NO995482L - Ergolinderivater og deres anvendelse som somatostatinreseptorantagonister - Google Patents

Ergolinderivater og deres anvendelse som somatostatinreseptorantagonister

Info

Publication number
NO995482L
NO995482L NO995482A NO995482A NO995482L NO 995482 L NO995482 L NO 995482L NO 995482 A NO995482 A NO 995482A NO 995482 A NO995482 A NO 995482A NO 995482 L NO995482 L NO 995482L
Authority
NO
Norway
Prior art keywords
receptor antagonists
somatostatin receptor
ergoline derivatives
ergoline
derivatives
Prior art date
Application number
NO995482A
Other languages
English (en)
Norwegian (no)
Other versions
NO995482D0 (no
Inventor
Paul Pfaeffli
Peter Neumann
Robert Swoboda
Peter Stuetz
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO995482L publication Critical patent/NO995482L/no
Publication of NO995482D0 publication Critical patent/NO995482D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/04—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
    • C07D457/06—Lysergic acid amides
    • C07D457/08—Lysergic acid amides in which the amide nitrogen is a member of a heterocyclic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO995482A 1997-05-29 1999-11-09 Ergolinderivater og deres anvendelse som somatostatinreseptorantagonister NO995482D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9711043.1A GB9711043D0 (en) 1997-05-29 1997-05-29 Organic compounds
PCT/EP1998/003125 WO1998054183A2 (en) 1997-05-29 1998-05-27 Ergoline derivatives and their use as somatostatin receptor antagonists

Publications (2)

Publication Number Publication Date
NO995482L true NO995482L (no) 1999-11-09
NO995482D0 NO995482D0 (no) 1999-11-09

Family

ID=10813201

Family Applications (1)

Application Number Title Priority Date Filing Date
NO995482A NO995482D0 (no) 1997-05-29 1999-11-09 Ergolinderivater og deres anvendelse som somatostatinreseptorantagonister

Country Status (24)

Country Link
US (1) US6221870B1 (ru)
EP (1) EP0986558A2 (ru)
JP (1) JP2001527580A (ru)
KR (1) KR20010013103A (ru)
CN (1) CN1259946A (ru)
AR (1) AR012870A1 (ru)
AU (1) AU727841B2 (ru)
BR (1) BR9809491A (ru)
CA (1) CA2288810A1 (ru)
CO (1) CO4950561A1 (ru)
CZ (1) CZ289466B6 (ru)
GB (1) GB9711043D0 (ru)
HU (1) HUP0002311A3 (ru)
ID (1) ID22916A (ru)
IL (1) IL132571A0 (ru)
NO (1) NO995482D0 (ru)
NZ (1) NZ500386A (ru)
PE (1) PE74899A1 (ru)
PL (1) PL336502A1 (ru)
RU (1) RU2191776C2 (ru)
SK (1) SK160899A3 (ru)
TR (1) TR199902848T2 (ru)
WO (1) WO1998054183A2 (ru)
ZA (1) ZA984560B (ru)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10066158B4 (de) * 2000-08-24 2007-08-09 Neurobiotec Gmbh Verwendung eines transdermalen therapeutischen Systems zur Behandlung des Restless-Legs-Syndroms
DE10053397A1 (de) * 2000-10-20 2002-05-02 Schering Ag Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen
DE10341317B4 (de) * 2003-09-03 2008-10-23 Axxonis Pharma Ag Transdermales therapeutisches System (TTS) zur Verabreichung von Ergolinverbindungen ausgenommen Pergolid
US20070243240A9 (en) * 2000-08-24 2007-10-18 Fred Windt-Hanke Transdermal therapeutic system
AU2002305845B2 (en) * 2001-06-08 2006-03-30 Ipsen Pharma S.A.S. Somatostatin-dopamine chimeric analogs
FI20031454A0 (fi) 2003-10-06 2003-10-06 Juvantia Pharma Ltd Oy Selektiivisiä somatostatiinireseptori 1 ja/tai 4 -agonisteja ja -antagonisteja
KR101000923B1 (ko) * 2004-01-08 2010-12-13 삼성전자주식회사 원격 제어기의 매크로 설정 장치 및 방법
US20100048549A1 (en) * 2005-05-18 2010-02-25 Siegfried Wurster Peptidomimetics selective for the somatostatin receptor subtypes 1 and/or 4
JP2007067096A (ja) * 2005-08-30 2007-03-15 Fujitsu Ltd 半導体装置
EP2515654A4 (en) * 2009-12-23 2013-04-24 Map Pharmaceuticals Inc NEW ERGOLINANALOGA
MX2013015373A (es) 2011-06-23 2014-02-11 Map Pharmaceuticals Inc Nuevos analogos de fluoroergolina.
CA2859173A1 (en) 2011-12-19 2013-06-27 Map Pharmaceuticals, Inc. Novel iso-ergoline derivatives
CA2859175A1 (en) 2011-12-21 2013-06-27 Map Pharmaceuticals, Inc. Novel neuromodulatory compounds
US9012640B2 (en) 2012-06-22 2015-04-21 Map Pharmaceuticals, Inc. Cabergoline derivatives
WO2014070965A2 (en) 2012-11-01 2014-05-08 Ipsen Pharma S.A.S Somatostatin analogs and dimers thereof
TWI523863B (zh) 2012-11-01 2016-03-01 艾普森藥品公司 體抑素－多巴胺嵌合體類似物
CA2974113A1 (en) 2015-01-20 2016-07-28 Xoc Pharmaceuticals, Inc. Isoergoline compounds and uses thereof
CN113149982A (zh) 2015-01-20 2021-07-23 Xoc制药股份有限公司 麦角灵化合物及其用途
WO2018223065A1 (en) 2017-06-01 2018-12-06 Xoc Pharmaceuticals, Inc. Ergoline derivatives for use in medicine
JP7099717B2 (ja) 2019-09-30 2022-07-12 株式会社理研バイオ ソマトスタチン受容体

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH475252A (de) * 1966-02-08 1969-07-15 Sandoz Ag Verfahren zur Herstellung neuer Lysergsäure-Derivate
US3592816A (en) 1966-02-08 1971-07-13 Sandoz Ltd N-substituted piperazides of lysergic acid
GB1188197A (en) 1967-10-11 1970-04-15 Sandoz Ltd Lysergic Acid Derivatives
NL6818658A (ru) * 1968-01-18 1969-07-22
GB1580448A (en) * 1976-12-06 1980-12-03 Farmaceutici Italia 8 -acetyl-6-methyl-ergoline i derivatives
GB8501078D0 (en) * 1985-01-16 1985-02-20 Erba Farmitalia Piperazin-1-yl-ergo-line derivatives
TW357143B (en) * 1995-07-07 1999-05-01 Novartis Ag Benzo[g]quinoline derivatives

Also Published As

Publication number Publication date
NO995482D0 (no) 1999-11-09
ID22916A (id) 1999-12-16
CZ289466B6 (cs) 2002-01-16
PE74899A1 (es) 1999-09-14
BR9809491A (pt) 2000-10-17
EP0986558A2 (en) 2000-03-22
CA2288810A1 (en) 1998-12-03
PL336502A1 (en) 2000-07-03
GB9711043D0 (en) 1997-07-23
AR012870A1 (es) 2000-11-22
WO1998054183A2 (en) 1998-12-03
US6221870B1 (en) 2001-04-24
JP2001527580A (ja) 2001-12-25
KR20010013103A (ko) 2001-02-26
CZ424599A3 (cs) 2000-03-15
RU2191776C2 (ru) 2002-10-27
SK160899A3 (en) 2000-07-11
ZA984560B (en) 1998-11-30
HUP0002311A3 (en) 2002-08-28
AU8210898A (en) 1998-12-30
TR199902848T2 (xx) 2000-02-21
IL132571A0 (en) 2001-03-19
HUP0002311A2 (hu) 2000-12-28
NZ500386A (en) 2002-05-31
WO1998054183A3 (en) 1999-03-04
CO4950561A1 (es) 2000-09-01
AU727841B2 (en) 2001-01-04
CN1259946A (zh) 2000-07-12

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application