EE05287B1 - Tsklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon - Google Patents

Tsklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon

Info

Publication number
EE05287B1
EE05287B1 EEP200300033A EEP200300033A EE05287B1 EE 05287 B1 EE05287 B1 EE 05287B1 EE P200300033 A EEP200300033 A EE P200300033A EE P200300033 A EEP200300033 A EE P200300033A EE 05287 B1 EE05287 B1 EE 05287B1
Authority
EE
Estonia
Prior art keywords
clopentanoindoles
medicament
manufacture
called
pharmaceutical composition
Prior art date
Application number
EEP200300033A
Other languages
English (en)
Estonian (et)
Inventor
Labelle Marc
Sturino Claudio
Roy Bruno
Berthelette Carl
Boyd Michael
Lachance Nicolas
Scheigetz John
Original Assignee
Merck Frosst Canada & Co.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Frosst Canada & Co. filed Critical Merck Frosst Canada & Co.
Publication of EE200300033A publication Critical patent/EE200300033A/xx
Publication of EE05287B1 publication Critical patent/EE05287B1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/38TPC being performed in particular situations
    • H04W52/46TPC being performed in particular situations in multi-hop networks, e.g. wireless relay networks
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/94[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04BTRANSMISSION
    • H04B17/00Monitoring; Testing
    • H04B17/30Monitoring; Testing of propagation channels
    • H04B17/309Measuring or estimating channel quality parameters
    • H04B17/318Received signal strength
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W48/00Access restriction; Network selection; Access point selection
    • H04W48/02Access restriction performed under specific conditions
    • H04W48/04Access restriction performed under specific conditions based on user or terminal location or mobility data, e.g. moving direction, speed
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/06TPC algorithms
    • H04W52/14Separate analysis of uplink or downlink
    • H04W52/146Uplink power control
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/28TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission
    • H04W52/288TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission taking into account the usage mode, e.g. hands-free, data transmission or telephone
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W48/00Access restriction; Network selection; Access point selection
    • H04W48/20Selecting an access point
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • H04W52/245TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters taking into account received signal strength
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • H04W52/247TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters where the output power of a terminal is based on a path parameter sent by another terminal

Landscapes

  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Signal Processing (AREA)
  • Computer Networks & Wireless Communication (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Computer Security & Cryptography (AREA)
  • Quality & Reliability (AREA)
  • Physics & Mathematics (AREA)
  • Electromagnetism (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Materials For Photolithography (AREA)
EEP200300033A 2000-07-25 2001-07-23 Tsklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon EE05287B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22068300P 2000-07-25 2000-07-25
PCT/CA2001/001069 WO2002008186A2 (en) 2000-07-25 2001-07-23 Cyclopentanoindoles, compositions containing such compounds and methods of treatment

Publications (2)

Publication Number Publication Date
EE200300033A EE200300033A (et) 2004-10-15
EE05287B1 true EE05287B1 (et) 2010-04-15

Family

ID=22824535

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300033A EE05287B1 (et) 2000-07-25 2001-07-23 Tsklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon

Country Status (33)

Country Link
US (1) US6410583B1 (cs)
EP (1) EP1305286B1 (cs)
JP (1) JP4119745B2 (cs)
KR (1) KR100746814B1 (cs)
CN (1) CN1214007C (cs)
AT (1) ATE284388T1 (cs)
AU (2) AU2001277430B2 (cs)
BG (1) BG66084B1 (cs)
BR (1) BR0112756A (cs)
CA (1) CA2416867C (cs)
CZ (1) CZ2003236A3 (cs)
DE (1) DE60107687T2 (cs)
DK (1) DK1305286T3 (cs)
DZ (1) DZ3402A1 (cs)
EA (1) EA006765B1 (cs)
EC (1) ECSP034428A (cs)
EE (1) EE05287B1 (cs)
ES (1) ES2231526T3 (cs)
GE (1) GEP20053595B (cs)
HR (1) HRP20021039B1 (cs)
HU (1) HUP0301745A3 (cs)
IL (2) IL153406A0 (cs)
IS (1) IS2170B (cs)
MX (1) MXPA03000710A (cs)
NO (1) NO325011B1 (cs)
NZ (1) NZ523106A (cs)
PL (1) PL207342B1 (cs)
PT (1) PT1305286E (cs)
RS (1) RS50491B (cs)
SK (1) SK287507B6 (cs)
UA (1) UA73787C2 (cs)
WO (1) WO2002008186A2 (cs)
ZA (1) ZA200300554B (cs)

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AR031196A1 (es) 2000-11-03 2003-09-10 Wyeth Corp Procedimiento para la preparacion de ciclopenta (b) (1,4)-diazepino (6,7,1-hi) indoles y derivados
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US6858604B2 (en) 2000-11-03 2005-02-22 Wyeth Cyclohepta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
US6759405B2 (en) 2000-11-03 2004-07-06 Wyeth Cycloocta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
DE60106641T2 (de) * 2000-11-03 2005-12-01 Wyeth Cyclopenta[b][1,4] diazepino[6,7,1-hi]indole als 5ht2c antagonisten
AR038136A1 (es) * 2002-01-24 2004-12-29 Merck Frosst Canada Inc Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento
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Also Published As

Publication number Publication date
HK1058934A1 (en) 2004-06-11
JP2004504380A (ja) 2004-02-12
YU97902A (sh) 2006-05-25
NO20030374L (no) 2003-01-24
CA2416867A1 (en) 2002-01-31
NZ523106A (en) 2005-01-28
CZ2003236A3 (cs) 2003-05-14
US6410583B1 (en) 2002-06-25
IL153406A0 (en) 2003-07-06
RS50491B (sr) 2010-03-02
HRP20021039B1 (hr) 2011-03-31
WO2002008186A2 (en) 2002-01-31
EA200300171A1 (ru) 2003-06-26
ATE284388T1 (de) 2004-12-15
IS6655A (is) 2002-12-12
DE60107687D1 (de) 2005-01-13
IL153406A (en) 2008-03-20
KR100746814B1 (ko) 2007-08-06
NO20030374D0 (no) 2003-01-24
NO325011B1 (no) 2008-01-14
BR0112756A (pt) 2003-06-24
PL363168A1 (en) 2004-11-15
AU2001277430B2 (en) 2006-05-25
BG66084B1 (bg) 2011-03-31
ES2231526T3 (es) 2005-05-16
AU7743001A (en) 2002-02-05
CA2416867C (en) 2008-03-25
HRP20021039A2 (en) 2004-10-31
ZA200300554B (en) 2004-04-23
HUP0301745A2 (hu) 2003-09-29
EP1305286B1 (en) 2004-12-08
ECSP034428A (es) 2003-03-10
SK287507B6 (sk) 2010-12-07
GEP20053595B (en) 2005-08-10
HUP0301745A3 (en) 2010-03-29
WO2002008186A3 (en) 2002-03-21
MXPA03000710A (es) 2003-06-04
CN1214007C (zh) 2005-08-10
EE200300033A (et) 2004-10-15
PT1305286E (pt) 2005-04-29
CN1443165A (zh) 2003-09-17
DZ3402A1 (fr) 2002-01-31
EP1305286A2 (en) 2003-05-02
UA73787C2 (en) 2005-09-15
KR20030024810A (ko) 2003-03-26
IS2170B (is) 2006-11-15
EA006765B1 (ru) 2006-04-28
SK932003A3 (en) 2003-06-03
BG107438A (bg) 2003-09-30
JP4119745B2 (ja) 2008-07-16
DE60107687T2 (de) 2005-12-01
PL207342B1 (pl) 2010-12-31
DK1305286T3 (da) 2005-03-14

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