OA12159A - Monohydrate of cis-lithium-cyano-4-Ä3-(cyclopentyloxy)-4-methoxyphenylÜcyclohexanecar-boxylate. - Google Patents

Monohydrate of cis-lithium-cyano-4-Ä3-(cyclopentyloxy)-4-methoxyphenylÜcyclohexanecar-boxylate. Download PDF

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Publication number
OA12159A
OA12159A OA1200200211A OA1200200211A OA12159A OA 12159 A OA12159 A OA 12159A OA 1200200211 A OA1200200211 A OA 1200200211A OA 1200200211 A OA1200200211 A OA 1200200211A OA 12159 A OA12159 A OA 12159A
Authority
OA
OAPI
Prior art keywords
monohydrate
cyclopentyloxy
cyano
lithium
cis
Prior art date
Application number
OA1200200211A
Other languages
English (en)
Inventor
Kevin Scott Webb
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of OA12159A publication Critical patent/OA12159A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/45Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C255/46Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of non-condensed rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/49Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/50Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton to carbon atoms of non-condensed six-membered aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
OA1200200211A 2000-01-26 2001-01-18 Monohydrate of cis-lithium-cyano-4-Ä3-(cyclopentyloxy)-4-methoxyphenylÜcyclohexanecar-boxylate. OA12159A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17812900P 2000-01-26 2000-01-26

Publications (1)

Publication Number Publication Date
OA12159A true OA12159A (en) 2006-05-08

Family

ID=22651319

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200200211A OA12159A (en) 2000-01-26 2001-01-18 Monohydrate of cis-lithium-cyano-4-Ä3-(cyclopentyloxy)-4-methoxyphenylÜcyclohexanecar-boxylate.

Country Status (36)

Country Link
US (1) US6699903B2 (zh)
EP (1) EP1250313B1 (zh)
JP (1) JP2003520842A (zh)
KR (1) KR20020073183A (zh)
CN (1) CN1157371C (zh)
AP (1) AP1432A (zh)
AR (1) AR027273A1 (zh)
AT (1) ATE344235T1 (zh)
AU (1) AU3282201A (zh)
BG (1) BG106959A (zh)
BR (1) BR0107709A (zh)
CA (1) CA2397758A1 (zh)
CO (1) CO5300517A1 (zh)
CY (1) CY1108515T1 (zh)
CZ (1) CZ20022590A3 (zh)
DE (1) DE60124221T2 (zh)
DK (1) DK1250313T3 (zh)
DZ (1) DZ3285A1 (zh)
EA (1) EA200200791A1 (zh)
EG (1) EG24065A (zh)
ES (1) ES2273804T3 (zh)
HK (1) HK1051030A1 (zh)
HU (1) HUP0204150A3 (zh)
IL (1) IL150400A0 (zh)
MA (1) MA25652A1 (zh)
MX (1) MXPA02007300A (zh)
MY (1) MY122802A (zh)
NO (1) NO20023378L (zh)
NZ (1) NZ519799A (zh)
OA (1) OA12159A (zh)
PE (1) PE20011040A1 (zh)
PL (1) PL356832A1 (zh)
PT (1) PT1250313E (zh)
SK (1) SK10942002A3 (zh)
WO (1) WO2001055094A1 (zh)
ZA (1) ZA200205925B (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0011802D0 (en) * 2000-05-16 2000-07-05 Smithkline Beecham Method for enhancing cognitive function

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5552438A (en) 1992-04-02 1996-09-03 Smithkline Beecham Corporation Compounds useful for treating allergic and inflammatory diseases
UA67753C2 (uk) * 1997-10-10 2004-07-15 Смітклайн Бічам Корпорейшн Спосіб отримання заміщених 4-феніл-4-ціанциклогексанових кислот

Also Published As

Publication number Publication date
CY1108515T1 (el) 2014-04-09
EP1250313A4 (en) 2005-09-21
HUP0204150A2 (hu) 2003-04-28
HK1051030A1 (zh) 2003-07-18
MA25652A1 (fr) 2002-12-31
CN1395556A (zh) 2003-02-05
AU3282201A (en) 2001-08-07
WO2001055094A1 (en) 2001-08-02
US20030032670A1 (en) 2003-02-13
EG24065A (en) 2008-05-08
CZ20022590A3 (cs) 2003-01-15
DK1250313T3 (da) 2007-02-12
NO20023378D0 (no) 2002-07-12
BR0107709A (pt) 2002-11-19
JP2003520842A (ja) 2003-07-08
ZA200205925B (en) 2003-11-21
MY122802A (en) 2006-05-31
DZ3285A1 (fr) 2001-08-02
PE20011040A1 (es) 2001-10-31
AR027273A1 (es) 2003-03-19
ATE344235T1 (de) 2006-11-15
EP1250313B1 (en) 2006-11-02
ES2273804T3 (es) 2007-05-16
DE60124221T2 (de) 2007-09-13
KR20020073183A (ko) 2002-09-19
AP1432A (en) 2005-06-20
CO5300517A1 (es) 2003-07-31
CA2397758A1 (en) 2001-08-02
EA200200791A1 (ru) 2002-12-26
PL356832A1 (en) 2004-07-12
NZ519799A (en) 2004-04-30
AP2002002566A0 (en) 2002-06-30
CN1157371C (zh) 2004-07-14
US6699903B2 (en) 2004-03-02
PT1250313E (pt) 2007-01-31
DE60124221D1 (de) 2006-12-14
BG106959A (en) 2003-05-30
IL150400A0 (en) 2002-12-01
MXPA02007300A (es) 2002-11-29
NO20023378L (no) 2002-07-12
HUP0204150A3 (en) 2003-05-28
SK10942002A3 (sk) 2002-11-06
EP1250313A1 (en) 2002-10-23

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