DE60026169D1 - Selektive neurokinin-antagonisten - Google Patents

Selektive neurokinin-antagonisten

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Publication number
DE60026169D1
DE60026169D1 DE60026169T DE60026169T DE60026169D1 DE 60026169 D1 DE60026169 D1 DE 60026169D1 DE 60026169 T DE60026169 T DE 60026169T DE 60026169 T DE60026169 T DE 60026169T DE 60026169 D1 DE60026169 D1 DE 60026169D1
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Germany
Prior art keywords
selective
neurokinine
antagonists
neurokinine antagonists
selective neurokinine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60026169T
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English (en)
Other versions
DE60026169T2 (de
Inventor
Neng-Yang Shih
Ho-Jane Shue
A Reichard
Sunil Paliwal
J Blythin
J Piwinski
Dong Xiao
Xiao Chen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Sharp and Dohme Corp
Original Assignee
Schering Corp
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Publication date
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Publication of DE60026169D1 publication Critical patent/DE60026169D1/de
Publication of DE60026169T2 publication Critical patent/DE60026169T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503—Five-membered rings
    • C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3
DE60026169T 1999-12-17 2000-12-14 Selektive neurokinin-antagonisten Expired - Lifetime DE60026169T2 (de)

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WO2001044200A2 (en) 2001-06-21
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AR026990A1 (es) 2003-03-05
CO5261559A1 (es) 2003-03-31
WO2001044200A3 (en) 2001-12-13
CA2393672A1 (en) 2001-06-21
KR20020067548A (ko) 2002-08-22
EP1237874A2 (de) 2002-09-11
AU2097601A (en) 2001-06-25
EP1237874B1 (de) 2006-02-22
ECSP003828A (es) 2002-02-25
ES2258485T3 (es) 2006-09-01
ZA200204395B (en) 2003-11-26
JP2003522739A (ja) 2003-07-29
IL150033A0 (en) 2002-12-01
PE20011035A1 (es) 2001-10-13
DE60026169T2 (de) 2006-11-09
HUP0301607A2 (hu) 2003-12-29
HUP0301607A3 (en) 2004-03-29
HK1045308A1 (zh) 2002-11-22
ATE318259T1 (de) 2006-03-15

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