NO943826L - Heteroarylpiperidiner, fremgangsmåte for fremstilling og farmasöytiske blandinger hvor de er tilstede - Google Patents
Heteroarylpiperidiner, fremgangsmåte for fremstilling og farmasöytiske blandinger hvor de er tilstedeInfo
- Publication number
- NO943826L NO943826L NO943826A NO943826A NO943826L NO 943826 L NO943826 L NO 943826L NO 943826 A NO943826 A NO 943826A NO 943826 A NO943826 A NO 943826A NO 943826 L NO943826 L NO 943826L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- heteroberl
- piperidines
- present
- pharmaceutical compositions
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000003053 piperidines Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000000198 serotonin 5-HT3 receptor agonist Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Det beskrives nye heteroarylpiperidiner med formel (I) Hal Alk NH2 0) hvor Hal er et halogenatom, Alk er en (Cj-CJalkylgruppe og hver av X, Y og Z er -CH=, eller en av dem er et nitrogenatom og de øvrige er -CH=, og deres salter, en fremgangsmåte for deres fremstilling og deres anvendelse som medikamenter som virker som 5-HT3-agonister.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP93402498 | 1993-10-11 |
Publications (2)
Publication Number | Publication Date |
---|---|
NO943826D0 NO943826D0 (no) | 1994-10-10 |
NO943826L true NO943826L (no) | 1995-04-12 |
Family
ID=8214753
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO943826A NO943826L (no) | 1993-10-11 | 1994-10-10 | Heteroarylpiperidiner, fremgangsmåte for fremstilling og farmasöytiske blandinger hvor de er tilstede |
Country Status (15)
Country | Link |
---|---|
US (3) | US5502063A (no) |
JP (1) | JPH07165754A (no) |
KR (1) | KR950011436A (no) |
CN (1) | CN1106400A (no) |
AU (2) | AU687090B2 (no) |
CA (1) | CA2133855A1 (no) |
FI (1) | FI944751A (no) |
HU (1) | HUT71349A (no) |
IL (1) | IL111216A (no) |
NO (1) | NO943826L (no) |
NZ (1) | NZ264634A (no) |
RU (1) | RU94036762A (no) |
SG (1) | SG47476A1 (no) |
TW (1) | TW274548B (no) |
ZA (1) | ZA947924B (no) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2133855A1 (en) * | 1993-10-11 | 1995-04-12 | Marco Baroni | Heteroarylpiperidines, process for their preparation and pharmaceutical compositions in which they are present |
AU3463497A (en) * | 1996-07-23 | 1998-02-10 | Yamanouchi Pharmaceutical Co., Ltd. | Novel medicinal compositions for therapeutic use |
US6242473B1 (en) * | 1999-01-08 | 2001-06-05 | Maxim Pharmaceuticals, Inc. | Treatment and prevention of reactive oxygen metabolite-mediated cellular damage |
DE60011895T2 (de) * | 1999-05-21 | 2005-08-04 | Abbott Laboratories, Abbott Park | Heterocyclische subtituierte aminoazacyclische verbindungen mit zentraler nervensystemwirkung |
WO2006062063A1 (ja) * | 2004-12-08 | 2006-06-15 | Astellas Pharma Inc. | ピペリジン誘導体及びその製造法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4302455A (en) * | 1980-04-14 | 1981-11-24 | Merck & Co., Inc. | 2-(4-Aminopiperidino)pyrazines |
US5001125A (en) * | 1984-03-26 | 1991-03-19 | Janssen Pharmaceutica N.V. | Anti-virally active pyridazinamines |
US5196439A (en) * | 1987-11-27 | 1993-03-23 | Eisai Co., Ltd. | Piperidine compounds useful to treat cerebrovascular diseases |
ATE175113T1 (de) * | 1991-03-27 | 1999-01-15 | Sanofi Sa | Verwendung von 4-amino-1-(2-pyridyl)piperidinen als 5-ht3-agonisten zur behandlung und verhütung von serotoninergen dysfunktionen |
JPH0665203A (ja) * | 1992-06-25 | 1994-03-08 | Elf Sanofi | ピペラジンのヘテロ環誘導体 |
CA2133855A1 (en) * | 1993-10-11 | 1995-04-12 | Marco Baroni | Heteroarylpiperidines, process for their preparation and pharmaceutical compositions in which they are present |
-
1994
- 1994-10-07 CA CA002133855A patent/CA2133855A1/en not_active Abandoned
- 1994-10-07 NZ NZ264634A patent/NZ264634A/en unknown
- 1994-10-07 US US08/319,595 patent/US5502063A/en not_active Expired - Fee Related
- 1994-10-10 HU HU9402919A patent/HUT71349A/hu unknown
- 1994-10-10 NO NO943826A patent/NO943826L/no unknown
- 1994-10-10 IL IL11121694A patent/IL111216A/en not_active IP Right Cessation
- 1994-10-10 SG SG1996002107A patent/SG47476A1/en unknown
- 1994-10-10 RU RU94036762/04A patent/RU94036762A/ru unknown
- 1994-10-10 FI FI944751A patent/FI944751A/fi unknown
- 1994-10-11 JP JP6245145A patent/JPH07165754A/ja not_active Withdrawn
- 1994-10-11 AU AU75745/94A patent/AU687090B2/en not_active Ceased
- 1994-10-11 ZA ZA947924A patent/ZA947924B/xx unknown
- 1994-10-11 KR KR1019940026020A patent/KR950011436A/ko not_active Application Discontinuation
- 1994-10-11 CN CN94117118A patent/CN1106400A/zh active Pending
- 1994-10-11 TW TW083109398A patent/TW274548B/zh active
-
1995
- 1995-06-06 US US08/469,511 patent/US5595994A/en not_active Expired - Fee Related
- 1995-06-06 US US08/469,523 patent/US5723611A/en not_active Expired - Fee Related
-
1998
- 1998-05-13 AU AU64881/98A patent/AU6488198A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
KR950011436A (ko) | 1995-05-15 |
AU687090B2 (en) | 1998-02-19 |
US5723611A (en) | 1998-03-03 |
TW274548B (no) | 1996-04-21 |
FI944751A (fi) | 1995-04-12 |
AU7574594A (en) | 1995-04-27 |
SG47476A1 (en) | 1998-04-17 |
NZ264634A (en) | 1995-12-21 |
ZA947924B (en) | 1995-05-26 |
HU9402919D0 (en) | 1995-01-30 |
NO943826D0 (no) | 1994-10-10 |
JPH07165754A (ja) | 1995-06-27 |
FI944751A0 (fi) | 1994-10-10 |
AU6488198A (en) | 1998-07-02 |
US5502063A (en) | 1996-03-26 |
IL111216A0 (en) | 1994-12-29 |
HUT71349A (en) | 1995-11-28 |
CA2133855A1 (en) | 1995-04-12 |
RU94036762A (ru) | 1996-09-10 |
CN1106400A (zh) | 1995-08-09 |
US5595994A (en) | 1997-01-21 |
IL111216A (en) | 1999-03-12 |
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