PH19222A - Novel enkephalin derivatives - Google Patents

Novel enkephalin derivatives

Info

Publication number
PH19222A
PH19222A PH24144A PH24144A PH19222A PH 19222 A PH19222 A PH 19222A PH 24144 A PH24144 A PH 24144A PH 24144 A PH24144 A PH 24144A PH 19222 A PH19222 A PH 19222A
Authority
PH
Philippines
Prior art keywords
enkephalin derivatives
novel
novel enkephalin
derivatives
enkephalin
Prior art date
Application number
PH24144A
Other languages
English (en)
Inventor
Albert A Carr
Robert A Farr
John M Kane
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of PH19222A publication Critical patent/PH19222A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1024Tetrapeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
PH24144A 1979-06-21 1980-06-16 Novel enkephalin derivatives PH19222A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5095079A 1979-06-21 1979-06-21
US06/130,431 US4341698A (en) 1979-06-21 1980-03-14 Enkaphalin derivatives
AU91877/82A AU559278B2 (en) 1979-06-21 1982-12-24 Piperazines

Publications (1)

Publication Number Publication Date
PH19222A true PH19222A (en) 1986-02-12

Family

ID=36764304

Family Applications (1)

Application Number Title Priority Date Filing Date
PH24144A PH19222A (en) 1979-06-21 1980-06-16 Novel enkephalin derivatives

Country Status (17)

Country Link
US (1) US4341698A (no)
AU (1) AU559278B2 (no)
CA (1) CA1161838A (no)
CH (2) CH648835A5 (no)
DE (1) DE3022401A1 (no)
DK (1) DK265780A (no)
ES (1) ES8105720A1 (no)
FR (2) FR2459236A1 (no)
GB (3) GB2051821B (no)
IE (1) IE49834B1 (no)
IL (1) IL60245A (no)
IT (1) IT1148277B (no)
NL (1) NL8003580A (no)
NO (1) NO801855L (no)
NZ (1) NZ193934A (no)
PH (1) PH19222A (no)
SE (3) SE447250B (no)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6369080B2 (en) 1996-10-11 2002-04-09 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6063794A (en) 1996-10-11 2000-05-16 Cor Therapeutics Inc. Selective factor Xa inhibitors
US6194435B1 (en) 1996-10-11 2001-02-27 Cor Therapeutics, Inc. Lactams as selective factor Xa inhibitors
US6262047B1 (en) 1996-10-11 2001-07-17 Cor Therapeutics, Inc. Selective factor Xa inhibitors
NZ500353A (en) 1997-04-14 2002-02-01 Cor Therapeutics Inc Cyclic diaza compounds that are selective inhibitors of factor Xa
AU741099B2 (en) * 1997-04-14 2001-11-22 Millennium Pharmaceuticals, Inc. Selective factor Xa inhibitors
US6369063B1 (en) 1997-04-14 2002-04-09 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6218382B1 (en) 1997-08-11 2001-04-17 Cor Therapeutics, Inc Selective factor Xa inhibitors
US6333321B1 (en) 1997-08-11 2001-12-25 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6228854B1 (en) 1997-08-11 2001-05-08 Cor Therapeutics, Inc. Selective factor Xa inhibitors
EP1868434A4 (en) 2005-03-22 2011-10-26 Azevan Pharmaceuticals Inc BETA-LACTAMYL ALKANIC ACIDS FOR THE TREATMENT OF PREMIERSTRUELLEN FAULTS
KR101523776B1 (ko) 2005-07-19 2015-05-28 아제반 파마슈티칼스, 인코퍼레이티드 베타-락타민 페닐알라닌, 시스테인 그리고 세린 바소프레신길항물질
JP2009532385A (ja) * 2006-03-30 2009-09-10 パラティン・テクノロジーズ・インコーポレーテッド 線状ナトリウム利尿ペプチド構築物
WO2007115175A2 (en) * 2006-03-30 2007-10-11 Palatin Technologies, Inc. Cyclic natriuretic peptide constructs
US8580746B2 (en) 2006-03-30 2013-11-12 Palatin Technologies, Inc. Amide linkage cyclic natriuretic peptide constructs
US7964181B2 (en) * 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
MX2008012649A (es) * 2006-03-30 2008-10-13 Palatin Technologies Inc Sustitutos de aminoacido para constructos peptidicos.
US8114844B2 (en) * 2006-03-30 2012-02-14 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptidomimetics
EP2684871B1 (en) * 2006-12-19 2016-05-04 F. Hoffmann-La Roche AG Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives
CA2728373A1 (en) * 2008-06-18 2009-12-23 F.Hoffmann-La Roche Ag Aryl ketone as mri
PL2587919T3 (pl) 2010-07-01 2018-05-30 Azevan Pharmaceuticals, Inc. Sposoby leczenia zespołu stresu pourazowego
NZ724718A (en) 2014-03-28 2023-04-28 Azevan Pharmaceuticals Inc Compositions and methods for treating neurodegenerative diseases
CA3075759A1 (en) 2017-09-15 2019-03-21 Azevan Pharmaceuticals, Inc. Compositions and methods for treating brain injury

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604845A1 (de) * 1976-02-07 1977-08-18 Knoll Ag Neue piperazinderivate
US4254107A (en) * 1979-11-27 1981-03-03 Merck & Co., Inc. Long-lasting agonists of enkephalin

Also Published As

Publication number Publication date
SE8500877D0 (sv) 1985-02-22
US4341698A (en) 1982-07-27
FR2473042A1 (fr) 1981-07-10
DE3022401A1 (de) 1981-01-08
GB2132605A (en) 1984-07-11
GB2106515B (en) 1983-11-23
FR2473042B1 (no) 1983-07-01
GB2106515A (en) 1983-04-13
IE801152L (en) 1980-12-21
ES492566A0 (es) 1981-06-16
FR2459236B1 (no) 1984-01-06
ES8105720A1 (es) 1981-06-16
SE8500877L (sv) 1985-02-22
CA1161838A (en) 1984-02-07
IT8049032A0 (it) 1980-06-20
NZ193934A (en) 1983-02-15
SE460540B (sv) 1989-10-23
NL8003580A (nl) 1980-12-23
CH648835A5 (de) 1985-04-15
IT1148277B (it) 1986-11-26
GB2132605B (en) 1985-01-03
CH645363A5 (de) 1984-09-28
GB2051821B (en) 1983-04-27
DK265780A (da) 1980-12-22
SE8004254L (sv) 1980-12-22
FR2459236A1 (fr) 1981-01-09
SE460541B (sv) 1989-10-23
IE49834B1 (en) 1985-12-25
SE447250B (sv) 1986-11-03
AU9187782A (en) 1983-04-21
IL60245A (en) 1985-08-30
GB2051821A (en) 1981-01-21
AU559278B2 (en) 1987-03-05
NO801855L (no) 1980-12-22
SE8500878D0 (sv) 1985-02-22

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