PE20120325A1 - Aminopirimidinas sustituidas con arilo como agentes fungicidas - Google Patents

Aminopirimidinas sustituidas con arilo como agentes fungicidas

Info

Publication number
PE20120325A1
PE20120325A1 PE2011001972A PE2011001972A PE20120325A1 PE 20120325 A1 PE20120325 A1 PE 20120325A1 PE 2011001972 A PE2011001972 A PE 2011001972A PE 2011001972 A PE2011001972 A PE 2011001972A PE 20120325 A1 PE20120325 A1 PE 20120325A1
Authority
PE
Peru
Prior art keywords
aminopyrimidines
aryl
substituted
fungicide
compounds
Prior art date
Application number
PE2011001972A
Other languages
English (en)
Inventor
George Davis
William Lo
James Renga
Francis Tisdell
Maurice Yap
David Young
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PE20120325A1 publication Critical patent/PE20120325A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

SE REFIERE A COMPUESTOS DERIVADOS DE AMINOPIRIMIDINAS DE FORMULA (1) DONDE X1 ES N O C-R3; X2 ES N O C-R4 CON LA CONDICION DE QUE X1 Y X2 NO SEAN AMBOS N; R1 A R7 SON CADA UNO H, CN, CHO, F, ALQUILO(C1-C4), ALCOXI(C1-C4), ENTRE OTROS, OPCIONALMENTE SUSTITUIDOS CON F, OH, CN, NO2, ENTRE OTROS; Q ES ARILO O HETEROCICLO OPCIONALMENTE SUSTITUIDO CON R1 A R7. SON COMPUESTOS PREFERIDOS LOS DE FORMULA (i), (ii), ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FUNGICIDA QUE ADEMAS PUEDE CONTENER UN INSECTICIDA, HERBICIDA O FUNGICIDA. DICHOS COMPUESTOS SON UTILES PARA CONTROLAR HONGOS PATOGENOS EN PLANTAS
PE2011001972A 2009-05-19 2010-05-03 Aminopirimidinas sustituidas con arilo como agentes fungicidas PE20120325A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17940209P 2009-05-19 2009-05-19

Publications (1)

Publication Number Publication Date
PE20120325A1 true PE20120325A1 (es) 2012-04-12

Family

ID=42315653

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2011001972A PE20120325A1 (es) 2009-05-19 2010-05-03 Aminopirimidinas sustituidas con arilo como agentes fungicidas

Country Status (24)

Country Link
US (2) US8759356B2 (es)
EP (1) EP2432767B1 (es)
JP (1) JP2012527461A (es)
KR (1) KR20120016247A (es)
CN (1) CN102438993A (es)
AU (1) AU2010250017B2 (es)
BR (1) BRPI1011058A2 (es)
CA (1) CA2760911A1 (es)
CL (1) CL2011002922A1 (es)
CO (1) CO6460778A2 (es)
CR (1) CR20110589A (es)
DK (1) DK2432767T3 (es)
EC (1) ECSP11011467A (es)
ES (1) ES2417355T3 (es)
HN (1) HN2011003040A (es)
MX (1) MX2011012343A (es)
NZ (1) NZ596123A (es)
PE (1) PE20120325A1 (es)
PL (1) PL2432767T3 (es)
PT (1) PT2432767E (es)
RU (1) RU2011151603A (es)
SI (1) SI2432767T1 (es)
TW (1) TW201041512A (es)
WO (1) WO2010135070A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA025183B1 (ru) 2011-09-27 2016-11-30 Новартис Аг 3-пиримидин-4-ил-оксазолидин-2-оны в качестве ингибиторов мутантной idh
UY34632A (es) 2012-02-24 2013-05-31 Novartis Ag Compuestos de oxazolidin- 2- ona y usos de los mismos
US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
US9434719B2 (en) 2013-03-14 2016-09-06 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH

Family Cites Families (64)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1345640A (en) * 1971-02-01 1974-01-30 Shell Int Research Piperazinyl pyrimidines
JPS6052146B2 (ja) 1979-12-25 1985-11-18 石原産業株式会社 Ｎ−ピリジルアニリン系化合物、それらの製造方法及びそれらを含有する有害生物防除剤
FR2503162A1 (fr) * 1981-04-07 1982-10-08 Pharmindustrie Nouveaux derives de piperazino-2 pyrimidine, procedes pour leur preparation et leur utilisation comme medicaments ou comme intermediaires pour la fabrication de medicaments
ZA85853B (en) * 1984-02-17 1986-09-24 Warner Lambert Co Antibacterial agents
US4791110A (en) * 1985-06-14 1988-12-13 Eli Lilly And Company Fungicidal pyridazines
DE3922735A1 (de) * 1989-07-11 1991-01-24 Hoechst Ag Aminopyrimidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
US5792778A (en) * 1995-08-10 1998-08-11 Merck & Co., Inc. 2-substituted aryl pyrroles, compositions containing such compounds and methods of use
US5958934A (en) * 1996-05-23 1999-09-28 Syntex (U.S.A.) Inc. Aryl pyrimidine derivatives and uses thereof
TW440563B (en) * 1996-05-23 2001-06-16 Hoffmann La Roche Aryl pyrimidine derivatives and a pharmaceutical composition thereof
AU708883B2 (en) * 1996-06-10 1999-08-12 Merck & Co., Inc. Substituted imidazoles having cytokine inhibitory activity
US6979686B1 (en) * 2001-12-07 2005-12-27 Pharmacia Corporation Substituted pyrazoles as p38 kinase inhibitors
US6514977B1 (en) * 1997-05-22 2003-02-04 G.D. Searle & Company Substituted pyrazoles as p38 kinase inhibitors
EP0988301B1 (en) * 1997-06-12 2006-08-09 Aventis Pharma Limited Imidazolyl-cyclic acetals
US6331538B1 (en) * 1997-10-28 2001-12-18 Warner-Lambert Company 7-substituted quinazolin-2,4-diones useful as antibacterial agents
CO5170501A1 (es) * 1999-04-14 2002-06-27 Novartis Ag AZOLES SUSTITUIDOS UTILES PARA EL TRATAMIENTO DE ENFERMEDADES MEDIADAS POR TNFa eIL-1 Y ENFERMEDADES DEL METABOLISMO OSEO
CO5210940A1 (es) * 1999-05-04 2002-10-30 Novartis Ag Compuestos plaguicidas derivados de pirimidina y composiciones que los contienen
WO2001030778A1 (en) * 1999-10-27 2001-05-03 Novartis Ag Thiazole and imidazo [4,5-b] pyridine compounds and their pharmaceutical use
GB9927844D0 (en) * 1999-11-26 2000-01-26 Glaxo Group Ltd Chemical compounds
EP1289523A1 (en) * 2000-06-01 2003-03-12 Merck & Co., Inc. Use of (di-substituted-phenyl)-pyrimidinyl-imidazole derivatives as jnk-inhibitors
PE20020506A1 (es) * 2000-08-22 2002-07-09 Glaxo Group Ltd Derivados de pirazol fusionados como inhibidores de la proteina cinasa
DE60201074T2 (de) * 2001-03-08 2005-09-15 Smithkline Beecham Corp. Pyrazolopyridinderivate
JP2004525150A (ja) * 2001-03-30 2004-08-19 スミスクライン ビーチャム コーポレーション 治療用化合物としてのピラゾロピリジン類の使用
JP4237497B2 (ja) * 2001-03-30 2009-03-11 スミスクライン ビーチャム コーポレーション ピラゾロピリジン類、その調製方法及びその治療用化合物としての使用
WO2003000682A1 (en) * 2001-06-25 2003-01-03 Merck & Co., Inc. (pyrimidyl)(phenyl)substituted fused heteroaryl p38 inhibiting and pkg kinase inhibiting compounds
WO2003026661A1 (fr) * 2001-09-14 2003-04-03 Yamanouchi Pharmaceutical Co., Ltd. Accelerateur de secretion de l'insuline et nouveau derive de pyrimidine
US6566357B1 (en) * 2001-09-20 2003-05-20 The Procter & Gamble Co. Spirocyclic-6,7-dihydro-5H-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
US6730668B2 (en) * 2001-09-20 2004-05-04 The Procter & Gamble Company 6,7-dihydro-5H-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
PL375447A1 (en) * 2002-08-14 2005-11-28 Vertex Pharmaceuticals Incorporated Protein kinase inhibitors and uses thereof
MXPA05002036A (es) * 2002-08-21 2005-10-19 Xact Design & Engineering Pty Mecanismo de transmision de torsion.
UA80296C2 (en) * 2002-09-06 2007-09-10 Biogen Inc Imidazolopyridines and methods of making and using the same
JP2006504755A (ja) * 2002-10-15 2006-02-09 スミスクライン ビーチャム コーポレーション Ｇｓｋ−３阻害薬としてのピリダジン化合物
JP4356504B2 (ja) * 2003-04-21 2009-11-04 田辺三菱製薬株式会社 ｐ３８ＭＡＰキナーゼ阻害剤
AU2004247626B8 (en) * 2003-05-15 2011-05-19 Arqule, Inc. Imidazothiazoles and imidazoxazole derivatives as inhibitors of p38
US7566712B2 (en) * 2003-07-16 2009-07-28 Neurogen Corporation Biaryl piperazinyl-pyridine analogues
ES2234433B1 (es) * 2003-12-15 2006-11-01 Almirall Prodesfarma, S.A. 4-aminopirimidinas como antagonistas de receptores de adenosina.
EA010568B1 (ru) * 2003-12-15 2008-10-30 Ньюрокрайн Байосайнсиз Инк. 2,6-бисгетероарил-4-аминопиримидины в качестве антагонистов аденозиновых рецепторов
DE102004010194A1 (de) * 2004-03-02 2005-10-13 Aventis Pharma Deutschland Gmbh 4-Benzimidazol-2-yl-pyridazin-3-on-Derivate, ihre Herstellung und Verwendung in Arzneimitteln
ES2241496B1 (es) * 2004-04-15 2006-12-01 Almirall Prodesfarma, S.A. Nuevos derivados de piridina.
BRPI0512306A (pt) * 2004-06-25 2008-02-26 Basf Ag compostos, processo para a preparação dos mesmos, agente pesticida, e, processos para o combate de fungos nocivos fitopatogênicos e de pragas de animais em agricultura
TW200616974A (en) * 2004-07-01 2006-06-01 Astrazeneca Ab Chemical compounds
AU2005295734A1 (en) * 2004-10-15 2006-04-27 Biogen Idec Ma Inc. Methods of treating vascular injuries
CN101146789A (zh) * 2005-01-25 2008-03-19 阿斯利康(瑞典)有限公司 化合物
WO2006137658A1 (en) * 2005-06-20 2006-12-28 Dongbu Hitek Co., Ltd. New substituted 1,3-thiazole derivatives or pharmaceutically acceptable salts thereof having immunosuppression and inflammation inhibitory acitivity, intermediate compounds or pharmaceutically acceptable salts thereof, a process for the preparation thereof, and pharmaceutical composition comprising the same
CA2620223A1 (en) * 2005-09-02 2007-03-08 Abbott Laboratories Novel imidazo based heterocycles
US20080004271A1 (en) * 2006-01-17 2008-01-03 Mckenna Jeffrey M Inhibitors of TNFalpha, PDE4 and B-RAF, compositions thereof and methods of use therewith
WO2007083692A1 (ja) * 2006-01-23 2007-07-26 Kumiai Chemical Industry Co., Ltd. アミノピリミジン誘導体及び農園芸用植物病害防除剤
WO2007146087A2 (en) * 2006-06-06 2007-12-21 Avigen, Inc. SUBSTITUTED PYRAZOLO [1,5-α] PYRIDINE COMPOUNDS AND THEIR METHODS OF USE
US7870698B2 (en) * 2006-06-27 2011-01-18 United States Gypsum Company Non-combustible reinforced cementitious lightweight panels and metal frame system for building foundations
TW200838517A (en) * 2006-12-21 2008-10-01 Vertex Pharma Compounds useful as protein kinases inhibitors
TW200835487A (en) * 2006-12-28 2008-09-01 Basf Ag 2-substituted pyridines I in therapy
DE102007010801A1 (de) * 2007-03-02 2008-09-04 Bayer Cropscience Ag Diaminopyrimidine als Fungizide
US8603081B2 (en) * 2007-08-23 2013-12-10 Ntk Enterprises, Inc. System and method for defining and controlling LTK and other surgical eye procedures to produce little or no stromal collagen shrinkage
WO2009029793A1 (en) * 2007-08-31 2009-03-05 Martek Biosciences Corporation Polyunsaturated fatty acid-containing solid fat compositions and uses and production thereof
DE102007044388B4 (de) * 2007-09-18 2012-08-02 Airbus Operations Gmbh Druckschott und Verfahren zum Unterteilen eines Luft- oder Raumfahrzeugs
CN101821813B (zh) * 2007-10-04 2013-11-27 劳伦斯·利弗莫尔国家安全有限责任公司 用于聚变-裂变发动机的固体空芯燃料
CA2707989A1 (en) * 2007-12-07 2009-06-11 Novartis Ag Pyrazole derivatives and use thereof as inhibitors of cyclin dependent kinases
AU2008335151A1 (en) * 2007-12-12 2009-06-18 E. I. Du Pont De Nemours And Company Fungicidal bicyclic pyrazoles
DE102007061756A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte 4-Aminopyrimidin-5-carbonsäuren und ihre Verwendung
GB0725218D0 (en) * 2007-12-24 2008-02-06 Syngenta Ltd Chemical compounds
US8343966B2 (en) * 2008-01-11 2013-01-01 Novartis Ag Organic compounds
DE102008011983B4 (de) * 2008-02-29 2013-11-28 O-Flexx Technologies Gmbh Thermische Solaranlage
CN101965346A (zh) * 2008-03-06 2011-02-02 埃科特莱茵药品有限公司 新颖嘧啶-吡啶衍生物
EP2280948A1 (en) 2008-04-09 2011-02-09 Mitsubishi Tanabe Pharma Corporation Pyrimidine, pyridine and triazine derivatives as maxi-k channel openers.
BRPI0915720A2 (pt) * 2008-06-12 2015-08-04 Janssen Pharmaceutica Nv Moduladores de diaminopiridina, pirimidina, e piridazina do receptor de histamina h4

Also Published As

Publication number Publication date
PL2432767T3 (pl) 2013-11-29
CO6460778A2 (es) 2012-06-15
CL2011002922A1 (es) 2012-04-13
US20100298143A1 (en) 2010-11-25
AU2010250017A1 (en) 2011-11-24
TW201041512A (en) 2010-12-01
PT2432767E (pt) 2013-07-25
AU2010250017B2 (en) 2015-02-12
CR20110589A (es) 2012-03-06
SI2432767T1 (sl) 2013-10-30
KR20120016247A (ko) 2012-02-23
JP2012527461A (ja) 2012-11-08
BRPI1011058A2 (pt) 2015-08-25
ES2417355T3 (es) 2013-08-07
US8759356B2 (en) 2014-06-24
NZ596123A (en) 2014-08-29
EP2432767A1 (en) 2012-03-28
ECSP11011467A (es) 2011-12-30
EP2432767B1 (en) 2013-06-26
US20140275123A1 (en) 2014-09-18
RU2011151603A (ru) 2013-06-27
MX2011012343A (es) 2011-12-14
WO2010135070A1 (en) 2010-11-25
HN2011003040A (es) 2013-10-22
DK2432767T3 (da) 2013-09-30
CA2760911A1 (en) 2010-11-25
CN102438993A (zh) 2012-05-02

Similar Documents

Publication Publication Date Title
PE20140776A1 (es) Composicion fungicida y metodo para controlar enfermedades de las plantas
EA201500386A1 (ru) Пестицидные смеси, содержащие жасмоновую кислоту или её производное
CO6280578A2 (es) Diaminopirimidinas como agentes fitosanitarios
CR9776A (es) Derivados plaguicidas de fenilamidina sustituida con tiazoliloxi
EA201400231A1 (ru) Фунгицидные замещенные 1-{2-[2-галоген-4-(4-галогенфенокси)фенил]-2-алкокси-2-алкинил/алкенилэтил}-1н-[1,2,4]триазольные соединения
UY32212A (es) Piridinas sustituidas con accion herbicida
CL2012000310A1 (es) Compuesto derivado de 5-fluoro pirimidinona; composicion fungicida que comprende a dicho compuesto; y un metodo para el control diferencial de ataque fungico en plantas.
ECSP088596A (es) Compuestos de piperazina con accion herbicida
CR11172A (es) Compuestos de piperazina con accion herbicida
CR9780A (es) Derivados plaguicidas de bifenilamidina
UY31148A1 (es) Compuestos de piperazina con accion herbicida (ii)
CR20120064A (es) Heterociclos microbicidas
UY32313A (es) Composiciones herbicidas que contienen compuestos de benzoilpirazol y otro compuesto herbicida
ECSP088313A (es) Derivados plaguicidas de fenilamidina sustituida con pirimidiniloxi
EA200901329A1 (ru) Применение пиридин-2-окси-3-карбонамидов в качестве защитных средств
UY30895A1 (es) Mezclas fungicidas que comprenden 1-metilipirazol-4-ilcarboxanilidas sustituidas
PE20170443A1 (es) Derivados de heteroarilpiperidina y de piperazina como fungicidas
CR20110043A (es) Mezclas fungicidas que comprenden 1-metilpirazol-4-ilcarboxanilidas sustituidas
AR106257A1 (es) 3-fenilpirrolidina-2,4-dionas sustituidas con alquinilo y su uso como herbicidas
AR058040A1 (es) Derivados plaguicidas de fenilamidina sustituida con feniloxi
ECSP10010726A (es) Composición fungicida y
AR058042A1 (es) Derivados plaguicidas de fenilamidina sustituida con naftiloxi
UY33907A (es) Derivados de pirazol microbicidas
CR20150396A (es) Composiciones herbicidas que comprenden un cornexistin
EA201691626A1 (ru) Фунгицидные композиции алкоксиамидов пиразолкарбоновой кислоты

Legal Events

Date Code Title Description
FG Grant, registration
FD Application declared void or lapsed