NO881544L - Nye 2-acylpyrrolidinderivater, samt fremgangsmaater for fremstilling derav. - Google Patents
Nye 2-acylpyrrolidinderivater, samt fremgangsmaater for fremstilling derav.Info
- Publication number
- NO881544L NO881544L NO881544A NO881544A NO881544L NO 881544 L NO881544 L NO 881544L NO 881544 A NO881544 A NO 881544A NO 881544 A NO881544 A NO 881544A NO 881544 L NO881544 L NO 881544L
- Authority
- NO
- Norway
- Prior art keywords
- acylpyrrolide
- ingredients
- procedures
- preparing
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19873712365 DE3712365A1 (de) | 1987-04-11 | 1987-04-11 | Neue 2-acylpyrrolidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel sowie deren verwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
NO881544D0 NO881544D0 (no) | 1988-04-08 |
NO881544L true NO881544L (no) | 1988-10-12 |
Family
ID=6325457
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO881544A NO881544L (no) | 1987-04-11 | 1988-04-08 | Nye 2-acylpyrrolidinderivater, samt fremgangsmaater for fremstilling derav. |
Country Status (14)
Country | Link |
---|---|
US (1) | US4912127A (hu) |
EP (1) | EP0286928A3 (hu) |
JP (1) | JPS63267755A (hu) |
KR (1) | KR880012543A (hu) |
AU (1) | AU607754B2 (hu) |
DE (1) | DE3712365A1 (hu) |
DK (1) | DK193088A (hu) |
FI (1) | FI881613A (hu) |
HU (1) | HU199784B (hu) |
IL (1) | IL86027A (hu) |
NO (1) | NO881544L (hu) |
PH (1) | PH25713A (hu) |
PT (1) | PT87195B (hu) |
ZA (1) | ZA882459B (hu) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3712364A1 (de) * | 1987-04-11 | 1988-10-27 | Hoechst Ag | Neue pyrrolidin-2-(1,3-dicarbonyl)-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel sowie deren verwendung |
DE3742431A1 (de) * | 1987-12-15 | 1989-07-13 | Hoechst Ag | Neue derivate cyclischer aminosaeuren, verfahren zu ihrer herstellung, sie enthaltende mittel und deren verwendung |
US5053414A (en) * | 1988-04-08 | 1991-10-01 | Ono Pharmaceutical Co., Ltd. | Heterocyclic compounds |
JPH0825995B2 (ja) * | 1988-04-08 | 1996-03-13 | 小野薬品工業株式会社 | 複素環化合物 |
DE3817468A1 (de) * | 1988-05-21 | 1989-11-30 | Hoechst Ag | Ethylenisch ungesaettigte harnstoffderivate und verfahren zu ihrer herstellung |
US5254696A (en) * | 1990-09-13 | 1993-10-19 | Bayer Aktiengesellschaft | N-acylpyrrolidine derivatives |
DE4029054A1 (de) * | 1990-09-13 | 1992-03-19 | Bayer Ag | N-acylpyrrolidin-derivate |
DE69431359T2 (de) * | 1993-12-02 | 2003-07-31 | Merrell Pharmaceuticals Inc., Cincinnati | Prolyl-endopeptidaseinhibitoren |
DE19527574A1 (de) * | 1995-07-28 | 1997-01-30 | Basf Ag | Verfahren zur Herstellung vona-(N,N-Dialkyl)-aminocaarbonsäureamiden |
AR038967A1 (es) * | 2002-03-18 | 2005-02-02 | Solvay Pharm Bv | Derivados de 2,3 - diaril - pirazolidinas como inhibidores de enzimas que degradan la neurotensina |
ATE462432T1 (de) | 2003-05-05 | 2010-04-15 | Probiodrug Ag | Glutaminylcyclase-hemmer |
NZ546887A (en) * | 2003-11-03 | 2009-04-30 | Probiodrug Ag | Combinations useful for the treatment of neuronal disorders |
AU2005210004B2 (en) | 2004-02-05 | 2010-10-28 | Probiodrug Ag | Novel inhibitors of glutaminyl cyclase |
WO2008144748A1 (en) | 2007-05-21 | 2008-11-27 | The Uab Research Foundation | Prolyl endopeptidase inhibitors for reducing or preventing neutrophilic inflammation |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1492640A (en) * | 1975-07-08 | 1977-11-23 | Ucb Sa | L-pyroglutamyl-l-prolinamide |
US4560795A (en) * | 1979-04-10 | 1985-12-24 | Merrell Dow France et Cie. | α-Halomethyl derivatives of α-amino acids |
US4499102A (en) * | 1979-12-13 | 1985-02-12 | Santen Pharmaceutical Co., Ltd. | Thiazolidine and pyrrolidine compounds and pharmaceutical compositions containing them |
US4277395A (en) * | 1980-06-16 | 1981-07-07 | Richardson-Merrell Inc. | Novel enzyme inhibitors |
GB2083030B (en) * | 1980-08-23 | 1984-03-07 | Merrell Toraude & Co | Fluorinated pentene diamine derivatives |
US4456594A (en) * | 1981-11-06 | 1984-06-26 | Smithkline Beckman Corporation | N-Carboxyalkylproline-containing tripeptides |
US4483991A (en) * | 1983-01-17 | 1984-11-20 | American Home Products Corporation | Hypotensive agents |
US4518528A (en) * | 1983-05-19 | 1985-05-21 | Rasnick David W | α Amino fluoro ketones |
JPS6137764A (ja) * | 1984-07-31 | 1986-02-22 | Suntory Ltd | 抗プロリルエンドペプチダ−ゼ活性を有する新規生理活性化合物 |
JPH0655758B2 (ja) * | 1984-08-24 | 1994-07-27 | 味の素株式会社 | アミノ酸誘導体 |
US4626545A (en) * | 1984-08-27 | 1986-12-02 | Merck & Co., Inc. | Amino acid derivatives as enzyme inhibitors |
US4762821A (en) * | 1985-03-22 | 1988-08-09 | Syntex (U.S.A.) Inc. | N',N"-dialkylguanidino dipeptides |
DE3680578D1 (de) * | 1985-04-16 | 1991-09-05 | Suntory Ltd | Dipeptid-derivate, verfahren zur herstellung, pharmazeutische zusammensetzungen und ihre anwendung. |
JPH0623190B2 (ja) * | 1985-04-16 | 1994-03-30 | サントリー株式会社 | インヒビタ−活性を有するn−アシルピロリジン誘導体及びその製法並びに用途 |
JPH0653757B2 (ja) * | 1985-12-06 | 1994-07-20 | 味の素株式会社 | プロリン誘導体の芳香族スルホン酸塩 |
JPH08806B2 (ja) * | 1986-11-18 | 1996-01-10 | サントリー株式会社 | プロリルエンドペプチダ−ゼ阻害作用を有する新規ピロリジンアミド誘導体 |
DE3712364A1 (de) * | 1987-04-11 | 1988-10-27 | Hoechst Ag | Neue pyrrolidin-2-(1,3-dicarbonyl)-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel sowie deren verwendung |
DE3712363A1 (de) * | 1987-04-11 | 1988-10-27 | Hoechst Ag | Neue pyrrolidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel sowie deren verwendung |
-
1987
- 1987-04-11 DE DE19873712365 patent/DE3712365A1/de not_active Withdrawn
-
1988
- 1988-04-01 EP EP19880105332 patent/EP0286928A3/de not_active Withdrawn
- 1988-04-07 FI FI881613A patent/FI881613A/fi not_active Application Discontinuation
- 1988-04-08 US US07/179,292 patent/US4912127A/en not_active Expired - Fee Related
- 1988-04-08 PT PT87195A patent/PT87195B/pt not_active IP Right Cessation
- 1988-04-08 JP JP63085539A patent/JPS63267755A/ja active Pending
- 1988-04-08 DK DK193088A patent/DK193088A/da not_active Application Discontinuation
- 1988-04-08 NO NO881544A patent/NO881544L/no unknown
- 1988-04-08 HU HU881780A patent/HU199784B/hu not_active IP Right Cessation
- 1988-04-08 ZA ZA882459A patent/ZA882459B/xx unknown
- 1988-04-11 IL IL86027A patent/IL86027A/xx unknown
- 1988-04-11 AU AU14466/88A patent/AU607754B2/en not_active Ceased
- 1988-04-11 PH PH36780A patent/PH25713A/en unknown
- 1988-04-11 KR KR1019880004071A patent/KR880012543A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JPS63267755A (ja) | 1988-11-04 |
DE3712365A1 (de) | 1988-10-27 |
FI881613A0 (fi) | 1988-04-07 |
EP0286928A3 (de) | 1991-05-08 |
EP0286928A2 (de) | 1988-10-19 |
AU1446688A (en) | 1988-10-13 |
US4912127A (en) | 1990-03-27 |
HUT46888A (en) | 1988-12-28 |
ZA882459B (en) | 1988-09-29 |
KR880012543A (ko) | 1988-11-28 |
PH25713A (en) | 1991-09-18 |
NO881544D0 (no) | 1988-04-08 |
IL86027A (en) | 1992-05-25 |
IL86027A0 (en) | 1988-09-30 |
HU199784B (en) | 1990-03-28 |
AU607754B2 (en) | 1991-03-14 |
DK193088D0 (da) | 1988-04-08 |
FI881613A (fi) | 1988-10-12 |
DK193088A (da) | 1988-10-12 |
PT87195A (pt) | 1988-05-01 |
PT87195B (pt) | 1992-07-31 |
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