PA8773901A1 - Procedimiento para la preparación de derivados de epotilona por epoxidación catalítica selectiva - Google Patents

Procedimiento para la preparación de derivados de epotilona por epoxidación catalítica selectiva

Info

Publication number
PA8773901A1
PA8773901A1 PA20088773901A PA8773901A PA8773901A1 PA 8773901 A1 PA8773901 A1 PA 8773901A1 PA 20088773901 A PA20088773901 A PA 20088773901A PA 8773901 A PA8773901 A PA 8773901A PA 8773901 A1 PA8773901 A1 PA 8773901A1
Authority
PA
Panama
Prior art keywords
epotilone
procedure
derivatives
preparation
selective catalytic
Prior art date
Application number
PA20088773901A
Other languages
English (en)
Spanish (es)
Inventor
Platzek Johannes
Petrov Orlin
Pruhs Stephan
Original Assignee
Bayer Shering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Shering Pharma Ag filed Critical Bayer Shering Pharma Ag
Publication of PA8773901A1 publication Critical patent/PA8773901A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PA20088773901A 2007-03-30 2008-03-28 Procedimiento para la preparación de derivados de epotilona por epoxidación catalítica selectiva PA8773901A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102007016046A DE102007016046A1 (de) 2007-03-30 2007-03-30 Verfahren zur Herstellung von Epothilonderivaten durch selektive katalytische Epoxidierung

Publications (1)

Publication Number Publication Date
PA8773901A1 true PA8773901A1 (es) 2008-11-19

Family

ID=39551678

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20088773901A PA8773901A1 (es) 2007-03-30 2008-03-28 Procedimiento para la preparación de derivados de epotilona por epoxidación catalítica selectiva

Country Status (13)

Country Link
US (2) US20080242868A1 (enExample)
EP (1) EP2142539A2 (enExample)
JP (1) JP2010523481A (enExample)
KR (1) KR20090125259A (enExample)
CN (1) CN101652362B (enExample)
AR (1) AR066692A1 (enExample)
CA (1) CA2681806A1 (enExample)
CL (1) CL2008000901A1 (enExample)
DE (1) DE102007016046A1 (enExample)
PA (1) PA8773901A1 (enExample)
TW (1) TW200902538A (enExample)
UY (1) UY30985A1 (enExample)
WO (1) WO2008119563A2 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114539143A (zh) * 2022-01-28 2022-05-27 安徽瑞邦生物科技有限公司 一种4-氰基吡啶的纯化方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69910831T2 (de) * 1998-12-22 2004-07-15 Novartis Ag Epothilonderivate und ihre verwendung als antitumormittel
AR023792A1 (es) 1999-04-30 2002-09-04 Bayer Schering Pharma Ag Derivados 6-alquenilo- y 6-alquinilo-epotilona, los procedimientos para prepararlos y su empleo en productos farmaceuticos
EP1340498A1 (en) * 2002-03-01 2003-09-03 Schering Aktiengesellschaft Use of epothilones in the treatment of brain diseases associated with proliferative processes
GB0405898D0 (en) * 2004-03-16 2004-04-21 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
WO2008119563A2 (de) 2008-10-09
JP2010523481A (ja) 2010-07-15
WO2008119563A3 (de) 2009-02-12
CL2008000901A1 (es) 2008-10-17
UY30985A1 (es) 2008-10-31
DE102007016046A1 (de) 2008-10-23
CN101652362B (zh) 2012-10-10
US8314248B2 (en) 2012-11-20
EP2142539A2 (de) 2010-01-13
AR066692A1 (es) 2009-09-09
US20080242868A1 (en) 2008-10-02
CA2681806A1 (en) 2008-10-09
KR20090125259A (ko) 2009-12-04
TW200902538A (en) 2009-01-16
CN101652362A (zh) 2010-02-17
US20120077984A1 (en) 2012-03-29

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