NO951640L - Antimikrobielle 5-hydrazinokinolonderivater - Google Patents
Antimikrobielle 5-hydrazinokinolonderivaterInfo
- Publication number
- NO951640L NO951640L NO951640A NO951640A NO951640L NO 951640 L NO951640 L NO 951640L NO 951640 A NO951640 A NO 951640A NO 951640 A NO951640 A NO 951640A NO 951640 L NO951640 L NO 951640L
- Authority
- NO
- Norway
- Prior art keywords
- hydrazinoquinolone
- antimicrobial
- derivatives
- lower alkyl
- heterocyclic ring
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US96896092A | 1992-10-30 | 1992-10-30 | |
PCT/US1993/010091 WO1994010163A1 (fr) | 1992-10-30 | 1993-10-22 | Derives antimicrobiens de 5-hydrazino-quinolone |
Publications (2)
Publication Number | Publication Date |
---|---|
NO951640D0 NO951640D0 (no) | 1995-04-28 |
NO951640L true NO951640L (no) | 1995-06-30 |
Family
ID=25514997
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO951640A NO951640L (no) | 1992-10-30 | 1995-04-28 | Antimikrobielle 5-hydrazinokinolonderivater |
Country Status (21)
Country | Link |
---|---|
EP (1) | EP0666853A1 (fr) |
JP (1) | JPH08502750A (fr) |
KR (1) | KR950704301A (fr) |
CN (1) | CN1064357C (fr) |
AU (1) | AU687018B2 (fr) |
BR (1) | BR9307347A (fr) |
CA (1) | CA2148003A1 (fr) |
CZ (1) | CZ282581B6 (fr) |
EG (1) | EG20543A (fr) |
FI (1) | FI952049A0 (fr) |
HU (1) | HUT72072A (fr) |
IL (1) | IL107323A (fr) |
MX (1) | MX9306814A (fr) |
NO (1) | NO951640L (fr) |
NZ (1) | NZ257470A (fr) |
PL (1) | PL178094B1 (fr) |
RU (1) | RU2126000C1 (fr) |
SG (1) | SG59979A1 (fr) |
SK (1) | SK54795A3 (fr) |
WO (1) | WO1994010163A1 (fr) |
ZA (1) | ZA938089B (fr) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5646163A (en) * | 1992-10-30 | 1997-07-08 | The Procter & Gamble Company | Quinolone 5-(N-heterosubstituted amino) antimicrobials |
NZ290722A (en) * | 1994-08-02 | 1999-03-29 | Procter & Gamble | A process for making derivatives of quinolonyl lactam (qla's); intermediates |
DE69515882T2 (de) * | 1994-08-02 | 2000-11-02 | Procter & Gamble | Verfahren zur herstellung von antimikrobiellen verbindungen |
CA2242242C (fr) * | 1996-02-09 | 2001-08-07 | Toyama Chemical Co., Ltd. | Derives de l'acide quinolonecarboxylique et leurs sels |
PT1901749T (pt) * | 2005-05-18 | 2016-11-04 | Raptor Pharmaceuticals Inc | Fluoroquinolonas aerossolizadas e suas utilizações |
US8546423B2 (en) | 2005-05-18 | 2013-10-01 | Mpex Pharmaceuticals, Inc. | Aerosolized fluoroquinolones and uses thereof |
CA2528849C (fr) | 2005-06-08 | 2014-01-14 | Janssen Pharmaceutica N.V. | Derives de quinoleine utilises comme agents antibacteriens |
EA010601B1 (ru) * | 2005-06-09 | 2008-10-30 | Янссен Фармацевтика Н.В. | Производные хинолина в качестве антибактериальных агентов |
CN101020647B (zh) * | 2007-02-14 | 2011-03-30 | 杭州师范学院 | 一种β-环丙胺基丙烯酸(酯)的合成方法 |
JP5363350B2 (ja) * | 2007-03-19 | 2013-12-11 | 武田薬品工業株式会社 | Mapk/erkキナーゼ阻害剤 |
EP3092901B1 (fr) * | 2007-10-05 | 2020-04-29 | Senhwa Biosciences, Inc. | Analogues de quinolone et procédés associés |
WO2009147616A1 (fr) * | 2008-06-03 | 2009-12-10 | Actelion Pharmaceuticals Ltd | Dérivés de [4-(1-amino-éthyl)-cyclohexyl]-méthyl-amine et de [6-(1-amino-ethyl)-tétrahydro-pyran-3-yl]-méthyl-amine |
MX345158B (es) | 2008-10-07 | 2017-01-18 | Raptor Pharmaceuticals Inc | Formulaciones de fluoroquinolona en aerosol para farmacocinetica mejorada. |
HUE050147T2 (hu) | 2008-10-07 | 2020-11-30 | Horizon Orphan Llc | Tüdõgyulladás csökkentése levofloxacin belélegzése útján |
AR076222A1 (es) * | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen |
AU2010289326B2 (en) | 2009-09-04 | 2015-09-24 | Horizon Therapeutics U.S. Holding Llc | Use of aerosolized levofloxacin for treating cystic fibrosis |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4668680A (en) * | 1985-12-12 | 1987-05-26 | Warner-Lambert Company | 5-amino-6,8-difluoroquinolones as antibacterial agents |
JPH0228178A (ja) * | 1988-04-23 | 1990-01-30 | Toyama Chem Co Ltd | 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法 |
DE3906365A1 (de) * | 1988-07-15 | 1990-01-18 | Bayer Ag | 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe |
WO1991002526A1 (fr) * | 1989-08-16 | 1991-03-07 | Pfizer Inc. | Acides azabicyclo quinolone carboxyliques |
ES2147721T3 (es) * | 1990-04-18 | 2000-10-01 | Procter & Gamble Pharma | Quinolonil lactamas antimicrobianas. |
CA2095338C (fr) * | 1990-11-30 | 2002-04-09 | John Michael Domagala | Utilisation des stereoisomeres individuels des 7-[3-(aminoalkyl)-1-pyrrolidinyl]-quinolones et des naphthyridones comme agents antibacteriens |
-
1993
- 1993-01-30 EG EG68693A patent/EG20543A/xx active
- 1993-10-19 IL IL10732393A patent/IL107323A/xx not_active IP Right Cessation
- 1993-10-22 SK SK547-95A patent/SK54795A3/sk unknown
- 1993-10-22 EP EP93924393A patent/EP0666853A1/fr not_active Withdrawn
- 1993-10-22 BR BR9307347A patent/BR9307347A/pt not_active Application Discontinuation
- 1993-10-22 CA CA002148003A patent/CA2148003A1/fr not_active Abandoned
- 1993-10-22 WO PCT/US1993/010091 patent/WO1994010163A1/fr not_active Application Discontinuation
- 1993-10-22 CZ CZ951097A patent/CZ282581B6/cs not_active IP Right Cessation
- 1993-10-22 KR KR1019950701690A patent/KR950704301A/ko active IP Right Grant
- 1993-10-22 AU AU54097/94A patent/AU687018B2/en not_active Ceased
- 1993-10-22 SG SG1996007851A patent/SG59979A1/en unknown
- 1993-10-22 JP JP6511167A patent/JPH08502750A/ja active Pending
- 1993-10-22 PL PL93308671A patent/PL178094B1/pl unknown
- 1993-10-22 HU HU9501237A patent/HUT72072A/hu unknown
- 1993-10-22 RU RU95110762A patent/RU2126000C1/ru active
- 1993-10-22 NZ NZ257470A patent/NZ257470A/xx unknown
- 1993-10-29 MX MX9306814A patent/MX9306814A/es not_active IP Right Cessation
- 1993-10-29 ZA ZA938089A patent/ZA938089B/xx unknown
- 1993-10-30 CN CN93120224A patent/CN1064357C/zh not_active Expired - Fee Related
-
1995
- 1995-04-28 FI FI952049A patent/FI952049A0/fi unknown
- 1995-04-28 NO NO951640A patent/NO951640L/no unknown
Also Published As
Publication number | Publication date |
---|---|
CZ109795A3 (en) | 1995-12-13 |
IL107323A (en) | 2000-06-01 |
RU95110762A (ru) | 1997-01-10 |
MX9306814A (es) | 1994-07-29 |
NZ257470A (en) | 1997-08-22 |
SG59979A1 (en) | 1999-02-22 |
CA2148003A1 (fr) | 1994-05-11 |
KR950704301A (ko) | 1995-11-17 |
HUT72072A (en) | 1996-03-28 |
FI952049A (fi) | 1995-04-28 |
CN1092773A (zh) | 1994-09-28 |
IL107323A0 (en) | 1994-01-25 |
PL178094B1 (pl) | 2000-02-29 |
PL308671A1 (en) | 1995-08-21 |
BR9307347A (pt) | 1999-05-25 |
ZA938089B (en) | 1994-06-07 |
AU687018B2 (en) | 1998-02-19 |
AU5409794A (en) | 1994-05-24 |
EP0666853A1 (fr) | 1995-08-16 |
CN1064357C (zh) | 2001-04-11 |
HU9501237D0 (en) | 1995-06-28 |
WO1994010163A1 (fr) | 1994-05-11 |
FI952049A0 (fi) | 1995-04-28 |
NO951640D0 (no) | 1995-04-28 |
CZ282581B6 (cs) | 1997-08-13 |
SK54795A3 (en) | 1995-12-06 |
RU2126000C1 (ru) | 1999-02-10 |
EG20543A (en) | 1999-07-31 |
JPH08502750A (ja) | 1996-03-26 |
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