PE20020792A1 - Antagonistas de receptores de aminoacidos excitadores - Google Patents

Antagonistas de receptores de aminoacidos excitadores

Info

Publication number
PE20020792A1
PE20020792A1 PE2002000003A PE2002000003A PE20020792A1 PE 20020792 A1 PE20020792 A1 PE 20020792A1 PE 2002000003 A PE2002000003 A PE 2002000003A PE 2002000003 A PE2002000003 A PE 2002000003A PE 20020792 A1 PE20020792 A1 PE 20020792A1
Authority
PE
Peru
Prior art keywords
alkyl
refers
acid
antagonists
amino acid
Prior art date
Application number
PE2002000003A
Other languages
English (en)
Spanish (es)
Inventor
Michael Edward Letourneau
Khau Vien Van
Michael John Martinelli
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PE20020792A1 publication Critical patent/PE20020792A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PE2002000003A 2001-01-05 2002-01-04 Antagonistas de receptores de aminoacidos excitadores PE20020792A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US26001401P 2001-01-05 2001-01-05

Publications (1)

Publication Number Publication Date
PE20020792A1 true PE20020792A1 (es) 2002-09-06

Family

ID=22987455

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2002000003A PE20020792A1 (es) 2001-01-05 2002-01-04 Antagonistas de receptores de aminoacidos excitadores

Country Status (23)

Country Link
EP (1) EP1351955A1 (ja)
JP (1) JP2004520335A (ja)
KR (1) KR20030066797A (ja)
CN (1) CN1484642A (ja)
AR (1) AR035679A1 (ja)
BR (1) BR0116672A (ja)
CA (1) CA2431545A1 (ja)
CZ (1) CZ20031856A3 (ja)
DZ (1) DZ3460A1 (ja)
EA (1) EA200300770A1 (ja)
EC (1) ECSP034682A (ja)
HR (1) HRP20030544A2 (ja)
HU (1) HUP0302528A2 (ja)
IL (1) IL156138A0 (ja)
MX (1) MXPA03005981A (ja)
NO (1) NO20032973D0 (ja)
NZ (1) NZ525821A (ja)
PE (1) PE20020792A1 (ja)
PL (1) PL361934A1 (ja)
SK (1) SK8242003A3 (ja)
TW (1) TW591023B (ja)
WO (1) WO2002053561A1 (ja)
ZA (1) ZA200304311B (ja)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5284957A (en) * 1992-09-03 1994-02-08 Eli Lilly And Company Excitatory amino acid receptor antagonists
JP2002505254A (ja) * 1998-02-06 2002-02-19 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー パロキセチン塩
GB9908175D0 (en) * 1999-04-09 1999-06-02 Lilly Co Eli Method of treating neurological disorders
DE60032905T2 (de) * 1999-07-06 2007-10-18 Eli Lilly And Co., Indianapolis Selektive iglur5 rezeptorantagonisten zur behandlung der migräne

Also Published As

Publication number Publication date
NZ525821A (en) 2004-07-30
MXPA03005981A (es) 2003-09-10
CZ20031856A3 (cs) 2003-09-17
BR0116672A (pt) 2003-09-23
AR035679A1 (es) 2004-06-23
DZ3460A1 (fr) 2002-07-11
EP1351955A1 (en) 2003-10-15
ZA200304311B (en) 2004-09-02
TW591023B (en) 2004-06-11
PL361934A1 (en) 2004-10-18
SK8242003A3 (en) 2004-01-08
CA2431545A1 (en) 2002-07-11
HRP20030544A2 (en) 2004-08-31
HUP0302528A2 (hu) 2003-11-28
WO2002053561A1 (en) 2002-07-11
EA200300770A1 (ru) 2003-10-30
KR20030066797A (ko) 2003-08-09
NO20032973L (no) 2003-06-27
NO20032973D0 (no) 2003-06-27
ECSP034682A (es) 2003-08-29
CN1484642A (zh) 2004-03-24
JP2004520335A (ja) 2004-07-08
IL156138A0 (en) 2003-12-23

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