PH12015502280A1 - Transdermal delivery system comprising donepezil or its salt - Google Patents
Transdermal delivery system comprising donepezil or its saltInfo
- Publication number
- PH12015502280A1 PH12015502280A1 PH12015502280A PH12015502280A PH12015502280A1 PH 12015502280 A1 PH12015502280 A1 PH 12015502280A1 PH 12015502280 A PH12015502280 A PH 12015502280A PH 12015502280 A PH12015502280 A PH 12015502280A PH 12015502280 A1 PH12015502280 A1 PH 12015502280A1
- Authority
- PH
- Philippines
- Prior art keywords
- molecular weight
- donepezil
- weight
- drug
- delivery system
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20140007556A KR101485822B1 (ko) | 2014-01-22 | 2014-01-22 | 도네페질 또는 그의 염을 함유하는 경피흡수제제 |
PCT/KR2015/000277 WO2015111862A1 (fr) | 2014-01-22 | 2015-01-12 | Système d'administration transdermique comprenant du donépézil ou un sel de ce dernier |
Publications (2)
Publication Number | Publication Date |
---|---|
PH12015502280A1 true PH12015502280A1 (en) | 2016-02-01 |
PH12015502280B1 PH12015502280B1 (en) | 2016-02-01 |
Family
ID=52592456
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PH12015502280A PH12015502280B1 (en) | 2014-01-22 | 2015-09-30 | Transdermal delivery system comprising donepezil or its salt |
Country Status (11)
Country | Link |
---|---|
US (1) | US9931307B2 (fr) |
EP (1) | EP3096745B1 (fr) |
JP (1) | JP6405391B2 (fr) |
KR (1) | KR101485822B1 (fr) |
CN (1) | CN105025890B (fr) |
AU (1) | AU2015209915B2 (fr) |
BR (1) | BR112015024271B1 (fr) |
CA (1) | CA2908340C (fr) |
ES (1) | ES2874508T3 (fr) |
PH (1) | PH12015502280B1 (fr) |
WO (1) | WO2015111862A1 (fr) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN108778272A (zh) * | 2015-12-10 | 2018-11-09 | Km特兰斯达股份有限公司 | 经皮吸收制剂 |
IL303255A (en) | 2015-12-30 | 2023-07-01 | Corium Inc | Systems and methods for long-term percutaneous administration |
EP3474831A1 (fr) | 2016-06-23 | 2019-05-01 | Corium International, Inc. | Matrice adhésive à un domaine hydrophile, un domaine hydrophobes et un agent thérapeutique |
CN109789106B (zh) | 2016-07-27 | 2023-06-27 | 考里安有限责任公司 | 碳酸氢钠原位转化驱动胺药物的透皮递送 |
KR102424270B1 (ko) | 2016-07-27 | 2022-07-25 | 코리움, 인크. | 경구 전달과 생물학적으로 동등한 약물동역학을 가진 경피 전달 시스템 |
SG11201900712SA (en) | 2016-07-27 | 2019-02-27 | Corium Int Inc | Memantine transdermal delivery systems |
WO2019126531A1 (fr) | 2017-12-20 | 2019-06-27 | Corium, Inc. | Composition adhésive transdermique comprenant un agent thérapeutique liquide volatil à bas point de fusion |
KR102024996B1 (ko) | 2017-12-27 | 2019-09-25 | 동아에스티 주식회사 | 도네페질을 함유하는 치매 치료용 경피흡수제제 |
KR102372630B1 (ko) | 2019-05-15 | 2022-03-14 | 주식회사 대웅제약 | 고함량의 도네페질 또는 그의 염을 포함하는 경피흡수제제 |
KR102218593B1 (ko) * | 2020-05-13 | 2021-02-22 | 동아에스티 주식회사 | 안정성이 향상된 도네페질 함유 경피 흡수제제 |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6193993B1 (en) | 1998-03-03 | 2001-02-27 | Eisai Co., Ltd. | Suppository containing an antidementia medicament |
KR100342388B1 (ko) * | 1999-11-03 | 2002-07-04 | 김충섭 | 경피 투과용 약물 전달 시스템 |
JP4394443B2 (ja) | 2001-10-17 | 2010-01-06 | 久光製薬株式会社 | 経皮吸収型製剤 |
KR100623077B1 (ko) * | 2002-08-26 | 2006-09-18 | 지상철 | 에스(+)-이부프로펜을 함유하는 경피투여용 조성물 및이를 함유하는 경피투여용 패취제 |
KR100682729B1 (ko) * | 2004-06-15 | 2007-02-15 | (주)아모레퍼시픽 | 신규 경피흡수제제 및 그 제조방법 |
EP2316437B1 (fr) * | 2005-05-13 | 2014-07-30 | Alza Corporation | Système d'administration de médicaments multicouche avec protection contre le flux de matériaux du réservoir |
JP5097359B2 (ja) * | 2006-05-09 | 2012-12-12 | 久光製薬株式会社 | ドネペジル経皮吸収型製剤 |
US9248104B2 (en) * | 2006-08-17 | 2016-02-02 | Core Tech Solutions, Inc. | Transdermal methods and systems for treating Alzheimer's disease |
KR101454362B1 (ko) | 2008-03-24 | 2014-10-23 | 아이큐어 주식회사 | 도네페질을 유효성분으로 함유하는 치매 치료용경피흡수제제 |
EP2328582A4 (fr) | 2008-09-30 | 2012-02-22 | Teikoku Pharma Usa Inc | Compositions de donépézil à administration transdermique étendue et leurs procédés d'utilisation |
EP2399607B1 (fr) | 2009-02-18 | 2017-11-29 | Hisamitsu Pharmaceutical Co., Inc. | Préparation transdermique |
KR101325104B1 (ko) | 2009-09-16 | 2013-11-07 | 주식회사 삼양바이오팜 | 경피 투여 제형 및 그 제조 방법 |
BR112012011334A2 (pt) * | 2009-10-21 | 2020-08-25 | Teikoku Seiyaku Co., Ltd. | formulação transdermicamente absorvível contendo donepezil |
JP5766475B2 (ja) | 2010-03-30 | 2015-08-19 | 日東電工株式会社 | 貼付製剤およびその製造方法 |
KR101292768B1 (ko) * | 2010-04-23 | 2013-08-05 | 아이큐어 주식회사 | 경피 흡수 제제 |
TWI433904B (zh) * | 2011-01-12 | 2014-04-11 | Taiwan Biotech Co Ltd | 多奈哌齊經皮貼片 |
KR101239150B1 (ko) * | 2012-02-28 | 2013-03-06 | 에스케이케미칼주식회사 | 도네페질-함유 경피흡수제제 및 그의 제조방법 |
CN102895217A (zh) * | 2012-11-13 | 2013-01-30 | 沈阳药科大学 | 长效多奈哌齐经皮吸收贴剂 |
-
2014
- 2014-01-22 KR KR20140007556A patent/KR101485822B1/ko active IP Right Grant
-
2015
- 2015-01-12 AU AU2015209915A patent/AU2015209915B2/en not_active Ceased
- 2015-01-12 JP JP2016566588A patent/JP6405391B2/ja active Active
- 2015-01-12 WO PCT/KR2015/000277 patent/WO2015111862A1/fr active Application Filing
- 2015-01-12 BR BR112015024271-5A patent/BR112015024271B1/pt active IP Right Grant
- 2015-01-12 EP EP15739978.3A patent/EP3096745B1/fr active Active
- 2015-01-12 US US14/779,649 patent/US9931307B2/en active Active
- 2015-01-12 ES ES15739978T patent/ES2874508T3/es active Active
- 2015-01-12 CN CN201580000338.XA patent/CN105025890B/zh active Active
- 2015-01-12 CA CA2908340A patent/CA2908340C/fr active Active
- 2015-09-30 PH PH12015502280A patent/PH12015502280B1/en unknown
Also Published As
Publication number | Publication date |
---|---|
AU2015209915A1 (en) | 2015-08-27 |
KR101485822B1 (ko) | 2015-01-23 |
EP3096745A4 (fr) | 2017-08-02 |
WO2015111862A1 (fr) | 2015-07-30 |
ES2874508T3 (es) | 2021-11-05 |
CA2908340A1 (fr) | 2015-07-30 |
BR112015024271B1 (pt) | 2023-10-31 |
BR112015024271A2 (pt) | 2017-07-18 |
JP6405391B2 (ja) | 2018-10-17 |
CA2908340C (fr) | 2021-11-30 |
US20160051486A1 (en) | 2016-02-25 |
EP3096745B1 (fr) | 2021-05-12 |
PH12015502280B1 (en) | 2016-02-01 |
CN105025890A (zh) | 2015-11-04 |
AU2015209915B2 (en) | 2019-09-12 |
CN105025890B (zh) | 2020-03-10 |
JP2017503865A (ja) | 2017-02-02 |
EP3096745A1 (fr) | 2016-11-30 |
US9931307B2 (en) | 2018-04-03 |
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