NO333656B1 - Benzimidazo[2,1-b][3]benzazepin-forbindelse og anvendelse derav - Google Patents
Benzimidazo[2,1-b][3]benzazepin-forbindelse og anvendelse derav Download PDFInfo
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- NO333656B1 NO333656B1 NO20042618A NO20042618A NO333656B1 NO 333656 B1 NO333656 B1 NO 333656B1 NO 20042618 A NO20042618 A NO 20042618A NO 20042618 A NO20042618 A NO 20042618A NO 333656 B1 NO333656 B1 NO 333656B1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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EP01204574 | 2001-11-23 | ||
PCT/EP2002/013180 WO2003044023A1 (en) | 2001-11-23 | 2002-11-22 | The use of anti-histaminics for acute reduction of elevated intracranial pressure |
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NO20042618L NO20042618L (no) | 2004-06-22 |
NO333656B1 true NO333656B1 (no) | 2013-08-05 |
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NO20042618A NO333656B1 (no) | 2001-11-23 | 2004-06-22 | Benzimidazo[2,1-b][3]benzazepin-forbindelse og anvendelse derav |
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EP (2) | EP1451196B1 (pt) |
JP (2) | JP4505226B2 (pt) |
KR (1) | KR100967601B1 (pt) |
CN (2) | CN100478031C (pt) |
AT (2) | ATE370149T1 (pt) |
AU (1) | AU2002356715B2 (pt) |
CA (2) | CA2467097C (pt) |
CY (2) | CY1107472T1 (pt) |
DE (2) | DE60231351D1 (pt) |
DK (2) | DK1451196T3 (pt) |
ES (2) | ES2290364T3 (pt) |
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HR (1) | HRP20040427B1 (pt) |
HU (1) | HU229118B1 (pt) |
IL (4) | IL162109A0 (pt) |
MX (1) | MXPA04004867A (pt) |
NO (1) | NO333656B1 (pt) |
NZ (2) | NZ550723A (pt) |
PL (1) | PL209953B1 (pt) |
PT (2) | PT1451196E (pt) |
RU (1) | RU2311418C2 (pt) |
SI (2) | SI1451196T1 (pt) |
UA (1) | UA76803C2 (pt) |
WO (1) | WO2003044023A1 (pt) |
ZA (1) | ZA200403923B (pt) |
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DK1451196T3 (da) | 2001-11-23 | 2007-11-12 | Janssen Pharmaceutica Nv | Anvendelse af substituerede tetracykliske imidazolderivater som antihistaminstoffer |
TWI290140B (en) * | 2003-08-25 | 2007-11-21 | Schering Corp | 2-Substituted benzimidazole derivatives as selective melanin concentrating hormone receptor antagonists for thr treatment of obesity and related disorders |
EP2796683A4 (en) * | 2011-12-20 | 2015-05-20 | Toyota Motor Co Ltd | ERROR DETECTION DEVICE FOR AN ELECTRICALLY HEATABLE CATALYST |
US9717726B2 (en) * | 2013-03-14 | 2017-08-01 | Maregade Rx, LLC | Product and method for treating diarrhea |
EP3558296B1 (en) | 2016-12-23 | 2023-06-28 | Maregade RX, LLC | Low dose product and method for treating diarrhea |
US10947253B2 (en) | 2019-08-05 | 2021-03-16 | Ankh Life Sciences Limited | Fused polycyclic dimers |
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US5595988A (en) * | 1992-12-04 | 1997-01-21 | Janssen Pharmaceutica N.V. | Triazolo(pyrrolo, thieno or furano)azepine derivatives |
TW382017B (en) * | 1995-12-27 | 2000-02-11 | Janssen Pharmaceutica Nv | 1-(1,2-disubstituted piperidinyl)-4-(fused imidazole)-piperidine derivatives |
TW429256B (en) | 1995-12-27 | 2001-04-11 | Janssen Pharmaceutica Nv | 1-(1,2-disubstituted piperidinyl)-4-(benzimidazolyl- and imidazopyridinyl)-piperidine derivatives |
TW527186B (en) * | 1996-03-19 | 2003-04-11 | Janssen Pharmaceutica Nv | Fused imidazole derivatives as multidrug resistance modulators |
EP1011726B1 (en) * | 1997-09-18 | 2003-02-26 | Janssen Pharmaceutica N.V. | Fused imidazole derivatives for improving oral bioavailability of pharmaceutical agents |
EP1401838B1 (en) * | 2001-06-12 | 2014-03-26 | Janssen Pharmaceutica NV | Novel substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine |
DK1451196T3 (da) | 2001-11-23 | 2007-11-12 | Janssen Pharmaceutica Nv | Anvendelse af substituerede tetracykliske imidazolderivater som antihistaminstoffer |
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