PE20220427A1 - Compuestos triciclicos - Google Patents

Compuestos triciclicos

Info

Publication number
PE20220427A1
PE20220427A1 PE2021001952A PE2021001952A PE20220427A1 PE 20220427 A1 PE20220427 A1 PE 20220427A1 PE 2021001952 A PE2021001952 A PE 2021001952A PE 2021001952 A PE2021001952 A PE 2021001952A PE 20220427 A1 PE20220427 A1 PE 20220427A1
Authority
PE
Peru
Prior art keywords
options
alkyl
haloalkyl
hepatitis
aryl
Prior art date
Application number
PE2021001952A
Other languages
English (en)
Spanish (es)
Inventor
Sandrine Vendeville
Original Assignee
Aligos Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aligos Therapeutics Inc filed Critical Aligos Therapeutics Inc
Publication of PE20220427A1 publication Critical patent/PE20220427A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PE2021001952A 2019-05-30 2020-05-27 Compuestos triciclicos PE20220427A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962854597P 2019-05-30 2019-05-30
PCT/US2020/034746 WO2020243199A1 (en) 2019-05-30 2020-05-27 Tricyclic compounds

Publications (1)

Publication Number Publication Date
PE20220427A1 true PE20220427A1 (es) 2022-03-29

Family

ID=73552666

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2021001952A PE20220427A1 (es) 2019-05-30 2020-05-27 Compuestos triciclicos

Country Status (19)

Country Link
US (1) US11136321B2 (enExample)
EP (1) EP3976618A4 (enExample)
JP (1) JP2022534501A (enExample)
KR (1) KR20220016177A (enExample)
CN (1) CN113906029A (enExample)
AU (1) AU2020282707B2 (enExample)
BR (1) BR112021023967A2 (enExample)
CA (1) CA3138938A1 (enExample)
CL (1) CL2021003139A1 (enExample)
CO (1) CO2021017202A2 (enExample)
EA (1) EA202192760A1 (enExample)
IL (1) IL287813A (enExample)
MA (1) MA56058A (enExample)
MX (1) MX2021014458A (enExample)
PE (1) PE20220427A1 (enExample)
PH (1) PH12021552953A1 (enExample)
SG (1) SG11202113214QA (enExample)
TW (1) TW202110845A (enExample)
WO (1) WO2020243199A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20220000874A1 (en) * 2019-05-30 2022-01-06 Aligos Therapeutics, Inc. Tricyclic compounds
CN114222746B (zh) * 2019-12-10 2024-08-02 上海翰森生物医药科技有限公司 含吡唑多环类衍生物抑制剂、其制备方法和应用
GB202103704D0 (en) * 2021-03-17 2021-04-28 Pathios Therapeutics Ltd Compounds
EP4251625A4 (en) * 2020-11-24 2024-10-09 Aligos Therapeutics, Inc. Tricyclic compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0701273D0 (en) 2007-01-24 2007-02-28 Angeletti P Ist Richerche Bio New compounds
WO2008157273A1 (en) 2007-06-14 2008-12-24 Smithkline Beecham Corporation Chemical compounds
WO2015065338A1 (en) 2013-10-29 2015-05-07 Medivir Ab Quinazoline based respiratory syncytial virus inhibitors
AU2017231817B2 (en) 2016-03-09 2021-02-25 Emory University Elimination of hepatitis B virus with antiviral agents
CN110066278B (zh) * 2017-06-01 2021-06-08 广东东阳光药业有限公司 稠合三环类化合物及其在药物中的应用

Also Published As

Publication number Publication date
TW202110845A (zh) 2021-03-16
WO2020243199A1 (en) 2020-12-03
US11136321B2 (en) 2021-10-05
IL287813A (en) 2022-01-01
KR20220016177A (ko) 2022-02-08
MA56058A (fr) 2022-04-06
BR112021023967A2 (pt) 2022-03-08
PH12021552953A1 (en) 2022-07-25
SG11202113214QA (en) 2021-12-30
AU2020282707A1 (en) 2021-12-02
EA202192760A1 (ru) 2022-03-05
AU2020282707B2 (en) 2025-06-19
CL2021003139A1 (es) 2022-09-23
CO2021017202A2 (es) 2022-01-17
CA3138938A1 (en) 2020-12-03
JP2022534501A (ja) 2022-08-01
EP3976618A4 (en) 2023-01-04
CN113906029A (zh) 2022-01-07
MX2021014458A (es) 2022-01-06
EP3976618A1 (en) 2022-04-06
US20200407361A1 (en) 2020-12-31

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