NO904031D0 - Fremgangsmaate ved fremstilling av beta-karbonyl-karboksyamider av 1,3-tiazolidiner. - Google Patents

Fremgangsmaate ved fremstilling av beta-karbonyl-karboksyamider av 1,3-tiazolidiner.

Info

Publication number
NO904031D0
NO904031D0 NO1990904031A NO904031A NO904031D0 NO 904031 D0 NO904031 D0 NO 904031D0 NO 1990904031 A NO1990904031 A NO 1990904031A NO 904031 A NO904031 A NO 904031A NO 904031 D0 NO904031 D0 NO 904031D0
Authority
NO
Norway
Prior art keywords
carboxyamides
thiazolidines
carbonyl
beta
procedure
Prior art date
Application number
NO1990904031A
Other languages
English (en)
Other versions
NO904031L (no
NO179370C (no
NO179370B (no
Inventor
Carmelo A Gandolfi
Roberto Di Domenico
Silvano Spinelli
Licia Gallico
Bruno Lumachi
Sergio Tognella
Original Assignee
Boehringer Biochemia Srl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Biochemia Srl filed Critical Boehringer Biochemia Srl
Publication of NO904031D0 publication Critical patent/NO904031D0/no
Publication of NO904031L publication Critical patent/NO904031L/no
Publication of NO179370B publication Critical patent/NO179370B/no
Publication of NO179370C publication Critical patent/NO179370C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Electric Double-Layer Capacitors Or The Like (AREA)
  • Carbon And Carbon Compounds (AREA)
NO904031A 1988-03-17 1990-09-14 Analogifremgangsmåte ved fremstilling av terapeutisk aktive -karbonyl-karboksyamider av 1,3-tiazolidiner NO179370C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT8819813A IT1216119B (it) 1988-03-17 1988-03-17 Beta_carbonil_carbossiamidi di 1,3_tiazolidine.
PCT/EP1989/000205 WO1989008648A1 (en) 1988-03-17 1989-03-02 beta-CARBONYL-CARBOXYAMIDES OF 1,3-THIAZOLIDINES

Publications (4)

Publication Number Publication Date
NO904031D0 true NO904031D0 (no) 1990-09-14
NO904031L NO904031L (no) 1990-11-16
NO179370B NO179370B (no) 1996-06-17
NO179370C NO179370C (no) 1996-09-25

Family

ID=11161493

Family Applications (1)

Application Number Title Priority Date Filing Date
NO904031A NO179370C (no) 1988-03-17 1990-09-14 Analogifremgangsmåte ved fremstilling av terapeutisk aktive -karbonyl-karboksyamider av 1,3-tiazolidiner

Country Status (19)

Country Link
US (1) US5206254A (no)
EP (2) EP0407403A1 (no)
JP (1) JPH0688987B2 (no)
KR (1) KR960011381B1 (no)
AT (1) ATE95814T1 (no)
AU (1) AU624124B2 (no)
BG (1) BG60459B1 (no)
CA (1) CA1325632C (no)
DE (1) DE68909815T2 (no)
DK (1) DK168486B1 (no)
ES (1) ES2059595T3 (no)
FI (1) FI95247C (no)
HU (1) HU205920B (no)
IT (1) IT1216119B (no)
NO (1) NO179370C (no)
RO (1) RO107656B1 (no)
RU (1) RU1833378C (no)
WO (1) WO1989008648A1 (no)
ZA (1) ZA892014B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1245712B (it) * 1991-04-09 1994-10-14 Boehringer Mannheim Italia Ammine eterocicliche utili terapia dell'asma e dell'infiammazione delle vie aeree
IT1270594B (it) * 1994-07-07 1997-05-07 Recordati Chem Pharm Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
US6586466B2 (en) 1995-10-30 2003-07-01 Smithkline Beecham Corporation Carbohydrazide-protease inhibitors
US6083964A (en) * 1998-02-18 2000-07-04 K And K Biosciences, Inc. Optical resolution of racemic aminoalkylpyridine anticonvulsants and (+) aminoalkylpyridine enantiomers as highly potent orally effective anticonvulsant drugs and excitatory amino acid antagonists
JP5558648B2 (ja) 1998-11-23 2014-07-23 デイビス、ボニー アセチルコリンエステラーゼ阻害剤のための投与製剤
CN1319955C (zh) * 2003-06-10 2007-06-06 浙江海正药业股份有限公司 莫吉斯坦晶型
WO2008144956A1 (fr) * 2007-05-28 2008-12-04 Tianjin Institute Of Pharmaceutical Research Nouveaux composés ambroxol, leurs procédés de préparation et leurs utilisations
EP2070915A1 (en) * 2007-12-03 2009-06-17 A.M.S.A. ANONIMA MATERIE SINTETICHE E AFFINI S.p.A. New process for the synthesis of moguisteine
CN102653527A (zh) * 2011-12-22 2012-09-05 东莞达信生物技术有限公司 一种莫吉司坦合成工艺

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU195492B (en) * 1984-07-27 1988-05-30 Boehringer Biochemia Srl Process for producing 2-substituted thiazolidine derivatives with antitussive and mucus regulating action and pharmaceuticals comprising these compounds as active ingredient
GB2164333B (en) * 1984-07-27 1988-11-16 Boehringer Biochemia Srl Antitussive and mucus regulating 2-substituted thiazolidines
IT1201489B (it) * 1985-11-13 1989-02-02 Chiesi Farma Spa Derivati di tiazolidina,loro procedimento di preparazione e formulazioni farmaceutiche
IT1228251B (it) * 1987-07-02 1991-06-05 Boehringer Biochemia Srl Amidi di amino-tioacetali ciclici, procedimento per la loro preparazione e composizioni farmaceutiche che li contengono

Also Published As

Publication number Publication date
DK221490A (da) 1990-09-14
DK168486B1 (da) 1994-04-05
NO904031L (no) 1990-11-16
ATE95814T1 (de) 1993-10-15
RU1833378C (en) 1993-08-07
DE68909815D1 (de) 1993-11-18
DK221490D0 (da) 1990-09-14
KR900700470A (ko) 1990-08-13
KR960011381B1 (ko) 1996-08-22
NO179370C (no) 1996-09-25
ES2059595T3 (es) 1994-11-16
FI904512A0 (fi) 1990-09-13
AU624124B2 (en) 1992-06-04
HU205920B (en) 1992-07-28
AU3189289A (en) 1989-10-05
HUT56355A (en) 1991-08-28
NO179370B (no) 1996-06-17
FI95247C (fi) 1996-01-10
DE68909815T2 (de) 1994-03-24
CA1325632C (en) 1993-12-28
IT8819813A0 (it) 1988-03-17
WO1989008648A1 (en) 1989-09-21
BG92842A (bg) 1993-12-24
RO107656B1 (ro) 1993-12-30
EP0407403A1 (en) 1991-01-16
FI95247B (fi) 1995-09-29
ZA892014B (en) 1989-11-29
BG60459B1 (bg) 1995-04-28
JPH0688987B2 (ja) 1994-11-09
JPH03504123A (ja) 1991-09-12
US5206254A (en) 1993-04-27
EP0333080A1 (en) 1989-09-20
EP0333080B1 (en) 1993-10-13
IT1216119B (it) 1990-02-22
HU891559D0 (en) 1991-06-28

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Legal Events

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