NO321062B1 - Krystallinske former av celecoksib, farmasoytisk sammensetning omfattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av samme. - Google Patents
Krystallinske former av celecoksib, farmasoytisk sammensetning omfattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av samme. Download PDFInfo
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- NO321062B1 NO321062B1 NO20013868A NO20013868A NO321062B1 NO 321062 B1 NO321062 B1 NO 321062B1 NO 20013868 A NO20013868 A NO 20013868A NO 20013868 A NO20013868 A NO 20013868A NO 321062 B1 NO321062 B1 NO 321062B1
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- celecoxib
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- cyclooxygenase
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Applications Claiming Priority (2)
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US16985699P | 1999-12-08 | 1999-12-08 | |
PCT/US2000/032760 WO2001042222A1 (en) | 1999-12-08 | 2000-12-01 | Polymorphic crystalline forms of celecoxib |
Publications (3)
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NO20013868D0 NO20013868D0 (no) | 2001-08-08 |
NO20013868L NO20013868L (no) | 2001-10-03 |
NO321062B1 true NO321062B1 (no) | 2006-03-06 |
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NO20013868A NO321062B1 (no) | 1999-12-08 | 2001-08-08 | Krystallinske former av celecoksib, farmasoytisk sammensetning omfattende samme, anvendelse av samme for fremstilling av medikament og fremgangsmate for fremstilling av samme. |
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EP (2) | EP1528058A1 (ru) |
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UA (1) | UA74539C2 (ru) |
WO (1) | WO2001042222A1 (ru) |
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TR200001872A3 (tr) | 2000-06-26 | 2002-01-21 | Fako Ilaclari A.S | 4-[5-(4-Metilfenil-3-(triflorometil)-1H-pirazol-1-il] benzensulfonamit' in yeni kristal biçimi "Biçim I" ve bu ürünün üretilmesine iliskin yöntem. |
US20030224006A1 (en) | 2002-03-01 | 2003-12-04 | Zaworotko Michael J. | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
WO2004078161A1 (en) | 2003-02-28 | 2004-09-16 | Transform Pharmaceuticals, Inc. | Pharmaceutical co-crystal compositions of drugs such as carbamazeptine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen |
US7790905B2 (en) | 2002-02-15 | 2010-09-07 | Mcneil-Ppc, Inc. | Pharmaceutical propylene glycol solvate compositions |
US7927613B2 (en) | 2002-02-15 | 2011-04-19 | University Of South Florida | Pharmaceutical co-crystal compositions |
AU2002251330A1 (en) * | 2002-04-25 | 2003-11-10 | Generics (Uk) Limited | Celecoxib forms |
AU2002251329A1 (en) * | 2002-04-25 | 2003-11-10 | Generics (Uk) Limited | Novel crystalline forms of celecoxib and other compounds |
US7968569B2 (en) * | 2002-05-17 | 2011-06-28 | Celgene Corporation | Methods for treatment of multiple myeloma using 3-(4-amino-1-oxo-1,3-dihydro-isoindol-2-yl)-piperidine-2,6-dione |
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CA2514733A1 (en) * | 2003-02-28 | 2004-09-16 | Transform Pharmaceuticals, Inc. | Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen |
AU2003264861A1 (en) * | 2003-08-08 | 2005-02-25 | Hetero Drugs Limited | Novel crystalline forms of celecoxib |
CA2574326A1 (en) * | 2004-07-22 | 2006-05-18 | Pliva-Istrazivanje I Razvoj D.O.O. | Novel form of celecoxib |
WO2006056770A1 (en) | 2004-11-23 | 2006-06-01 | Pliva Hrvatska D.O.O. | Extended release pharmaceutical composition of celecoxib |
JP2008528568A (ja) * | 2005-01-31 | 2008-07-31 | ファルマシア・アンド・アップジョン・カンパニー・エルエルシー | Iv型結晶のセレコキシブ |
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EP3208272B1 (en) | 2005-11-08 | 2020-01-08 | Vertex Pharmaceuticals Incorporated | Heterocyclic modulators of atp-binding cassette transporters |
EP2164840A2 (en) | 2007-05-09 | 2010-03-24 | Vertex Pharmaceuticals Incorporated | Modulators of cftr |
RS55559B1 (sr) | 2007-12-07 | 2017-05-31 | Vertex Pharma | Čvrste forme 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioksol-5-il)ciklopropankarboksamido)-3-metilpiridin-2-il) benzoeve kiseline |
EA201070700A1 (ru) | 2007-12-07 | 2011-06-30 | Вертекс Фармасьютикалз Инкорпорейтед | Способы получения циклоалкилкарбоксамидопиридинбензойных кислот |
JP5523352B2 (ja) | 2008-02-28 | 2014-06-18 | バーテックス ファーマシューティカルズ インコーポレイテッド | Cftr修飾因子としてのへテロアリール誘導体 |
JP2011527668A (ja) * | 2008-07-11 | 2011-11-04 | ビーエーエスエフ ソシエタス・ヨーロピア | 形態改質剤としての両親媒性タンパク質 |
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WO2011055233A2 (en) | 2009-11-03 | 2011-05-12 | Actavis Group Ptc Ehf | Improved process for preparing celecoxib polymorph |
US20110213159A1 (en) | 2010-03-01 | 2011-09-01 | Vamsee Krishna Muppidi | Process for preparation of celecoxib crystalline form |
NZ602838A (en) | 2010-04-07 | 2015-06-26 | Vertex Pharma | Pharmaceutical compositions of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid and administration thereof |
EP2468258A1 (en) | 2010-12-22 | 2012-06-27 | LEK Pharmaceuticals d.d. | Process for the preparation of a pharmaceutical composition comprising a low soluble pharmaceutically active ingredient |
CN103193677A (zh) * | 2013-03-22 | 2013-07-10 | 南开大学 | 美索巴莫磷酸二钠盐的多晶型及其制备方法 |
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- 2000-12-01 DZ DZ003140A patent/DZ3140A1/xx active
- 2000-12-01 EP EP05002575A patent/EP1528058A1/en not_active Withdrawn
- 2000-12-01 EP EP00983865A patent/EP1150960B1/en not_active Expired - Lifetime
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- 2000-12-01 JP JP2001543523A patent/JP2003516394A/ja not_active Withdrawn
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