OA10955A - A process for preparing naphthyridones and intermediates - Google Patents

A process for preparing naphthyridones and intermediates Download PDF

Info

Publication number
OA10955A
OA10955A OA9900005A OA9900005A OA10955A OA 10955 A OA10955 A OA 10955A OA 9900005 A OA9900005 A OA 9900005A OA 9900005 A OA9900005 A OA 9900005A OA 10955 A OA10955 A OA 10955A
Authority
OA
OAPI
Prior art keywords
formula
compound
alkyl
trifluoromethyl
process according
Prior art date
Application number
OA9900005A
Other languages
English (en)
Inventor
Kwok-Fung Chiu Charles
Lewin Theophilus Wint
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of OA10955A publication Critical patent/OA10955A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Indole Compounds (AREA)
OA9900005A 1998-01-16 1999-01-08 A process for preparing naphthyridones and intermediates OA10955A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7160198P 1998-01-16 1998-01-16

Publications (1)

Publication Number Publication Date
OA10955A true OA10955A (en) 2001-10-31

Family

ID=22102373

Family Applications (1)

Application Number Title Priority Date Filing Date
OA9900005A OA10955A (en) 1998-01-16 1999-01-08 A process for preparing naphthyridones and intermediates

Country Status (39)

Country Link
EP (1) EP0930297B1 (xx)
JP (1) JPH11255745A (xx)
KR (1) KR19990067905A (xx)
CN (1) CN1228422A (xx)
AP (1) AP9901440A0 (xx)
AR (1) AR017228A1 (xx)
AT (1) ATE238281T1 (xx)
AU (1) AU9711598A (xx)
BG (1) BG64094B1 (xx)
BR (1) BR9900066A (xx)
CA (1) CA2258960C (xx)
DE (1) DE69907042T2 (xx)
DK (1) DK0930297T3 (xx)
EA (1) EA199900020A3 (xx)
EG (1) EG21514A (xx)
ES (1) ES2195513T3 (xx)
GT (1) GT199800199A (xx)
HR (1) HRP990013A2 (xx)
HU (1) HUP9900121A3 (xx)
ID (1) ID23612A (xx)
IL (1) IL127945A0 (xx)
IS (1) IS4943A (xx)
MA (1) MA24745A1 (xx)
NO (1) NO990185L (xx)
NZ (1) NZ333769A (xx)
OA (1) OA10955A (xx)
PA (1) PA8464701A1 (xx)
PE (1) PE20000172A1 (xx)
PL (1) PL330859A1 (xx)
PT (1) PT930297E (xx)
SA (1) SA99190971A (xx)
SG (1) SG76584A1 (xx)
SI (1) SI0930297T1 (xx)
SK (1) SK3899A3 (xx)
TN (1) TNSN99005A1 (xx)
TR (1) TR199900070A2 (xx)
TW (1) TW483890B (xx)
YU (1) YU1799A (xx)
ZA (1) ZA99277B (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7019142B2 (en) * 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
HN1999000141A (es) * 1998-09-03 2000-06-19 Pfizer Prod Inc Procedimiento para preparar sales de trovafloxacina de adicion de acidos.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
IE66202B1 (en) * 1989-08-16 1995-12-13 Pfizer Azabicyclo quinolone carboxylic acids
US5256791A (en) * 1992-03-02 1993-10-26 Pfizer Inc. Preparation of intermediates in the synthesis of quinoline antibiotics
US5475116A (en) * 1994-04-29 1995-12-12 Pfizer Inc. Aza bicyclo[3,1,0]hexane intermediates useful in the synthesis of quinolones
DE19733439A1 (de) * 1997-08-02 1999-02-04 Bayer Ag Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften

Also Published As

Publication number Publication date
AP9901440A0 (en) 1999-03-31
TR199900070A3 (tr) 1999-10-21
JPH11255745A (ja) 1999-09-21
DE69907042D1 (de) 2003-05-28
TW483890B (en) 2002-04-21
AR017228A1 (es) 2001-08-22
KR19990067905A (ko) 1999-08-25
ID23612A (id) 2000-05-04
ES2195513T3 (es) 2003-12-01
TR199900070A2 (xx) 1999-10-21
NO990185L (no) 1999-07-19
HUP9900121A2 (hu) 1999-09-28
PE20000172A1 (es) 2000-03-09
DK0930297T3 (da) 2003-07-21
NZ333769A (en) 2000-03-27
HU9900121D0 (en) 1999-03-29
CA2258960A1 (en) 1999-07-16
GT199800199A (es) 2000-06-07
ZA99277B (en) 2000-07-17
AU9711598A (en) 1999-08-05
SG76584A1 (en) 2000-11-21
BG103087A (en) 1999-08-31
BG64094B1 (bg) 2003-12-31
PT930297E (pt) 2003-08-29
EP0930297B1 (en) 2003-04-23
IL127945A0 (en) 1999-11-30
CN1228422A (zh) 1999-09-15
EA199900020A2 (ru) 1999-08-26
TNSN99005A1 (fr) 2005-11-10
EG21514A (en) 2001-11-28
SI0930297T1 (en) 2003-08-31
DE69907042T2 (de) 2003-10-16
YU1799A (sh) 2000-03-21
SK3899A3 (en) 2000-03-13
NO990185D0 (no) 1999-01-15
IS4943A (is) 1999-07-17
ATE238281T1 (de) 2003-05-15
BR9900066A (pt) 2000-05-09
SA99190971A (ar) 2005-12-03
EP0930297A1 (en) 1999-07-21
HRP990013A2 (en) 1999-10-31
PA8464701A1 (es) 2000-09-29
CA2258960C (en) 2002-09-03
EA199900020A3 (ru) 1999-12-29
HUP9900121A3 (en) 2000-02-28
PL330859A1 (en) 1999-07-19
MA24745A1 (fr) 1999-10-01

Similar Documents

Publication Publication Date Title
US7038053B2 (en) Process for imidazo[4,5-c]pyridin-4-amines
US6184380B1 (en) Process for preparing naphthyridones and intermediates
EP0695755A1 (en) Pyrrolocarbazoles
AU8680598A (en) Alpha 1a adrenergic receptor antagonist
CA2368815A1 (en) Novel synthesis and crystallization of piperazine ring-containing compounds
OA10955A (en) A process for preparing naphthyridones and intermediates
AU694149B2 (en) Process and intermediates for preparing naphthyridonecarboxylic acid salts
US6576764B2 (en) Synthesis and crystallization of piperazine ring-containing compounds
US7019142B2 (en) Process for preparing naphthyridones and intermediates
US20030069417A1 (en) Novel synthesis and crystallization of piperazine ring-containing compounds
US6114531A (en) Process for preparing quinolone and naphthyridone carboxylic acids
US5442065A (en) Synthesis of tetrahydroquinoline enediyne core analogs of dynemicin
AU761035B2 (en) Process for preparing trovafloxacin acid salts
US5929240A (en) Process and intermediates for preparing naphthyridonecarboxylic acid salts
CZ11999A3 (cs) Způsob výroby naftyridonů a meziprodukty
US20030135043A1 (en) Novel synthesis and crystallization of piperazine ring-containing compounds
CA2140453A1 (en) Novel diazabicycloalkenes and processes for the preparation thereof