NO20020314L - 2-arylimino-2,3-dihydrotiazoler og deres anvendelse som ligander for somatostatin-reseptorer - Google Patents

2-arylimino-2,3-dihydrotiazoler og deres anvendelse som ligander for somatostatin-reseptorer

Info

Publication number
NO20020314L
NO20020314L NO20020314A NO20020314A NO20020314L NO 20020314 L NO20020314 L NO 20020314L NO 20020314 A NO20020314 A NO 20020314A NO 20020314 A NO20020314 A NO 20020314A NO 20020314 L NO20020314 L NO 20020314L
Authority
NO
Norway
Prior art keywords
dihydrotiazoles
arylimino
ligands
somatostatin receptors
somatostatin
Prior art date
Application number
NO20020314A
Other languages
English (en)
Other versions
NO20020314D0 (no
NO322394B1 (no
Inventor
Christophe Philippe Moinet
Carole Sackur
Christophe Thurieau
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Publication of NO20020314D0 publication Critical patent/NO20020314D0/no
Publication of NO20020314L publication Critical patent/NO20020314L/no
Publication of NO322394B1 publication Critical patent/NO322394B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures
NO20020314A 1999-07-22 2002-01-21 2-arylimino-2,3-dihydrotiazoler, fremgangsmate for fremstilling av disse, farmasoytiske preparater inneholdende disse samt deres anvendelse for fremstilling av medikamenter for behandling av tilstander eller sykdommer der somatostatinreseptorene er innvolvert. NO322394B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9909496A FR2796643B1 (fr) 1999-07-22 1999-07-22 Derives de 2-arylimino-2, 3-dihydrothiazoles, leurs procedes de preparation et leur utilisation therapeutique
PCT/FR2000/002095 WO2001007424A1 (fr) 1999-07-22 2000-07-21 2-arylimino-2,3-dihydrothiazoles et leur utilisation comme ligands des recepteurs de la somatostatine

Publications (3)

Publication Number Publication Date
NO20020314D0 NO20020314D0 (no) 2002-01-21
NO20020314L true NO20020314L (no) 2002-03-06
NO322394B1 NO322394B1 (no) 2006-10-02

Family

ID=9548380

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20020314A NO322394B1 (no) 1999-07-22 2002-01-21 2-arylimino-2,3-dihydrotiazoler, fremgangsmate for fremstilling av disse, farmasoytiske preparater inneholdende disse samt deres anvendelse for fremstilling av medikamenter for behandling av tilstander eller sykdommer der somatostatinreseptorene er innvolvert.

Country Status (20)

Country Link
US (1) US6727269B1 (no)
EP (1) EP1202980A1 (no)
JP (2) JP4063537B2 (no)
KR (1) KR100692352B1 (no)
CN (1) CN100443479C (no)
AR (1) AR035321A1 (no)
AU (1) AU782187B2 (no)
BR (1) BR0012647A (no)
CA (1) CA2382940C (no)
CZ (1) CZ302073B6 (no)
FR (1) FR2796643B1 (no)
HK (1) HK1048314A1 (no)
HU (1) HUP0202425A3 (no)
IL (3) IL147582A0 (no)
MX (1) MXPA02000723A (no)
NO (1) NO322394B1 (no)
NZ (1) NZ516599A (no)
PL (1) PL353831A1 (no)
RU (1) RU2266287C2 (no)
WO (1) WO2001007424A1 (no)

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FR2819508B1 (fr) * 2001-01-12 2005-01-21 Sod Conseils Rech Applic Derives de 2-arylimino-2, 3-dihydorthiazoles, leurs procedes de preparation et leur utilisation therapeutiques
ATE451102T1 (de) * 2000-06-30 2009-12-15 Dainippon Sumitomo Pharma Co Thiazol-derivate zur verwendung als entzündungshemmende mittel
DE10133665A1 (de) * 2001-07-11 2003-01-30 Boehringer Ingelheim Pharma Carbonsäurederivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung
WO2003057214A1 (en) 2001-12-28 2003-07-17 Somatocor Pharmaceuticals, Inc. Imidazolidin-2,4-dione derivatives as non-peptide somatostatin receptor ligands
US7067538B2 (en) 2002-08-09 2006-06-27 Warner-Lambert Company, Llc MCP-1 receptor antagonists and methods of use thereof
JP4896387B2 (ja) * 2003-09-30 2012-03-14 武田薬品工業株式会社 チアゾリン誘導体およびその用途
EP1669352A4 (en) 2003-09-30 2008-12-17 Takeda Pharmaceutical THIAZOLINE DERIVATIVE AND ITS USE
WO2005082845A1 (en) * 2004-02-27 2005-09-09 Oy Juvantia Pharma Ltd Novel therapies with somatostatin receptor agonists
WO2005082844A1 (en) * 2004-02-27 2005-09-09 Oy Juvantia Pharma Ltd Treatment of diseases by using a somatostatin receptor agonist
PL2653465T3 (pl) 2004-03-15 2017-01-31 Janssen Pharmaceutica Nv Modulatory receptora opioidowego
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US7910613B2 (en) * 2004-09-22 2011-03-22 H. Lundbeck A/S 2-acylaminothiazole derivatives
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US8841334B2 (en) 2006-05-31 2014-09-23 Abbvie Inc. Compounds as cannabinoid receptor ligands and uses thereof
BRPI0712720A2 (pt) * 2006-05-31 2012-11-20 Abbott Lab compostos tiazàis como ligantes do receptor canabinàide e usos dos mesmos
WO2008028094A1 (en) 2006-08-31 2008-03-06 Abbott Laboratories Compounds as cb2 cannabinoid receptor ligands
US7868038B2 (en) 2006-08-31 2011-01-11 Abbott Laboratories Compounds as cannabinoid receptor ligands
EP2142522A1 (en) 2007-03-28 2010-01-13 Abbott Laboratories 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands
US7872033B2 (en) 2007-04-17 2011-01-18 Abbott Laboratories Compounds as cannabinoid receptor ligands
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CZ302073B6 (cs) 2010-09-29
NO20020314D0 (no) 2002-01-21
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US6727269B1 (en) 2004-04-27
HK1048314A1 (en) 2003-03-28
BR0012647A (pt) 2002-04-09
CN100443479C (zh) 2008-12-17
AU782187B2 (en) 2005-07-07
JP2006257093A (ja) 2006-09-28
CN1362952A (zh) 2002-08-07
FR2796643B1 (fr) 2005-04-29
FR2796643A1 (fr) 2001-01-26
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KR20020088405A (ko) 2002-11-27
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