NO333196B1 - Anvendelse av gemifloksasin eller et salt derav, og et betalaktamantibiotikum for fremstilling av et medikament til behandling av bakterielle infeksjoner, samt sett omfattende gemifloksasin eller et salt derav og en betalaktamantibiotikaformulering - Google Patents
Anvendelse av gemifloksasin eller et salt derav, og et betalaktamantibiotikum for fremstilling av et medikament til behandling av bakterielle infeksjoner, samt sett omfattende gemifloksasin eller et salt derav og en betalaktamantibiotikaformulering Download PDFInfo
- Publication number
- NO333196B1 NO333196B1 NO20042711A NO20042711A NO333196B1 NO 333196 B1 NO333196 B1 NO 333196B1 NO 20042711 A NO20042711 A NO 20042711A NO 20042711 A NO20042711 A NO 20042711A NO 333196 B1 NO333196 B1 NO 333196B1
- Authority
- NO
- Norway
- Prior art keywords
- gemifloxacin
- salt
- lactam antibiotic
- beta
- treatment
- Prior art date
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- HGBLNBBNRORJKI-WCABBAIRSA-N cyclacillin Chemical compound N([C@H]1[C@H]2SC([C@@H](N2C1=O)C(O)=O)(C)C)C(=O)C1(N)CCCCC1 HGBLNBBNRORJKI-WCABBAIRSA-N 0.000 description 1
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- ZKUKMWMSYCIYRD-ZXFNITATSA-N lenampicillin Chemical compound O1C(=O)OC(COC(=O)[C@H]2C(S[C@H]3N2C([C@H]3NC(=O)[C@H](N)C=2C=CC=CC=2)=O)(C)C)=C1C ZKUKMWMSYCIYRD-ZXFNITATSA-N 0.000 description 1
- 229950005831 lenampicillin Drugs 0.000 description 1
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- 231100000417 nephrotoxicity Toxicity 0.000 description 1
- 229960001180 norfloxacin Drugs 0.000 description 1
- 239000003883 ointment base Substances 0.000 description 1
- 229940055577 oleyl alcohol Drugs 0.000 description 1
- XMLQWXUVTXCDDL-UHFFFAOYSA-N oleyl alcohol Natural products CCCCCCC=CCCCCCCCCCCO XMLQWXUVTXCDDL-UHFFFAOYSA-N 0.000 description 1
- 230000035515 penetration Effects 0.000 description 1
- 235000019371 penicillin G benzathine Nutrition 0.000 description 1
- 229940056360 penicillin g Drugs 0.000 description 1
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- 150000002960 penicillins Chemical class 0.000 description 1
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- BPLBGHOLXOTWMN-MBNYWOFBSA-N phenoxymethylpenicillin Chemical compound N([C@H]1[C@H]2SC([C@@H](N2C1=O)C(O)=O)(C)C)C(=O)COC1=CC=CC=C1 BPLBGHOLXOTWMN-MBNYWOFBSA-N 0.000 description 1
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- WCMIIGXFCMNQDS-IDYPWDAWSA-M piperacillin sodium Chemical compound [Na+].O=C1C(=O)N(CC)CCN1C(=O)N[C@H](C=1C=CC=CC=1)C(=O)N[C@@H]1C(=O)N2[C@@H](C([O-])=O)C(C)(C)S[C@@H]21 WCMIIGXFCMNQDS-IDYPWDAWSA-M 0.000 description 1
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- OHKOGUYZJXTSFX-KZFFXBSXSA-N ticarcillin Chemical compound C=1([C@@H](C(O)=O)C(=O)N[C@H]2[C@H]3SC([C@@H](N3C2=O)C(O)=O)(C)C)C=CSC=1 OHKOGUYZJXTSFX-KZFFXBSXSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
- A61K31/546—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33449501P | 2001-11-30 | 2001-11-30 | |
| PCT/KR2002/002248 WO2003045390A1 (en) | 2001-11-30 | 2002-11-29 | A METHOD OF TREATING BACTERIAL INFECTIONS USING GEMIFLOXACIN OR A SALT THEREOF AND A β -LACTAM ANTIBIOTIC |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20042711L NO20042711L (no) | 2004-06-30 |
| NO333196B1 true NO333196B1 (no) | 2013-04-02 |
Family
ID=23307473
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20042711A NO333196B1 (no) | 2001-11-30 | 2004-06-28 | Anvendelse av gemifloksasin eller et salt derav, og et betalaktamantibiotikum for fremstilling av et medikament til behandling av bakterielle infeksjoner, samt sett omfattende gemifloksasin eller et salt derav og en betalaktamantibiotikaformulering |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US7169792B2 (de) |
| EP (1) | EP1458391B1 (de) |
| AT (1) | ATE372119T1 (de) |
| AU (1) | AU2002360218A1 (de) |
| CA (1) | CA2468036C (de) |
| CY (1) | CY1107038T1 (de) |
| DE (1) | DE60222298T2 (de) |
| DK (1) | DK1458391T3 (de) |
| ES (1) | ES2292844T3 (de) |
| MX (1) | MXPA04005179A (de) |
| NO (1) | NO333196B1 (de) |
| PT (1) | PT1458391E (de) |
| WO (1) | WO2003045390A1 (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011101710A1 (en) * | 2010-02-16 | 2011-08-25 | Wockhardt Research Centre | Efflux pump inhibitors |
| ITMI20080289A1 (it) * | 2008-02-22 | 2009-08-23 | S I F I Societa Industria Farmaceutica Italia | Composizioni di gemifloxacina con elevata efficacia su patologie oculari |
| EP2143422A1 (de) * | 2008-07-11 | 2010-01-13 | S.I.F.I - Società Industria Farmaceutica Italiana - S.P.A. | Ophthalmische Zusammensetzungen enthaltend Gemifloxacin zur Behandlung von Augeninfektionen |
| MX349603B (es) * | 2010-02-25 | 2017-08-03 | Santen Pharmaceutical Co Ltd | Solucion oftalmica para tratar infeccion ocular que comprende levofloxacina o sal de la misma o solvato de la misma, metodo para tratar infeccion ocular, levofloxacina o sal de la misma o solvato de la misma, y uso de la misma. |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3711343A1 (de) * | 1987-04-03 | 1988-10-20 | Bayer Ag | Cephalosporinderivate, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
| MA24500A1 (fr) * | 1997-03-21 | 1998-10-01 | Lg Life Sciences Ltd | Derive du sel d'acide carboxylique de naphthyridine . |
| US6576224B1 (en) * | 1999-07-06 | 2003-06-10 | Sinuspharma, Inc. | Aerosolized anti-infectives, anti-inflammatories, and decongestants for the treatment of sinusitis |
-
2002
- 2002-11-29 DE DE60222298T patent/DE60222298T2/de not_active Expired - Lifetime
- 2002-11-29 US US10/496,809 patent/US7169792B2/en not_active Expired - Lifetime
- 2002-11-29 ES ES02795444T patent/ES2292844T3/es not_active Expired - Lifetime
- 2002-11-29 PT PT02795444T patent/PT1458391E/pt unknown
- 2002-11-29 CA CA002468036A patent/CA2468036C/en not_active Expired - Lifetime
- 2002-11-29 AU AU2002360218A patent/AU2002360218A1/en not_active Abandoned
- 2002-11-29 WO PCT/KR2002/002248 patent/WO2003045390A1/en active IP Right Grant
- 2002-11-29 EP EP02795444A patent/EP1458391B1/de not_active Expired - Lifetime
- 2002-11-29 MX MXPA04005179A patent/MXPA04005179A/es active IP Right Grant
- 2002-11-29 DK DK02795444T patent/DK1458391T3/da active
- 2002-11-29 AT AT02795444T patent/ATE372119T1/de active
-
2004
- 2004-06-28 NO NO20042711A patent/NO333196B1/no not_active IP Right Cessation
-
2007
- 2007-11-28 CY CY20071101521T patent/CY1107038T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA04005179A (es) | 2004-08-11 |
| EP1458391B1 (de) | 2007-09-05 |
| PT1458391E (pt) | 2007-12-10 |
| NO20042711L (no) | 2004-06-30 |
| WO2003045390A1 (en) | 2003-06-05 |
| CY1107038T1 (el) | 2012-09-26 |
| DE60222298T2 (de) | 2008-01-03 |
| EP1458391A1 (de) | 2004-09-22 |
| ATE372119T1 (de) | 2007-09-15 |
| DE60222298D1 (de) | 2007-10-18 |
| US20050148571A1 (en) | 2005-07-07 |
| CA2468036C (en) | 2008-01-22 |
| US7169792B2 (en) | 2007-01-30 |
| EP1458391A4 (de) | 2005-05-11 |
| DK1458391T3 (da) | 2008-01-07 |
| CA2468036A1 (en) | 2003-06-05 |
| ES2292844T3 (es) | 2008-03-16 |
| AU2002360218A1 (en) | 2003-06-10 |
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