PH24313A - Emulsion composition for administration of sparingly water soluble ionizable hydrophobic drugs - Google Patents

Emulsion composition for administration of sparingly water soluble ionizable hydrophobic drugs

Info

Publication number
PH24313A
PH24313A PH34241A PH34241A PH24313A PH 24313 A PH24313 A PH 24313A PH 34241 A PH34241 A PH 34241A PH 34241 A PH34241 A PH 34241A PH 24313 A PH24313 A PH 24313A
Authority
PH
Philippines
Prior art keywords
administration
water soluble
sparingly water
emulsion composition
hydrophobic drugs
Prior art date
Application number
PH34241A
Other languages
English (en)
Inventor
Narendra Raghunathji Desai
Madurai Ganesan
Eugene Albert Carpenter
Edward Charles Shinal
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of PH24313A publication Critical patent/PH24313A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/541—Organic ions forming an ion pair complex with the pharmacologically or therapeutically active agent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Colloid Chemistry (AREA)
PH34241A 1985-09-11 1986-09-10 Emulsion composition for administration of sparingly water soluble ionizable hydrophobic drugs PH24313A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/774,762 US4816247A (en) 1985-09-11 1985-09-11 Emulsion compositions for administration of sparingly water soluble ionizable hydrophobic drugs

Publications (1)

Publication Number Publication Date
PH24313A true PH24313A (en) 1990-05-29

Family

ID=25102201

Family Applications (1)

Application Number Title Priority Date Filing Date
PH34241A PH24313A (en) 1985-09-11 1986-09-10 Emulsion composition for administration of sparingly water soluble ionizable hydrophobic drugs

Country Status (18)

Country Link
US (1) US4816247A (de)
EP (1) EP0214501B1 (de)
JP (1) JPS62111915A (de)
KR (1) KR900000211B1 (de)
AT (1) ATE80795T1 (de)
AU (1) AU593014B2 (de)
CA (1) CA1272685A (de)
DE (1) DE3686797T2 (de)
DK (1) DK432586A (de)
ES (1) ES2001950A6 (de)
FI (1) FI86142C (de)
GR (1) GR862316B (de)
HU (1) HU196700B (de)
IE (1) IE59828B1 (de)
NO (1) NO171145C (de)
NZ (1) NZ217483A (de)
PH (1) PH24313A (de)
ZA (1) ZA866899B (de)

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JPH06157294A (ja) * 1992-11-19 1994-06-03 Tanabe Seiyaku Co Ltd 脂肪微粒子製剤
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US6682758B1 (en) 1998-12-22 2004-01-27 The United States Of America As Represented By The Department Of Health And Human Services Water-insoluble drug delivery system
US6383471B1 (en) * 1999-04-06 2002-05-07 Lipocine, Inc. Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents
US6720001B2 (en) 1999-10-18 2004-04-13 Lipocine, Inc. Emulsion compositions for polyfunctional active ingredients
EP1280556A1 (de) 2000-05-05 2003-02-05 Wisconsin Alumni Research Foundation Zusammensetzungen und verfahren zum schutz von zellen während der chemotherpie und strahlentherapie
EP1303261B1 (de) * 2000-07-24 2005-03-09 Pharmacia & Upjohn Company Selbstemulgierendes system zur abgabe von sehr wasserunlöslichen und lipophilen arzneimitteln
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AU2003235360A1 (en) * 2002-05-22 2003-12-02 Nihon Pharmaceutical Co., Ltd. Smooth muscle peristole inhibitor
US20040053895A1 (en) * 2002-09-18 2004-03-18 Bone Care International, Inc. Multi-use vessels for vitamin D formulations
US20040058895A1 (en) * 2002-09-18 2004-03-25 Bone Care International, Inc. Multi-use vessels for vitamin D formulations
US7148211B2 (en) * 2002-09-18 2006-12-12 Genzyme Corporation Formulation for lipophilic agents
US20050026877A1 (en) * 2002-12-03 2005-02-03 Novacea, Inc. Pharmaceutical compositions comprising active vitamin D compounds
US9254294B2 (en) 2003-02-24 2016-02-09 Pharmaceutical Productions Inc. Transmucosal hormone delivery system
US10172810B2 (en) 2003-02-24 2019-01-08 Pharmaceutical Productions, Inc. Transmucosal ketamine delivery composition
WO2004075877A1 (en) * 2003-02-24 2004-09-10 Pharmaceutical Productions, Inc. Transmucosal drug delivery system
US9358296B2 (en) 2003-02-24 2016-06-07 Pharmaceutical Productions Inc. Transmucosal drug delivery system
US9498454B2 (en) 2003-02-24 2016-11-22 Pharmaceutical Productions Inc. Transmucosal drug delivery system
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US20060189586A1 (en) * 2003-06-11 2006-08-24 Cleland Jeffrey L Pharmaceutical compositions comprising active vitamin D compounds
US7871632B2 (en) 2004-07-12 2011-01-18 Adventrx Pharmaceuticals, Inc. Compositions for delivering highly water soluble drugs
US8557861B2 (en) * 2004-09-28 2013-10-15 Mast Therapeutics, Inc. Low oil emulsion compositions for delivering taxoids and other insoluble drugs
JP4940152B2 (ja) 2005-01-05 2012-05-30 イーライ リリー アンド カンパニー パモ酸オランザピン二水和物
TWI376239B (en) * 2006-02-01 2012-11-11 Andrew Xian Chen Vitamin e succinate stabilized pharmaceutical compositions, methods for the preparation and the use thereof
EP2200613B1 (de) 2007-09-21 2018-09-05 The Johns Hopkins University Phenazin-derivate und ihre verwendungen
BRPI0801417B8 (pt) * 2008-03-13 2021-05-25 Univ Minas Gerais processo para obtenção de composição farmacêutica de retinóides, produto derivado de retinóides e uso
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JP5468221B2 (ja) * 2008-08-04 2014-04-09 株式会社 メドレックス 難溶性薬物の静注用分散製剤
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Also Published As

Publication number Publication date
CA1272685A (en) 1990-08-14
KR870002834A (ko) 1987-04-13
JPS62111915A (ja) 1987-05-22
DE3686797D1 (de) 1992-10-29
ZA866899B (en) 1987-05-27
NO863620D0 (no) 1986-09-10
IE59828B1 (en) 1994-04-06
DK432586A (da) 1987-03-12
AU6253886A (en) 1987-03-12
GR862316B (en) 1987-01-13
KR900000211B1 (ko) 1990-01-23
IE862408L (en) 1987-03-11
ES2001950A6 (es) 1988-07-01
EP0214501A3 (en) 1987-09-09
AU593014B2 (en) 1990-02-01
FI86142B (fi) 1992-04-15
FI863664A0 (fi) 1986-09-10
DE3686797T2 (de) 1993-03-25
NO171145B (no) 1992-10-26
DK432586D0 (da) 1986-09-10
HU196700B (en) 1989-01-30
ATE80795T1 (de) 1992-10-15
EP0214501B1 (de) 1992-09-23
FI863664L (fi) 1987-03-12
EP0214501A2 (de) 1987-03-18
HUT43948A (en) 1988-01-28
US4816247A (en) 1989-03-28
FI86142C (fi) 1992-07-27
NO171145C (no) 1993-02-03
NZ217483A (en) 1990-08-28
NO863620L (no) 1987-03-12

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