 (ru)
DK (1) DK336387A (ru)
ES (1) ES2054653T3 (ru)
FI (1) FI90863C (ru)
HU (1) HU204254B (ru)
IE (1) IE60342B1 (ru)
IL (1) IL83045A (ru)
MA (1) MA21026A1 (ru)
NO (1) NO171908C (ru)
NZ (1) NZ220779A (ru)
PH (1) PH26678A (ru)
PT (1) PT85232B (ru)
SU (1) SU1620049A3 (ru)
TN (1) TNSN87085A1 (ru)
ZA (1) ZA874810B (ru)
ZM (1) ZM5487A1 (ru)
ZW (1) ZW12187A1 (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ225152A (en) * 1987-07-17 1990-04-26 Janssen Pharmaceutica Nv Heterocyclically substituted piperidinyl benzamides as pharmaceuticals
US5130312A (en) * 1987-07-17 1992-07-14 Janssen Pharmaceutica N.V. Substituted N-(3-hydroxy-4-piperidinyl)benzamides
CA1317940C (en) * 1987-09-25 1993-05-18 Georges H. P. Van Daele Substituted n-(1-alkyl-3-hydroxy-4-piperidinyl)benzamides
US4975439A (en) * 1987-09-25 1990-12-04 Janssen Pharmaceutical N.V. Novel substituted N-(1-alkyl-3-hydroxy-4-piperidinyl)benzamides
US5041454A (en) * 1987-09-25 1991-08-20 Janssen Pharmaceutica N.V. Novel substituted N-(1-alkyl-3-hydroxy-4-piperidinyl)benzamides
TW294595B (ru) * 1992-11-20 1997-01-01 Janssen Pharmaceutica Nv
JP3235913B2 (ja) * 1993-07-30 2001-12-04 エーザイ株式会社 アミノ安息香酸誘導体
US5585387A (en) * 1994-10-07 1996-12-17 Torcan Chemical Ltd. Prepration of cisapride
RU2008139599A (ru) 2006-03-07 2010-04-20 Эррэй Биофарма Инк. (Us) Гетеробициклические производные пиразола и способы их применения

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1183847A (en) * 1981-10-01 1985-03-12 Georges Van Daele N-(3-hydroxy-4-piperidinyl)benzamide derivatives

Also Published As

Publication number Publication date
HU204254B (en) 1991-12-30
IE60342B1 (en) 1994-06-29
KR880001593A (ko) 1988-04-25
MA21026A1 (fr) 1988-04-01
IE871766L (en) 1988-01-03
DK336387A (da) 1988-01-04
EP0251417A3 (en) 1989-04-26
JP2512755B2 (ja) 1996-07-03
ATE88181T1 (de) 1993-04-15
DE3785393D1 (de) 1993-05-19
FI872930A (fi) 1988-01-04
ES2054653T3 (es) 1994-08-16
CA1311755C (en) 1992-12-22
NZ220779A (en) 1989-09-27
IL83045A0 (en) 1987-12-31
FI90863B (fi) 1993-12-31
ZW12187A1 (en) 1989-02-01
PT85232B (pt) 1990-03-30
NO872781D0 (no) 1987-07-02
PT85232A (pt) 1987-08-01
AU593660B2 (en) 1990-02-15
BG80406A (bg) 1993-12-24
EP0251417A2 (en) 1988-01-07
NO872781L (no) 1988-01-04
KR960009422B1 (en) 1996-07-19
CN87104641A (zh) 1988-02-03
ZA874810B (en) 1989-02-22
AU7506787A (en) 1988-01-07
FI872930A0 (fi) 1987-07-02
IL83045A (en) 1991-07-18
DK336387D0 (da) 1987-06-30
TNSN87085A1 (fr) 1990-01-01
EP0251417B1 (en) 1993-04-14
DE3785393T2 (de) 1993-07-29
NO171908B (no) 1993-02-08
JPS6322575A (ja) 1988-01-30
NO171908C (no) 1993-05-19
HUT48588A (en) 1989-06-28
SU1620049A3 (ru) 1991-01-07
ZM5487A1 (en) 1988-06-27
FI90863C (fi) 1994-04-11

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