PH17719A - 1,4,9,10-tetrahydro-pyrazolo(4,3-e)pyrido(3,2-b)1,4-diazepin-10-ones - Google Patents

1,4,9,10-tetrahydro-pyrazolo(4,3-e)pyrido(3,2-b)1,4-diazepin-10-ones

Info

Publication number
PH17719A
PH17719A PH27402A PH27402A PH17719A PH 17719 A PH17719 A PH 17719A PH 27402 A PH27402 A PH 27402A PH 27402 A PH27402 A PH 27402A PH 17719 A PH17719 A PH 17719A
Authority
PH
Philippines
Prior art keywords
diazepin
pyrazolo
pyrido
tetrahydro
ones
Prior art date
Application number
PH27402A
Other languages
English (en)
Inventor
Gunther Schmidt
Wolfhard Engel
Wolfgang Eberlein
Gunter Engelhardt
Gunter Trummlitz
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of PH17719A publication Critical patent/PH17719A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PH27402A 1981-06-06 1982-06-04 1,4,9,10-tetrahydro-pyrazolo(4,3-e)pyrido(3,2-b)1,4-diazepin-10-ones PH17719A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813122670 DE3122670A1 (de) 1981-06-06 1981-06-06 "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen"

Publications (1)

Publication Number Publication Date
PH17719A true PH17719A (en) 1984-11-21

Family

ID=6134176

Family Applications (1)

Application Number Title Priority Date Filing Date
PH27402A PH17719A (en) 1981-06-06 1982-06-04 1,4,9,10-tetrahydro-pyrazolo(4,3-e)pyrido(3,2-b)1,4-diazepin-10-ones

Country Status (27)

Country Link
US (1) US4381303A (cs)
EP (1) EP0066774B1 (cs)
JP (1) JPS57212182A (cs)
KR (1) KR880001719B1 (cs)
AR (1) AR229124A1 (cs)
AT (1) ATE10744T1 (cs)
AU (1) AU552765B2 (cs)
CA (1) CA1167440A (cs)
CS (1) CS226743B2 (cs)
DD (1) DD202574A5 (cs)
DE (2) DE3122670A1 (cs)
DK (1) DK253382A (cs)
ES (1) ES512846A0 (cs)
FI (1) FI71560C (cs)
GB (1) GB2117755B (cs)
GR (1) GR76438B (cs)
HU (1) HU186067B (cs)
IE (1) IE53067B1 (cs)
IL (1) IL65977A (cs)
NO (1) NO158063C (cs)
NZ (1) NZ200859A (cs)
PH (1) PH17719A (cs)
PL (1) PL135845B1 (cs)
PT (1) PT75016B (cs)
SU (1) SU1103795A3 (cs)
YU (1) YU118282A (cs)
ZA (1) ZA823919B (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4749788A (en) * 1987-04-13 1988-06-07 A. H. Robins Company, Incorporated Process for the preparation of aryl-pyrido(1,4) benzodiazepines
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
DE69007891T2 (de) * 1989-06-28 1994-08-25 Boehringer Ingelheim Pharma 5,11-Dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one und -thione und ihre Verwendung bei der AIDS-Vorbeugung oder -Behandlung.
CA2052946A1 (en) * 1990-10-19 1992-04-20 Karl G. Grozinger Method for the preparation of 5,11-dihydro-6h-dipyrido ¬3,2-b:2', 3'-e| ¬1,4|diazepines
ATE177099T1 (de) * 1993-12-29 1999-03-15 Pfizer Diazabicyclische neurokinin antagonisten
CN1043347C (zh) * 1994-02-18 1999-05-12 贝林格尔·英格海姆药物公司 2－杂芳基－5,11－二氢－6H－二吡啶并[3,2－b:2’,3’－e][1,4]二氮杂及其在预防或治疗HIV感染中的应用
ES2137113B1 (es) 1997-07-29 2000-09-16 Almirall Prodesfarma Sa Nuevos derivados de triazolo-piridazinas heterociclicos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3450694A (en) * 1966-02-23 1969-06-17 Abbott Lab Substituted benzoxazepines and benzothiazepines
DE2707269A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
CA1154762A (en) * 1979-08-03 1983-10-04 Georg Rainer Substituted tetraazatricyclic compounds, a process for their preparation, their use and medicaments containing them

Also Published As

Publication number Publication date
ES8304571A1 (es) 1983-03-01
DE3122670A1 (de) 1982-12-23
HU186067B (en) 1985-05-28
IL65977A (en) 1984-12-31
AU8460582A (en) 1982-12-16
NO158063C (no) 1988-07-06
PL135845B1 (en) 1985-12-31
EP0066774B1 (de) 1984-12-12
ES512846A0 (es) 1983-03-01
EP0066774A1 (de) 1982-12-15
GB2117755B (en) 1985-01-30
ATE10744T1 (de) 1984-12-15
AU552765B2 (en) 1986-06-19
JPS57212182A (en) 1982-12-27
CA1167440A (en) 1984-05-15
DD202574A5 (de) 1983-09-21
PT75016B (de) 1985-05-17
CS226743B2 (en) 1984-04-16
FI71560B (fi) 1986-10-10
IE821350L (en) 1982-12-06
SU1103795A3 (ru) 1984-07-15
FI821992A0 (fi) 1982-06-04
IE53067B1 (en) 1988-05-25
PT75016A (de) 1982-07-01
ZA823919B (en) 1984-02-29
PL236742A1 (en) 1984-03-26
DE3261530D1 (en) 1985-01-24
IL65977A0 (en) 1982-09-30
GR76438B (cs) 1984-08-10
FI71560C (fi) 1987-01-19
NZ200859A (en) 1985-08-16
US4381303A (en) 1983-04-26
KR840000543A (ko) 1984-02-25
KR880001719B1 (ko) 1988-09-08
YU118282A (en) 1986-04-30
GB2117755A (en) 1983-10-19
DK253382A (da) 1982-12-07
NO821882L (no) 1982-12-07
AR229124A1 (es) 1983-06-15
NO158063B (no) 1988-03-28

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