NZ189186A - 4-hydroxy-n-(thiazol-2-yl)/2h-1,2-benzothiazine-3-carboxamide-1,1-dioxide derivatives and pharmaceutical compositions - Google Patents

4-hydroxy-n-(thiazol-2-yl)/2h-1,2-benzothiazine-3-carboxamide-1,1-dioxide derivatives and pharmaceutical compositions

Info

Publication number
NZ189186A
NZ189186A NZ189186A NZ18918678A NZ189186A NZ 189186 A NZ189186 A NZ 189186A NZ 189186 A NZ189186 A NZ 189186A NZ 18918678 A NZ18918678 A NZ 18918678A NZ 189186 A NZ189186 A NZ 189186A
Authority
NZ
New Zealand
Prior art keywords
benzothiazine
thiazol
carboxamide
hydroxy
pharmaceutical compositions
Prior art date
Application number
NZ189186A
Other languages
English (en)
Inventor
W Engel
G Trummlitz
G Engelhardt
E Seeger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of NZ189186A publication Critical patent/NZ189186A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NZ189186A 1977-12-16 1978-12-15 4-hydroxy-n-(thiazol-2-yl)/2h-1,2-benzothiazine-3-carboxamide-1,1-dioxide derivatives and pharmaceutical compositions NZ189186A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772756113 DE2756113A1 (de) 1977-12-16 1977-12-16 Neue 4-hydroxy-2h-1,2-benzothiazin- 3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
NZ189186A true NZ189186A (en) 1981-03-16

Family

ID=6026297

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ189186A NZ189186A (en) 1977-12-16 1978-12-15 4-hydroxy-n-(thiazol-2-yl)/2h-1,2-benzothiazine-3-carboxamide-1,1-dioxide derivatives and pharmaceutical compositions

Country Status (27)

Country Link
US (1) US4233299A (https=)
EP (1) EP0002482B1 (https=)
JP (1) JPS5492976A (https=)
AT (1) AT365589B (https=)
AU (1) AU522538B2 (https=)
BG (2) BG33286A3 (https=)
CA (1) CA1102802A (https=)
CS (2) CS202515B2 (https=)
DD (1) DD140354A5 (https=)
DE (2) DE2756113A1 (https=)
DK (1) DK149344C (https=)
ES (2) ES475677A1 (https=)
FI (1) FI61896C (https=)
GR (1) GR65626B (https=)
HU (1) HU175846B (https=)
IE (1) IE48042B1 (https=)
IL (1) IL56206A (https=)
LU (1) LU88557I2 (https=)
MX (1) MX9202949A (https=)
NL (1) NL940002I2 (https=)
NO (2) NO150203C (https=)
NZ (1) NZ189186A (https=)
PL (1) PL115756B1 (https=)
PT (1) PT68915A (https=)
RO (1) RO75792A (https=)
SU (1) SU841588A3 (https=)
YU (1) YU294978A (https=)

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US3853862A (en) * 1973-04-23 1974-12-10 Pfizer Production of 4-hydroxy-1,2-benzothiazine-3-carboxamides
US3925371A (en) * 1974-09-23 1975-12-09 Mcneilab Inc Benzothiazine-1,1-dioxides
US3892740A (en) * 1974-10-15 1975-07-01 Pfizer Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides
US4074048A (en) * 1976-05-10 1978-02-14 Warner-Lambert Company Process for the preparation of 4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides
US4100347A (en) * 1976-06-10 1978-07-11 Pfizer Inc. 3,4-Dihydro-2-methyl-4-oxo-2H-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide

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HU175846B (hu) 1980-10-28
DD140354A5 (de) 1980-02-27
US4233299A (en) 1980-11-11
SU841588A3 (ru) 1981-06-23
FI61896B (fi) 1982-06-30
MX9202949A (es) 1992-07-01
ES550377A0 (es) 1988-06-16
EP0002482B1 (de) 1981-01-07
EP0002482A1 (de) 1979-06-27
PT68915A (de) 1979-01-01
ATA863078A (de) 1981-06-15
AU522538B2 (en) 1982-06-10
IL56206A0 (en) 1979-03-12
FI61896C (fi) 1982-10-11
AU4253078A (en) 1979-06-21
BG33286A3 (bg) 1983-01-14
ES8802454A3 (es) 1988-06-16
DE2756113A1 (de) 1979-06-21
YU294978A (en) 1982-10-31
DK149344C (da) 1986-10-13
LU88557I2 (fr) 1995-03-21
NL940002I1 (nl) 1994-03-16
NL940002I2 (nl) 1997-05-01
RO75792A (ro) 1981-02-28
CS202515B2 (en) 1981-01-30
DE2860445D1 (en) 1981-02-26
ES475677A1 (es) 1979-04-16
NO150203C (no) 1984-09-05
IE782482L (en) 1979-06-16
GR65626B (en) 1980-10-15
JPS6324997B2 (https=) 1988-05-23
NO1997002I1 (no) 1997-01-14
IE48042B1 (en) 1984-09-05
NO784231L (no) 1979-06-19
DK562078A (da) 1979-06-17
AT365589B (de) 1982-01-25
FI783867A7 (fi) 1979-06-17
DK149344B (da) 1986-05-12
IL56206A (en) 1982-04-30
CS410091A3 (en) 1992-06-17
PL115756B1 (en) 1981-04-30
PL211753A1 (pl) 1979-08-13
JPS5492976A (en) 1979-07-23
CA1102802A (en) 1981-06-09
BG60475B2 (bg) 1995-04-28
NO150203B (no) 1984-05-28

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