PH12014501653A1 - Metalloenzyme inhibitor compounds - Google Patents

Metalloenzyme inhibitor compounds

Info

Publication number
PH12014501653A1
PH12014501653A1 PH12014501653A PH12014501653A PH12014501653A1 PH 12014501653 A1 PH12014501653 A1 PH 12014501653A1 PH 12014501653 A PH12014501653 A PH 12014501653A PH 12014501653 A PH12014501653 A PH 12014501653A PH 12014501653 A1 PH12014501653 A1 PH 12014501653A1
Authority
PH
Philippines
Prior art keywords
inhibitor compounds
metalloenzyme inhibitor
metalloenzyme
compounds
present disclosure
Prior art date
Application number
PH12014501653A
Other languages
English (en)
Inventor
William J Hoekstra
Robert J Schotzinger
Stephen W Rafferty
Original Assignee
Viamet Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Viamet Pharmaceuticals Inc filed Critical Viamet Pharmaceuticals Inc
Publication of PH12014501653A1 publication Critical patent/PH12014501653A1/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/713—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
    • A01N57/16—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing heterocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catching Or Destruction (AREA)
  • Preventing Corrosion Or Incrustation Of Metals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PH12014501653A 2012-01-20 2014-07-18 Metalloenzyme inhibitor compounds PH12014501653A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261589064P 2012-01-20 2012-01-20
PCT/US2013/022317 WO2013110002A1 (en) 2012-01-20 2013-01-18 Metalloenzyme inhibitor compounds

Publications (1)

Publication Number Publication Date
PH12014501653A1 true PH12014501653A1 (en) 2014-10-13

Family

ID=48799720

Family Applications (1)

Application Number Title Priority Date Filing Date
PH12014501653A PH12014501653A1 (en) 2012-01-20 2014-07-18 Metalloenzyme inhibitor compounds

Country Status (17)

Country Link
US (1) US9414596B2 (en, 2012)
EP (1) EP2804479A4 (en, 2012)
JP (3) JP2015505538A (en, 2012)
KR (1) KR20140116515A (en, 2012)
CN (1) CN104135861A (en, 2012)
AU (1) AU2013209520A1 (en, 2012)
BR (1) BR112014017799A8 (en, 2012)
CA (1) CA2861341A1 (en, 2012)
CL (1) CL2014001892A1 (en, 2012)
CO (1) CO7111289A2 (en, 2012)
CR (1) CR20140387A (en, 2012)
EA (1) EA201491386A1 (en, 2012)
EC (1) ECSP14014530A (en, 2012)
IN (1) IN2014DN06812A (en, 2012)
MX (1) MX2014008729A (en, 2012)
PH (1) PH12014501653A1 (en, 2012)
WO (1) WO2013110002A1 (en, 2012)

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KR20180069123A (ko) 2009-10-07 2018-06-22 다우 아그로사이언시즈 엘엘씨 곡물에서 진균 방제를 위한 상승작용적 살진균성 혼합물
EA025266B1 (ru) 2011-06-23 2016-12-30 Ваймет Фармасьютикалс, Инк. Соединения, ингибирующие металлоферменты
CN104136427B (zh) * 2012-01-20 2017-03-01 威尔金制药有限公司 金属酶抑制剂化合物
EP2938191B1 (en) 2012-12-28 2018-01-31 Dow AgroSciences LLC Synergistic fungicidal mixtures for fungal control in cereals
DK2938190T3 (en) 2012-12-31 2018-02-05 Dow Agrosciences Llc MACROCYCLIC PICOLINAMIDS AS FUNGICIDES
CN106028815A (zh) 2013-12-26 2016-10-12 美国陶氏益农公司 作为杀真菌剂的大环吡啶酰胺
WO2015100181A1 (en) 2013-12-26 2015-07-02 Dow Agrosciences Llc Macrocyclic picolinamide compounds with fungicidal activity
JP6606508B2 (ja) 2014-03-19 2019-11-13 マイコヴィア ファーマシューティカルズ，インコーポレイテッド 抗真菌化合物の調製方法
EP3119753B1 (en) * 2014-03-19 2020-11-04 Dow AgroSciences LLC 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1h-tetrazol-1-yl)propan-2-ols and processes for their preparation
JP2017507991A (ja) * 2014-03-19 2017-03-23 ヴィアメット ファーマスーティカルズ，インコーポレイテッド 抗真菌化合物の調製方法
EP3119755B1 (en) * 2014-03-19 2019-03-06 Viamet Pharmaceuticals (NC), Inc. Antifungal compound process
CA2942932A1 (en) * 2014-03-19 2015-09-24 Viamet Pharmaceuticals, Inc. Antifungal compound process
CA2942231A1 (en) 2014-03-19 2015-09-24 Viamet Pharmaceuticals, Inc. Antifungal compound process
CA2942982C (en) * 2014-03-19 2023-09-19 Viamet Pharmaceuticals, Inc. 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1h-tetrazol-1-yl)propan-2-ols and processes for their preparation
EA037587B1 (ru) * 2014-03-19 2021-04-19 Майковиа Фармасьютикалс, Инк. Способ получения противогрибковых соединений
CA2942927A1 (en) * 2014-03-19 2015-09-24 Viamet Pharmaceuticals, Inc. Antifungal compound process
CA2942976C (en) * 2014-03-19 2022-05-10 Viamet Pharmaceuticals, Inc. Antifungal compound process
CA2945674A1 (en) * 2014-04-15 2015-10-22 Dow Agrosciences Llc Metalloenzyme inhibitor compounds as fungicides
US9663491B2 (en) 2014-04-15 2017-05-30 Dow Agrosciences Llc Metalloenzyme inhibitor compounds as fungicides
WO2015171408A1 (en) 2014-05-06 2015-11-12 Dow Agrosciences Llc Macrocyclic picolinamides as fungicides
BR112017000169A2 (pt) 2014-07-08 2017-10-31 Dow Agrosciences Llc picolinamidas macrocíclicas como fungicidas
US9686984B2 (en) 2014-07-08 2017-06-27 Dow Agrosciences Llc Macrocyclic picolinamides as fungicides
WO2016109302A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
CN107205386B (zh) 2014-12-30 2021-07-23 美国陶氏益农公司 具有杀真菌活性的吡啶酰胺
CA2972413A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
PT3240773T (pt) * 2014-12-30 2020-09-10 Dow Agrosciences Llc Compostos picolinamida com atividade fungicida
DK3240415T3 (da) 2014-12-30 2022-10-03 Corteva Agriscience Llc Fungicide sammensætninger
US20180002288A1 (en) 2014-12-30 2018-01-04 Dow Agrosciences Llc Use of picolinamides as fungicides
BR112017018823A2 (pt) 2015-03-19 2018-04-24 Viamet Pharmaceuticals, Inc. compostos antifúngicos e processos para a fabricação
BR112018005198A2 (pt) 2015-09-18 2018-10-09 Vps-3, Inc. compostos antifúngicos e processos de manufatura
CN108779094B (zh) * 2015-12-30 2021-11-16 Nqp 1598公司 金属酶抑制剂化合物
WO2018044996A1 (en) 2016-08-30 2018-03-08 Dow Agrosciences Llc Picolinamides as fungicides
WO2018044991A1 (en) 2016-08-30 2018-03-08 Dow Agrosciences Llc Thiopicolinamide compounds with fungicidal activity
WO2018045012A1 (en) 2016-08-30 2018-03-08 Dow Agrosciences Llc Pyrido-1,3-oxazine-2,4-dione compounds with fungicidal activity
US10111432B2 (en) 2016-08-30 2018-10-30 Dow Agrosciences Llc Picolinamide N-oxide compounds with fungicidal activity
BR102018000183B1 (pt) 2017-01-05 2023-04-25 Dow Agrosciences Llc Picolinamidas, composição para controle de um patógeno fúngico, e método para controle e prevenção de um ataque por fungos em uma planta
WO2018145934A1 (en) * 2017-02-08 2018-08-16 Bayer Cropscience Aktiengesellschaft Novel triazole derivatives
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN110996665B (zh) 2017-05-02 2021-10-26 陶氏益农公司 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
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CN110981810A (zh) * 2019-12-19 2020-04-10 东莞市维琪科技有限公司 一种脱羧肌肽的合成方法
WO2021143811A1 (zh) * 2020-01-17 2021-07-22 上海森辉医药有限公司 四氮唑类化合物的可药用盐及其结晶形式、制备方法和用途

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Also Published As

Publication number Publication date
ECSP14014530A (es) 2015-06-30
IN2014DN06812A (en, 2012) 2015-05-22
EP2804479A4 (en) 2015-07-22
US9414596B2 (en) 2016-08-16
AU2013209520A1 (en) 2014-08-28
CL2014001892A1 (es) 2014-11-14
BR112014017799A2 (en, 2012) 2017-06-20
JP2015505538A (ja) 2015-02-23
MX2014008729A (es) 2015-02-04
EA201491386A1 (ru) 2014-11-28
EP2804479A1 (en) 2014-11-26
CA2861341A1 (en) 2013-07-25
US20150024938A1 (en) 2015-01-22
JP2019116476A (ja) 2019-07-18
WO2013110002A1 (en) 2013-07-25
BR112014017799A8 (pt) 2017-07-11
JP2017110004A (ja) 2017-06-22
CN104135861A (zh) 2014-11-05
CR20140387A (es) 2014-11-27
CO7111289A2 (es) 2014-11-10
KR20140116515A (ko) 2014-10-02

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