OA11944A - 1-Trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives. - Google Patents

1-Trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives. Download PDF

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Publication number
OA11944A
OA11944A OA1200100302A OA1200100302A OA11944A OA 11944 A OA11944 A OA 11944A OA 1200100302 A OA1200100302 A OA 1200100302A OA 1200100302 A OA1200100302 A OA 1200100302A OA 11944 A OA11944 A OA 11944A
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OA
OAPI
Prior art keywords
disorder
disorders
syndrome
compound
alkyl
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Application number
OA1200100302A
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English (en)
Inventor
Ronald Scott Obach
Douglas Alan Scully
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Pfizer Prod Inc
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Publication of OA11944A publication Critical patent/OA11944A/en

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
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  • Reproductive Health (AREA)
  • Psychiatry (AREA)
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  • Dermatology (AREA)
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OA1200100302A 1999-05-21 2000-04-24 1-Trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives. OA11944A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13539999P 1999-05-21 1999-05-21

Publications (1)

Publication Number Publication Date
OA11944A true OA11944A (en) 2006-04-12

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ID=22467939

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Application Number Title Priority Date Filing Date
OA1200100302A OA11944A (en) 1999-05-21 2000-04-24 1-Trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives.

Country Status (49)

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US (1) US6239147B1 (es)
EP (1) EP1178984B1 (es)
JP (1) JP3802762B2 (es)
KR (1) KR100453301B1 (es)
CN (1) CN1140525C (es)
AP (1) AP1396A (es)
AR (1) AR020294A1 (es)
AT (1) ATE234832T1 (es)
AU (1) AU775861B2 (es)
BG (1) BG106152A (es)
BR (1) BR0011284A (es)
CA (1) CA2374643C (es)
CO (1) CO5170464A1 (es)
CR (1) CR6503A (es)
CZ (1) CZ20014164A3 (es)
DE (1) DE60001736T2 (es)
DK (1) DK1178984T3 (es)
DZ (1) DZ3044A1 (es)
EA (1) EA004233B1 (es)
EE (1) EE04719B1 (es)
ES (1) ES2190781T3 (es)
GC (1) GC0000254A (es)
GE (1) GEP20043225B (es)
GT (1) GT200000073A (es)
HK (1) HK1046280B (es)
HN (1) HN2000000057A (es)
HR (1) HRP20010861A2 (es)
HU (1) HUP0201443A3 (es)
IL (1) IL145949A0 (es)
IS (1) IS6123A (es)
MA (1) MA26734A1 (es)
MX (1) MXPA01011977A (es)
MY (1) MY123373A (es)
NO (1) NO322496B1 (es)
NZ (1) NZ514698A (es)
OA (1) OA11944A (es)
PA (1) PA8495201A1 (es)
PE (1) PE20010165A1 (es)
PL (1) PL198658B1 (es)
PT (1) PT1178984E (es)
SK (1) SK285819B6 (es)
SV (1) SV2002000077A (es)
TN (1) TNSN00105A1 (es)
TR (1) TR200103332T2 (es)
TW (1) TWI275588B (es)
UA (1) UA71004C2 (es)
UY (1) UY26147A1 (es)
WO (1) WO2000071538A2 (es)
ZA (1) ZA200109554B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists
ES2211455T3 (es) * 1999-10-18 2004-07-16 Pfizer Products Inc. Procedimiento para la preparacion de compuestos eteres ciclicos piperidinilaminometil trifluorometilicos.
DE10311984A1 (de) * 2003-03-12 2004-09-23 Freie Universität Berlin Verwendung von NEP-assoziierten Molekülen zur Behandlung von nichtimmunogenen-nichthypertensiven Zivilisationskrankheiten
US7122700B2 (en) * 2004-07-30 2006-10-17 Xerox Corporation Arylamine processes
US7868016B2 (en) * 2005-07-13 2011-01-11 Baxter International Inc. Pharmaceutical formulations of endo-N-(9-methyl-9-azabicyclo[3,3.1]non-3-yl)-1-methyl-1H-indazole-3-carboxamide hydrochloride
WO2009109001A1 (en) * 2008-03-04 2009-09-11 Adelaide Research & Innovation Pty Ltd Method for preventing and/or treating a disease, condition or state associated with reduced dopaminergic neuron function
EP3144303B1 (en) 2008-06-25 2018-09-26 Array Biopharma, Inc. 6-substituted phenoxychroman carboxylic acid derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY110227A (en) * 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
GB9317987D0 (en) * 1993-08-26 1993-10-13 Glaxo Group Ltd Chemical compounds
EP0826684B1 (en) * 1995-03-27 2001-11-21 Hisamitsu Pharmaceutical Co., Inc. Piperidine derivatives
RU2156250C2 (ru) * 1995-04-24 2000-09-20 Новартис Аг Производные хромона, способ их получения и фармацевтическая композиция
ATE199552T1 (de) * 1995-07-07 2001-03-15 Pfizer Substituierte benzolaktamverbindungen als substanz-p-antagonisten
TW340842B (en) * 1995-08-24 1998-09-21 Pfizer Substituted benzylaminopiperidine compounds
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists

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US6239147B1 (en) 2001-05-29
AU775861B2 (en) 2004-08-19
TWI275588B (en) 2007-03-11
CA2374643A1 (en) 2000-11-30
JP2003500405A (ja) 2003-01-07
IS6123A (is) 2001-10-23
HUP0201443A3 (en) 2005-09-28
HUP0201443A2 (en) 2002-08-28
EP1178984A2 (en) 2002-02-13
EA200101109A1 (ru) 2002-04-25
ZA200109554B (en) 2002-11-20
TR200103332T2 (tr) 2002-04-22
MY123373A (en) 2006-05-31
DE60001736T2 (de) 2003-09-18
PL352409A1 (en) 2003-08-25
HK1046280B (zh) 2004-10-21
PA8495201A1 (es) 2002-08-26
PT1178984E (pt) 2003-06-30
DE60001736D1 (de) 2003-04-24
EP1178984B1 (en) 2003-03-19
ATE234832T1 (de) 2003-04-15
CN1140525C (zh) 2004-03-03
AP1396A (en) 2005-04-19
JP3802762B2 (ja) 2006-07-26
MA26734A1 (fr) 2004-12-20
EE04719B1 (et) 2006-10-16
KR20020016793A (ko) 2002-03-06
UA71004C2 (uk) 2004-11-15
TNSN00105A1 (fr) 2005-11-10
CA2374643C (en) 2006-02-14
GEP20043225B (en) 2004-04-26
EA004233B1 (ru) 2004-02-26
PE20010165A1 (es) 2001-02-20
PL198658B1 (pl) 2008-07-31
HRP20010861A2 (en) 2003-04-30
EE200100612A (et) 2003-02-17
DZ3044A1 (fr) 2004-03-27
GT200000073A (es) 2001-11-09
IL145949A0 (en) 2002-07-25
CO5170464A1 (es) 2002-06-27
HK1046280A1 (en) 2003-01-03
ES2190781T3 (es) 2003-08-16
SV2002000077A (es) 2002-07-03
KR100453301B1 (ko) 2004-10-20
GC0000254A (en) 2006-11-01
WO2000071538A3 (en) 2001-02-22
BG106152A (en) 2002-06-28
AP2001002327A0 (en) 2001-12-31
DK1178984T3 (da) 2003-06-10
HN2000000057A (es) 2001-03-02
NO322496B1 (no) 2006-10-16
CN1355799A (zh) 2002-06-26
AR020294A1 (es) 2002-05-02
NO20015652D0 (no) 2001-11-20
WO2000071538A2 (en) 2000-11-30
SK16592001A3 (sk) 2003-03-04
MXPA01011977A (es) 2002-05-06
AU3667300A (en) 2000-12-12
NZ514698A (en) 2005-01-28
CR6503A (es) 2004-02-03
BR0011284A (pt) 2002-03-05
CZ20014164A3 (cs) 2003-01-15
SK285819B6 (sk) 2007-09-06
UY26147A1 (es) 2000-12-29
NO20015652L (no) 2002-01-14

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