NO995482L - Ergolinderivater og deres anvendelse som somatostatinreseptorantagonister - Google Patents
Ergolinderivater og deres anvendelse som somatostatinreseptorantagonisterInfo
- Publication number
- NO995482L NO995482L NO995482A NO995482A NO995482L NO 995482 L NO995482 L NO 995482L NO 995482 A NO995482 A NO 995482A NO 995482 A NO995482 A NO 995482A NO 995482 L NO995482 L NO 995482L
- Authority
- NO
- Norway
- Prior art keywords
- receptor antagonists
- somatostatin receptor
- ergoline derivatives
- ergoline
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/04—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
- C07D457/06—Lysergic acid amides
- C07D457/08—Lysergic acid amides in which the amide nitrogen is a member of a heterocyclic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9711043.1A GB9711043D0 (en) | 1997-05-29 | 1997-05-29 | Organic compounds |
PCT/EP1998/003125 WO1998054183A2 (en) | 1997-05-29 | 1998-05-27 | Ergoline derivatives and their use as somatostatin receptor antagonists |
Publications (2)
Publication Number | Publication Date |
---|---|
NO995482D0 NO995482D0 (no) | 1999-11-09 |
NO995482L true NO995482L (no) | 1999-11-09 |
Family
ID=10813201
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO995482A NO995482L (no) | 1997-05-29 | 1999-11-09 | Ergolinderivater og deres anvendelse som somatostatinreseptorantagonister |
Country Status (24)
Country | Link |
---|---|
US (1) | US6221870B1 (no) |
EP (1) | EP0986558A2 (no) |
JP (1) | JP2001527580A (no) |
KR (1) | KR20010013103A (no) |
CN (1) | CN1259946A (no) |
AR (1) | AR012870A1 (no) |
AU (1) | AU727841B2 (no) |
BR (1) | BR9809491A (no) |
CA (1) | CA2288810A1 (no) |
CO (1) | CO4950561A1 (no) |
CZ (1) | CZ289466B6 (no) |
GB (1) | GB9711043D0 (no) |
HU (1) | HUP0002311A3 (no) |
ID (1) | ID22916A (no) |
IL (1) | IL132571A0 (no) |
NO (1) | NO995482L (no) |
NZ (1) | NZ500386A (no) |
PE (1) | PE74899A1 (no) |
PL (1) | PL336502A1 (no) |
RU (1) | RU2191776C2 (no) |
SK (1) | SK160899A3 (no) |
TR (1) | TR199902848T2 (no) |
WO (1) | WO1998054183A2 (no) |
ZA (1) | ZA984560B (no) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10053397A1 (de) | 2000-10-20 | 2002-05-02 | Schering Ag | Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen |
DE10341317B4 (de) * | 2003-09-03 | 2008-10-23 | Axxonis Pharma Ag | Transdermales therapeutisches System (TTS) zur Verabreichung von Ergolinverbindungen ausgenommen Pergolid |
US20070243240A9 (en) * | 2000-08-24 | 2007-10-18 | Fred Windt-Hanke | Transdermal therapeutic system |
DE10043321B4 (de) * | 2000-08-24 | 2005-07-28 | Neurobiotec Gmbh | Verwendung eines transdermalen therapeutischen Systems zur Behandlung der Parkinsonschen Krankheit, zur Behandlung und Prävention des prämenstruellen Syndroms und zur Lactationshemmung |
ES2325880T3 (es) * | 2001-06-08 | 2009-09-23 | Ipsen Pharma | Analogos quimericos de somatostatina-dopamina. |
FI20031454A0 (fi) | 2003-10-06 | 2003-10-06 | Juvantia Pharma Ltd Oy | Selektiivisiä somatostatiinireseptori 1 ja/tai 4 -agonisteja ja -antagonisteja |
KR101000923B1 (ko) * | 2004-01-08 | 2010-12-13 | 삼성전자주식회사 | 원격 제어기의 매크로 설정 장치 및 방법 |
JP2008540618A (ja) * | 2005-05-18 | 2008-11-20 | ブルスター,ジークフリート | ソマトスタチン受容体サブタイプ1及び/又は4に選択的なペプチド模倣薬 |
JP2007067096A (ja) * | 2005-08-30 | 2007-03-15 | Fujitsu Ltd | 半導体装置 |
SG181896A1 (en) * | 2009-12-23 | 2012-07-30 | Map Pharmaceuticals Inc | Novel ergoline analogs |
US8604035B2 (en) * | 2011-06-23 | 2013-12-10 | Map Pharmaceuticals, Inc. | Fluoroergoline analogs |
SG11201403434YA (en) | 2011-12-19 | 2014-09-26 | Map Pharmaceuticals Inc | Novel iso-ergoline derivatives |
EP2793583A4 (en) | 2011-12-21 | 2015-08-12 | Map Pharmaceuticals Inc | NOVEL NEUROMODULATORY CONNECTIONS |
US9012640B2 (en) | 2012-06-22 | 2015-04-21 | Map Pharmaceuticals, Inc. | Cabergoline derivatives |
CN104768565B (zh) | 2012-11-01 | 2017-04-26 | 益普生制药股份有限公司 | 促生长素抑制素类似物及其二聚体 |
TWI523863B (zh) | 2012-11-01 | 2016-03-01 | 艾普森藥品公司 | 體抑素-多巴胺嵌合體類似物 |
US9676776B2 (en) | 2015-01-20 | 2017-06-13 | Xoc Pharmaceuticals, Inc. | Isoergoline compounds and uses thereof |
EP3253753A4 (en) | 2015-01-20 | 2018-06-27 | Xoc Pharmaceuticals, Inc | Ergoline compounds and uses thereof |
AU2018275873A1 (en) | 2017-06-01 | 2019-12-19 | Xoc Pharmaceuticals, Inc. | Ergoline derivatives for use in medicine |
JP7099717B2 (ja) | 2019-09-30 | 2022-07-12 | 株式会社理研バイオ | ソマトスタチン受容体 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3592816A (en) | 1966-02-08 | 1971-07-13 | Sandoz Ltd | N-substituted piperazides of lysergic acid |
CH475252A (de) * | 1966-02-08 | 1969-07-15 | Sandoz Ag | Verfahren zur Herstellung neuer Lysergsäure-Derivate |
GB1188197A (en) | 1967-10-11 | 1970-04-15 | Sandoz Ltd | Lysergic Acid Derivatives |
NL6818658A (no) * | 1968-01-18 | 1969-07-22 | ||
GB1580448A (en) * | 1976-12-06 | 1980-12-03 | Farmaceutici Italia | 8 -acetyl-6-methyl-ergoline i derivatives |
GB8501078D0 (en) * | 1985-01-16 | 1985-02-20 | Erba Farmitalia | Piperazin-1-yl-ergo-line derivatives |
TW357143B (en) * | 1995-07-07 | 1999-05-01 | Novartis Ag | Benzo[g]quinoline derivatives |
-
1997
- 1997-05-29 GB GBGB9711043.1A patent/GB9711043D0/en active Pending
-
1998
- 1998-05-27 AR ARP980102461A patent/AR012870A1/es unknown
- 1998-05-27 JP JP50023799A patent/JP2001527580A/ja active Pending
- 1998-05-27 HU HU0002311A patent/HUP0002311A3/hu unknown
- 1998-05-27 NZ NZ500386A patent/NZ500386A/en unknown
- 1998-05-27 KR KR19997011082A patent/KR20010013103A/ko active IP Right Grant
- 1998-05-27 AU AU82108/98A patent/AU727841B2/en not_active Ceased
- 1998-05-27 TR TR1999/02848T patent/TR199902848T2/xx unknown
- 1998-05-27 CZ CZ19994245A patent/CZ289466B6/cs not_active IP Right Cessation
- 1998-05-27 RU RU99127433/04A patent/RU2191776C2/ru active
- 1998-05-27 SK SK1608-99A patent/SK160899A3/sk unknown
- 1998-05-27 PE PE1998000425A patent/PE74899A1/es not_active Application Discontinuation
- 1998-05-27 BR BR9809491-2A patent/BR9809491A/pt not_active IP Right Cessation
- 1998-05-27 CA CA002288810A patent/CA2288810A1/en not_active Abandoned
- 1998-05-27 PL PL98336502A patent/PL336502A1/xx unknown
- 1998-05-27 CN CN98805488A patent/CN1259946A/zh active Pending
- 1998-05-27 ID IDW991445A patent/ID22916A/id unknown
- 1998-05-27 IL IL13257198A patent/IL132571A0/xx unknown
- 1998-05-27 EP EP98932090A patent/EP0986558A2/en not_active Withdrawn
- 1998-05-27 US US09/424,377 patent/US6221870B1/en not_active Expired - Fee Related
- 1998-05-27 WO PCT/EP1998/003125 patent/WO1998054183A2/en not_active Application Discontinuation
- 1998-05-28 CO CO98030085A patent/CO4950561A1/es unknown
- 1998-05-28 ZA ZA984560A patent/ZA984560B/xx unknown
-
1999
- 1999-11-09 NO NO995482A patent/NO995482L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
TR199902848T2 (xx) | 2000-02-21 |
RU2191776C2 (ru) | 2002-10-27 |
AU8210898A (en) | 1998-12-30 |
CZ289466B6 (cs) | 2002-01-16 |
NZ500386A (en) | 2002-05-31 |
CA2288810A1 (en) | 1998-12-03 |
WO1998054183A3 (en) | 1999-03-04 |
HUP0002311A2 (hu) | 2000-12-28 |
AR012870A1 (es) | 2000-11-22 |
ZA984560B (en) | 1998-11-30 |
EP0986558A2 (en) | 2000-03-22 |
US6221870B1 (en) | 2001-04-24 |
IL132571A0 (en) | 2001-03-19 |
GB9711043D0 (en) | 1997-07-23 |
WO1998054183A2 (en) | 1998-12-03 |
BR9809491A (pt) | 2000-10-17 |
CZ424599A3 (cs) | 2000-03-15 |
CO4950561A1 (es) | 2000-09-01 |
CN1259946A (zh) | 2000-07-12 |
ID22916A (id) | 1999-12-16 |
AU727841B2 (en) | 2001-01-04 |
PL336502A1 (en) | 2000-07-03 |
NO995482D0 (no) | 1999-11-09 |
KR20010013103A (ko) | 2001-02-26 |
HUP0002311A3 (en) | 2002-08-28 |
JP2001527580A (ja) | 2001-12-25 |
PE74899A1 (es) | 1999-09-14 |
SK160899A3 (en) | 2000-07-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |