NO310660B1 - Kondenserte tiazolderivater med 5-HT-reseptor-affinitet, anvendelse og fremstilling derav samt farmasöytisk blanding - Google Patents

Kondenserte tiazolderivater med 5-HT-reseptor-affinitet, anvendelse og fremstilling derav samt farmasöytisk blanding Download PDF

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Publication number
NO310660B1
NO310660B1 NO19976157A NO976157A NO310660B1 NO 310660 B1 NO310660 B1 NO 310660B1 NO 19976157 A NO19976157 A NO 19976157A NO 976157 A NO976157 A NO 976157A NO 310660 B1 NO310660 B1 NO 310660B1
Authority
NO
Norway
Prior art keywords
formula
compounds
mixture
compound
halogen
Prior art date
Application number
NO19976157A
Other languages
English (en)
Norwegian (no)
Other versions
NO976157D0 (no
NO976157L (no
Inventor
Frank Kerrigan
Sharon Crawford Cheetham
Roy Victor Davies
Original Assignee
Knoll Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Knoll Ag filed Critical Knoll Ag
Publication of NO976157D0 publication Critical patent/NO976157D0/no
Publication of NO976157L publication Critical patent/NO976157L/no
Publication of NO310660B1 publication Critical patent/NO310660B1/no

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/10Expectorants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
NO19976157A 1995-07-01 1997-12-30 Kondenserte tiazolderivater med 5-HT-reseptor-affinitet, anvendelse og fremstilling derav samt farmasöytisk blanding NO310660B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9513467.2A GB9513467D0 (en) 1995-07-01 1995-07-01 Therapeutic agents
PCT/EP1996/002676 WO1997002269A1 (en) 1995-07-01 1996-06-20 Condensed thiazole derivatives, having 5-ht receptor affinity

Publications (3)

Publication Number Publication Date
NO976157D0 NO976157D0 (no) 1997-12-30
NO976157L NO976157L (no) 1997-12-30
NO310660B1 true NO310660B1 (no) 2001-08-06

Family

ID=10777016

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19976157A NO310660B1 (no) 1995-07-01 1997-12-30 Kondenserte tiazolderivater med 5-HT-reseptor-affinitet, anvendelse og fremstilling derav samt farmasöytisk blanding

Country Status (30)

Country Link
US (1) US5869492A (ko)
EP (1) EP0836606B1 (ko)
JP (1) JPH11508568A (ko)
KR (1) KR19990028619A (ko)
CN (1) CN1064966C (ko)
AR (1) AR003963A1 (ko)
AT (1) ATE195942T1 (ko)
AU (1) AU708789B2 (ko)
BG (1) BG63206B1 (ko)
BR (1) BR9609525A (ko)
CA (1) CA2222725A1 (ko)
CO (1) CO4700463A1 (ko)
CZ (1) CZ376297A3 (ko)
DE (1) DE69610104T2 (ko)
DK (1) DK0836606T3 (ko)
ES (1) ES2151175T3 (ko)
GB (1) GB9513467D0 (ko)
GR (1) GR3034397T3 (ko)
HR (1) HRP960306B1 (ko)
HU (1) HUP9901258A3 (ko)
IL (1) IL122158A (ko)
NO (1) NO310660B1 (ko)
NZ (1) NZ312130A (ko)
PL (1) PL324337A1 (ko)
PT (1) PT836606E (ko)
SK (1) SK179297A3 (ko)
TR (1) TR199701756T1 (ko)
TW (1) TW474939B (ko)
WO (1) WO1997002269A1 (ko)
ZA (1) ZA965494B (ko)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9705428D0 (en) * 1997-03-15 1997-04-30 Knoll Ag Therapeutic agents
US6320060B1 (en) 1998-03-31 2001-11-20 Shionogi & Co., Ltd. Process for producing 5-hydroxybenzo[b] thiophene-3-carboxylic acid derivatives
DE19908536A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Polycyclische Thiazol-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
GB9911881D0 (en) * 1999-05-21 1999-07-21 Knoll Ag Therapeutic agents
GB9911863D0 (en) * 1999-05-21 1999-07-21 Knoll Ag Therapeutic agents
GB0005789D0 (en) * 2000-03-11 2000-05-03 Knoll Ag Therapeutic agents
GB0023610D0 (en) * 2000-09-27 2000-11-08 Knoll Ag Therapeutic agents
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
US8106074B2 (en) 2001-07-13 2012-01-31 Pierre Fabre Medicament Pyridin-2-yl-methylamine derivatives for treating opiate dependence

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002400A1 (fr) * 1977-11-24 1979-06-13 Synthelabo Dérivés de thiazole, leur préparation, intermédiaires et leur application en thérapeutique
PT672043E (pt) * 1992-07-13 2001-11-30 Janssen Pharmaceutica Nv Novos derivados de 4-(3-benzofuranil)piperidinilo e 4-(3-benzotienil)piperidinilo e composicoes farmaceuticas que os contem

Also Published As

Publication number Publication date
IL122158A (en) 2000-01-31
MX9709509A (es) 1998-03-29
GR3034397T3 (en) 2000-12-29
NO976157D0 (no) 1997-12-30
HUP9901258A3 (en) 2000-08-28
CA2222725A1 (en) 1997-01-23
PL324337A1 (en) 1998-05-25
IL122158A0 (en) 1998-04-05
CO4700463A1 (es) 1998-12-29
KR19990028619A (ko) 1999-04-15
EP0836606B1 (en) 2000-08-30
BR9609525A (pt) 1999-02-23
AR003963A1 (es) 1998-09-30
NO976157L (no) 1997-12-30
CN1064966C (zh) 2001-04-25
JPH11508568A (ja) 1999-07-27
DE69610104D1 (de) 2000-10-05
CN1189834A (zh) 1998-08-05
TW474939B (en) 2002-02-01
NZ312130A (en) 1999-08-30
BG63206B1 (bg) 2001-06-29
BG102084A (en) 1998-08-31
ZA965494B (en) 1997-12-29
WO1997002269A1 (en) 1997-01-23
CZ376297A3 (cs) 1998-06-17
GB9513467D0 (en) 1995-09-06
DK0836606T3 (da) 2000-11-20
US5869492A (en) 1999-02-09
HUP9901258A2 (hu) 1999-08-30
AU708789B2 (en) 1999-08-12
AU6358996A (en) 1997-02-05
ATE195942T1 (de) 2000-09-15
HRP960306B1 (en) 2001-08-31
SK179297A3 (en) 1998-07-08
DE69610104T2 (de) 2001-01-18
PT836606E (pt) 2001-02-28
EP0836606A1 (en) 1998-04-22
HRP960306A2 (en) 1998-04-30
TR199701756T1 (xx) 1998-04-21
ES2151175T3 (es) 2000-12-16

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