NO325011B1 - Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter - Google Patents

Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter Download PDF

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Publication number
NO325011B1
NO325011B1 NO20030374A NO20030374A NO325011B1 NO 325011 B1 NO325011 B1 NO 325011B1 NO 20030374 A NO20030374 A NO 20030374A NO 20030374 A NO20030374 A NO 20030374A NO 325011 B1 NO325011 B1 NO 325011B1
Authority
NO
Norway
Prior art keywords
formula
compound
acid
pharmaceutically acceptable
alkyl
Prior art date
Application number
NO20030374A
Other languages
English (en)
Norwegian (no)
Other versions
NO20030374D0 (no
NO20030374L (no
Inventor
Claudio Sturino
Bruno Roy
Carl Berthelette
Michael Boyd
Nicolas Lachance
John Scheigetz
Marc Labelle
Original Assignee
Merck Canada Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Canada Inc filed Critical Merck Canada Inc
Publication of NO20030374D0 publication Critical patent/NO20030374D0/no
Publication of NO20030374L publication Critical patent/NO20030374L/no
Publication of NO325011B1 publication Critical patent/NO325011B1/no

Links

Classifications

    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/38TPC being performed in particular situations
    • H04W52/46TPC being performed in particular situations in multi-hop networks, e.g. wireless relay networks
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/94[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04BTRANSMISSION
    • H04B17/00Monitoring; Testing
    • H04B17/30Monitoring; Testing of propagation channels
    • H04B17/309Measuring or estimating channel quality parameters
    • H04B17/318Received signal strength
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W48/00Access restriction; Network selection; Access point selection
    • H04W48/02Access restriction performed under specific conditions
    • H04W48/04Access restriction performed under specific conditions based on user or terminal location or mobility data, e.g. moving direction, speed
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/06TPC algorithms
    • H04W52/14Separate analysis of uplink or downlink
    • H04W52/146Uplink power control
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/28TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission
    • H04W52/288TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission taking into account the usage mode, e.g. hands-free, data transmission or telephone
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W48/00Access restriction; Network selection; Access point selection
    • H04W48/20Selecting an access point
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • H04W52/245TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters taking into account received signal strength
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • H04W52/247TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters where the output power of a terminal is based on a path parameter sent by another terminal

Landscapes

  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Signal Processing (AREA)
  • Computer Networks & Wireless Communication (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Computer Security & Cryptography (AREA)
  • Quality & Reliability (AREA)
  • Physics & Mathematics (AREA)
  • Electromagnetism (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Steroid Compounds (AREA)
  • Materials For Photolithography (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
NO20030374A 2000-07-25 2003-01-24 Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter NO325011B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22068300P 2000-07-25 2000-07-25
PCT/CA2001/001069 WO2002008186A2 (en) 2000-07-25 2001-07-23 Cyclopentanoindoles, compositions containing such compounds and methods of treatment

Publications (3)

Publication Number Publication Date
NO20030374D0 NO20030374D0 (no) 2003-01-24
NO20030374L NO20030374L (no) 2003-01-24
NO325011B1 true NO325011B1 (no) 2008-01-14

Family

ID=22824535

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20030374A NO325011B1 (no) 2000-07-25 2003-01-24 Syklopentanoindoler, preparater som inneholder slike forbindelser og anvendelse derav for fremstilling av medikamenter

Country Status (33)

Country Link
US (1) US6410583B1 (cs)
EP (1) EP1305286B1 (cs)
JP (1) JP4119745B2 (cs)
KR (1) KR100746814B1 (cs)
CN (1) CN1214007C (cs)
AT (1) ATE284388T1 (cs)
AU (2) AU7743001A (cs)
BG (1) BG66084B1 (cs)
BR (1) BR0112756A (cs)
CA (1) CA2416867C (cs)
CZ (1) CZ2003236A3 (cs)
DE (1) DE60107687T2 (cs)
DK (1) DK1305286T3 (cs)
DZ (1) DZ3402A1 (cs)
EA (1) EA006765B1 (cs)
EC (1) ECSP034428A (cs)
EE (1) EE05287B1 (cs)
ES (1) ES2231526T3 (cs)
GE (1) GEP20053595B (cs)
HR (1) HRP20021039B1 (cs)
HU (1) HUP0301745A3 (cs)
IL (2) IL153406A0 (cs)
IS (1) IS2170B (cs)
MX (1) MXPA03000710A (cs)
NO (1) NO325011B1 (cs)
NZ (1) NZ523106A (cs)
PL (1) PL207342B1 (cs)
PT (1) PT1305286E (cs)
RS (1) RS50491B (cs)
SK (1) SK287507B6 (cs)
UA (1) UA73787C2 (cs)
WO (1) WO2002008186A2 (cs)
ZA (1) ZA200300554B (cs)

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Publication number Publication date
BR0112756A (pt) 2003-06-24
JP2004504380A (ja) 2004-02-12
EE200300033A (et) 2004-10-15
CA2416867A1 (en) 2002-01-31
BG107438A (bg) 2003-09-30
PT1305286E (pt) 2005-04-29
EA200300171A1 (ru) 2003-06-26
ES2231526T3 (es) 2005-05-16
SK932003A3 (en) 2003-06-03
HRP20021039A2 (en) 2004-10-31
AU7743001A (en) 2002-02-05
EP1305286B1 (en) 2004-12-08
SK287507B6 (sk) 2010-12-07
IS6655A (is) 2002-12-12
HUP0301745A3 (en) 2010-03-29
IL153406A0 (en) 2003-07-06
RS50491B (sr) 2010-03-02
HK1058934A1 (en) 2004-06-11
PL363168A1 (en) 2004-11-15
PL207342B1 (pl) 2010-12-31
WO2002008186A2 (en) 2002-01-31
HUP0301745A2 (hu) 2003-09-29
DZ3402A1 (fr) 2002-01-31
EP1305286A2 (en) 2003-05-02
CZ2003236A3 (cs) 2003-05-14
DK1305286T3 (da) 2005-03-14
CN1443165A (zh) 2003-09-17
YU97902A (sh) 2006-05-25
ECSP034428A (es) 2003-03-10
GEP20053595B (en) 2005-08-10
NZ523106A (en) 2005-01-28
US6410583B1 (en) 2002-06-25
EE05287B1 (et) 2010-04-15
HRP20021039B1 (hr) 2011-03-31
DE60107687D1 (de) 2005-01-13
IS2170B (is) 2006-11-15
EA006765B1 (ru) 2006-04-28
CA2416867C (en) 2008-03-25
NO20030374D0 (no) 2003-01-24
KR100746814B1 (ko) 2007-08-06
NO20030374L (no) 2003-01-24
KR20030024810A (ko) 2003-03-26
ATE284388T1 (de) 2004-12-15
AU2001277430B2 (en) 2006-05-25
JP4119745B2 (ja) 2008-07-16
UA73787C2 (en) 2005-09-15
BG66084B1 (bg) 2011-03-31
MXPA03000710A (es) 2003-06-04
IL153406A (en) 2008-03-20
WO2002008186A3 (en) 2002-03-21
ZA200300554B (en) 2004-04-23
CN1214007C (zh) 2005-08-10
DE60107687T2 (de) 2005-12-01

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