NO325011B1 - Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter - Google Patents
Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter Download PDFInfo
- Publication number
- NO325011B1 NO325011B1 NO20030374A NO20030374A NO325011B1 NO 325011 B1 NO325011 B1 NO 325011B1 NO 20030374 A NO20030374 A NO 20030374A NO 20030374 A NO20030374 A NO 20030374A NO 325011 B1 NO325011 B1 NO 325011B1
- Authority
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- Norway
- Prior art keywords
- formula
- compound
- acid
- pharmaceutically acceptable
- alkyl
- Prior art date
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- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. Transmission Power Control [TPC] or power classes
- H04W52/04—Transmission power control [TPC]
- H04W52/06—TPC algorithms
- H04W52/14—Separate analysis of uplink or downlink
- H04W52/146—Uplink power control
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. Transmission Power Control [TPC] or power classes
- H04W52/04—Transmission power control [TPC]
- H04W52/18—TPC being performed according to specific parameters
- H04W52/24—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. Transmission Power Control [TPC] or power classes
- H04W52/04—Transmission power control [TPC]
- H04W52/18—TPC being performed according to specific parameters
- H04W52/28—TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission
- H04W52/288—TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission taking into account the usage mode, e.g. hands-free, data transmission or telephone
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W48/00—Access restriction; Network selection; Access point selection
- H04W48/20—Selecting an access point
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. Transmission Power Control [TPC] or power classes
- H04W52/04—Transmission power control [TPC]
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. Transmission Power Control [TPC] or power classes
- H04W52/04—Transmission power control [TPC]
- H04W52/18—TPC being performed according to specific parameters
- H04W52/24—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
- H04W52/245—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters taking into account received signal strength
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. Transmission Power Control [TPC] or power classes
- H04W52/04—Transmission power control [TPC]
- H04W52/18—TPC being performed according to specific parameters
- H04W52/24—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
- H04W52/247—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters where the output power of a terminal is based on a path parameter sent by another terminal
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- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Signal Processing (AREA)
- Computer Networks & Wireless Communication (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Computer Security & Cryptography (AREA)
- Quality & Reliability (AREA)
- Physics & Mathematics (AREA)
- Electromagnetism (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Steroid Compounds (AREA)
- Materials For Photolithography (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22068300P | 2000-07-25 | 2000-07-25 | |
| PCT/CA2001/001069 WO2002008186A2 (en) | 2000-07-25 | 2001-07-23 | Cyclopentanoindoles, compositions containing such compounds and methods of treatment |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20030374D0 NO20030374D0 (no) | 2003-01-24 |
| NO20030374L NO20030374L (no) | 2003-01-24 |
| NO325011B1 true NO325011B1 (no) | 2008-01-14 |
Family
ID=22824535
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20030374A NO325011B1 (no) | 2000-07-25 | 2003-01-24 | Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter |
Country Status (33)
| Country | Link |
|---|---|
| US (1) | US6410583B1 (cs) |
| EP (1) | EP1305286B1 (cs) |
| JP (1) | JP4119745B2 (cs) |
| KR (1) | KR100746814B1 (cs) |
| CN (1) | CN1214007C (cs) |
| AT (1) | ATE284388T1 (cs) |
| AU (2) | AU7743001A (cs) |
| BG (1) | BG66084B1 (cs) |
| BR (1) | BR0112756A (cs) |
| CA (1) | CA2416867C (cs) |
| CZ (1) | CZ2003236A3 (cs) |
| DE (1) | DE60107687T2 (cs) |
| DK (1) | DK1305286T3 (cs) |
| DZ (1) | DZ3402A1 (cs) |
| EA (1) | EA006765B1 (cs) |
| EC (1) | ECSP034428A (cs) |
| EE (1) | EE05287B1 (cs) |
| ES (1) | ES2231526T3 (cs) |
| GE (1) | GEP20053595B (cs) |
| HR (1) | HRP20021039B1 (cs) |
| HU (1) | HUP0301745A3 (cs) |
| IL (2) | IL153406A0 (cs) |
| IS (1) | IS2170B (cs) |
| MX (1) | MXPA03000710A (cs) |
| NO (1) | NO325011B1 (cs) |
| NZ (1) | NZ523106A (cs) |
| PL (1) | PL207342B1 (cs) |
| PT (1) | PT1305286E (cs) |
| RS (1) | RS50491B (cs) |
| SK (1) | SK287507B6 (cs) |
| UA (1) | UA73787C2 (cs) |
| WO (1) | WO2002008186A2 (cs) |
| ZA (1) | ZA200300554B (cs) |
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| US6784172B2 (en) | 2000-11-03 | 2004-08-31 | Wyeth | Processes for preparation of cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
| ES2230382T3 (es) * | 2000-11-03 | 2005-05-01 | Wyeth | Ciclopental(b)(1,4)diazpino(6,7,1-hi)indoles como antagonistas de 5ht2c. |
| US6858604B2 (en) | 2000-11-03 | 2005-02-22 | Wyeth | Cyclohepta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
| AR031197A1 (es) | 2000-11-03 | 2003-09-10 | Wyeth Corp | Procedimiento para la preparacion de derivados de 1,2,3,4,8,9,10,10a-octahidro-7bh-ciclopenta(b) diazepino(6,7,1-hi)indol |
| US6916922B2 (en) | 2000-11-03 | 2005-07-12 | Wyeth | Process for the preparation of 1,2,3,4,8,9,10,10a-octahydro-7bH-cyclopenta [B] [1,4] diazepino- [6,7,1-hi] indole derivatives |
| AR031200A1 (es) | 2000-11-03 | 2003-09-10 | Wyeth Corp | Cicloocta [b] [1,4] diazepino [6,7,1-hi] indoles y derivados |
| AR038136A1 (es) * | 2002-01-24 | 2004-12-29 | Merck Frosst Canada Inc | Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento |
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| TW200307540A (en) | 2002-04-25 | 2003-12-16 | Wyeth Corp | [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents |
| TWI312781B (en) | 2002-04-25 | 2009-08-01 | [1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents | |
| TW200400963A (en) | 2002-05-21 | 2004-01-16 | Wyeth Corp | R-enantiomers of pyranoindole derivatives and the use thereof for the treatment of hepatitis C virus infection or disease |
| TW200400818A (en) | 2002-05-21 | 2004-01-16 | Wyeth Corp | Method for the use of pyranoindole derivatives to treat infection with hepatitis C virus |
| AR041089A1 (es) * | 2003-05-15 | 2005-05-04 | Merck & Co Inc | Procedimiento y composiciones farmaceutiicas para tratar aterosclerosis, dislipidemias y afecciones relacionadas |
| US20070054951A1 (en) * | 2003-05-20 | 2007-03-08 | Lianhai Li | Fluoro-methanesulfonyl-substituted cycloalkanoindoles and their use as prostaglandin D2 antagonists |
| CN1805959A (zh) * | 2003-06-12 | 2006-07-19 | 麦克弗罗斯特加拿大有限公司 | 作为dp拮抗剂的环烷吡咯并吡啶 |
| WO2005013985A1 (en) * | 2003-08-07 | 2005-02-17 | Merck Sharp & Dohme Limited | Treatment for alzheimer's disease and related conditions |
| US20050107350A1 (en) * | 2003-08-22 | 2005-05-19 | Pharmacia Corporation | Method for the treatment or prevention of bone disorders with a cyclooxygenase-2 inhibitor alone and in combination with a bone disorder treatment agent and compositions therewith |
| PE20050483A1 (es) | 2003-10-31 | 2005-08-25 | Arena Pharm Inc | Derivados de tetrazol de formula (i), sus composiciones farmaceuticas y procesos para producir composiciones farmaceuticas |
| US7019022B2 (en) * | 2003-12-15 | 2006-03-28 | Merck Frosst Canada & Co. | Substituted tetrahydrocarbazole and cyclopentanoindole derivatives |
| JP5064216B2 (ja) | 2004-07-16 | 2012-10-31 | プロテオシス・アーゲー | 炎症性疾患用治療剤としての、ｐａｒｐ及びｓｉｒ調節活性を有するムスカリンアンタゴニスト |
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| KR20170044760A (ko) | 2008-07-23 | 2017-04-25 | 아레나 파마슈티칼스, 인크. | 자가면역성 및 염증성의 장애의 치료에 유용한 치환된 1,2,3,4-테트라히드로시클로펜타[ｂ]인돌-3-일)아세트산 유도체 |
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- 2001-07-23 EA EA200300171A patent/EA006765B1/ru not_active IP Right Cessation
- 2001-07-23 AU AU7743001A patent/AU7743001A/xx active Pending
- 2001-07-23 EP EP01955162A patent/EP1305286B1/en not_active Expired - Lifetime
- 2001-07-23 GE GE5105A patent/GEP20053595B/en unknown
- 2001-07-23 EE EEP200300033A patent/EE05287B1/xx not_active IP Right Cessation
- 2001-07-23 HU HU0301745A patent/HUP0301745A3/hu unknown
- 2001-07-23 DE DE60107687T patent/DE60107687T2/de not_active Expired - Lifetime
- 2001-07-23 MX MXPA03000710A patent/MXPA03000710A/es active IP Right Grant
- 2001-07-23 PL PL363168A patent/PL207342B1/pl not_active IP Right Cessation
- 2001-07-23 DZ DZ013402A patent/DZ3402A1/fr active
- 2001-07-23 IL IL15340601A patent/IL153406A0/xx active IP Right Grant
- 2001-07-23 SK SK93-2003A patent/SK287507B6/sk not_active IP Right Cessation
- 2001-07-23 KR KR1020037001117A patent/KR100746814B1/ko not_active Expired - Lifetime
- 2001-07-23 BR BR0112756-0A patent/BR0112756A/pt active Search and Examination
- 2001-07-23 PT PT01955162T patent/PT1305286E/pt unknown
- 2001-07-23 RS YUP-979/02A patent/RS50491B/sr unknown
- 2001-07-23 UA UA2003021565A patent/UA73787C2/uk unknown
- 2001-07-23 CZ CZ2003236A patent/CZ2003236A3/cs unknown
- 2001-07-23 JP JP2002514093A patent/JP4119745B2/ja not_active Expired - Fee Related
- 2001-07-23 AT AT01955162T patent/ATE284388T1/de active
- 2001-07-23 AU AU2001277430A patent/AU2001277430B2/en not_active Expired
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- 2001-07-23 DK DK01955162T patent/DK1305286T3/da active
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- 2001-07-23 ES ES01955162T patent/ES2231526T3/es not_active Expired - Lifetime
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Also Published As
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