NO20091935L - Nye krystalliske former - Google Patents

Nye krystalliske former

Info

Publication number
NO20091935L
NO20091935L NO20091935A NO20091935A NO20091935L NO 20091935 L NO20091935 L NO 20091935L NO 20091935 A NO20091935 A NO 20091935A NO 20091935 A NO20091935 A NO 20091935A NO 20091935 L NO20091935 L NO 20091935L
Authority
NO
Norway
Prior art keywords
crystalline forms
new crystalline
aze
pab
compound
Prior art date
Application number
NO20091935A
Other languages
English (en)
Inventor
Bo Ingvar Ymen
Bengt Leonard Aslund
Stefan Bengtsson
Gudrun Anita Bergman
Ursula Renata Maria Hohlneicher
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39232767&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20091935(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20091935L publication Critical patent/NO20091935L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
  • Investigating Or Analyzing Materials Using Thermal Means (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Det er gitt krystallinske former av forbindelsene Ph(3-Cl)(5-OCHF2)-(R)CH(OH)C(O)-Aze-Pab(OMe) (Forbindelse A) og Ph(3-Cl)(5-OCHF2)-(R)CH(OH)C(O)-Aze-Pab(OH) (Forbindelse B), farmasøytiske preparater som inneholder dem, prosesser for å oppnå dem og anvendelse av dem i medisinsk behandling.
NO20091935A 2006-12-06 2009-05-19 Nye krystalliske former NO20091935L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86875206P 2006-12-06 2006-12-06
PCT/GB2007/004640 WO2008068475A1 (en) 2006-12-06 2007-12-05 New crystalline forms

Publications (1)

Publication Number Publication Date
NO20091935L true NO20091935L (no) 2009-07-03

Family

ID=39232767

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20091935A NO20091935L (no) 2006-12-06 2009-05-19 Nye krystalliske former

Country Status (24)

Country Link
US (1) US7820645B2 (no)
EP (1) EP2099750A1 (no)
JP (1) JP2010511684A (no)
KR (1) KR20090087107A (no)
CN (1) CN101553466B (no)
AR (1) AR064123A1 (no)
AU (1) AU2007330605B2 (no)
BR (1) BRPI0719908A2 (no)
CA (1) CA2670678A1 (no)
CL (1) CL2007003522A1 (no)
CO (1) CO6180434A2 (no)
EC (1) ECSP099389A (no)
IL (1) IL198864A0 (no)
MX (1) MX2009006036A (no)
MY (1) MY147634A (no)
NO (1) NO20091935L (no)
NZ (1) NZ577240A (no)
PE (1) PE20081445A1 (no)
RU (1) RU2446156C2 (no)
SA (1) SA07280675B1 (no)
TW (1) TW200827336A (no)
UA (1) UA97122C2 (no)
WO (1) WO2008068475A1 (no)
ZA (1) ZA200903614B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035216A1 (es) 2000-12-01 2004-05-05 Astrazeneca Ab Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
AR034517A1 (es) 2001-06-21 2004-02-25 Astrazeneca Ab Formulacion farmaceutica
SE0201661D0 (sv) * 2002-05-31 2002-05-31 Astrazeneca Ab New salts
US7781424B2 (en) * 2003-05-27 2010-08-24 Astrazeneca Ab Modified release pharmaceutical formulation
TW200900033A (en) * 2007-06-21 2009-01-01 Wen-Qing Li Automatic brewing machine
US20090061000A1 (en) * 2007-08-31 2009-03-05 Astrazeneca Ab Pharmaceutical formulation use 030
US9375678B2 (en) * 2012-05-25 2016-06-28 Georgia Tech Research Corporation Metal-organic framework supported on porous polymer
US9687791B2 (en) 2013-05-07 2017-06-27 Georgia Tech Research Corporation Flow processing and characterization of metal-organic framework (MOF) membranes in hollow fiber and tubular modules
US9994501B2 (en) 2013-05-07 2018-06-12 Georgia Tech Research Corporation High efficiency, high performance metal-organic framework (MOF) membranes in hollow fibers and tubular modules

Family Cites Families (68)

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TW201303B (no) 1990-07-05 1993-03-01 Hoffmann La Roche
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DK0629212T3 (da) 1992-03-04 1998-05-25 Gyogyszerkutato Intezet Antikoagulerende peptidderivater og farmaceutiske præparater indeholdende disse samt fremgangsmåde til fremstilling deraf.
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SE9301916D0 (sv) 1993-06-03 1993-06-03 Ab Astra New peptides derivatives
SE9301912D0 (sv) 1993-06-03 1993-06-03 Ab Astra Process for the production of aminoalkylguandines
US5780631A (en) 1993-06-03 1998-07-14 Astra Aktiebolag Starting materials in the synthesis of thrombin and kininogenase inhibitors
US6984627B1 (en) 1993-06-03 2006-01-10 Astrazeneca Ab Peptide derivatives
EP0648780A1 (en) 1993-08-26 1995-04-19 Bristol-Myers Squibb Company Heterocyclic thrombin inhibitors
TW394760B (en) 1993-09-07 2000-06-21 Hoffmann La Roche Novel Carboxamides, process for their preparation and pharmaceutical composition containing the same
AU1025795A (en) 1994-01-27 1995-08-03 Mitsubishi Chemical Corporation Prolineamide derivatives
US5707966A (en) 1994-03-04 1998-01-13 Eli Lilly And Company Antithrombotic agents
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SE0201661D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab New salts
SE0201658D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab Immediate release pharmaceutical formulation
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Also Published As

Publication number Publication date
JP2010511684A (ja) 2010-04-15
CN101553466B (zh) 2012-08-08
TW200827336A (en) 2008-07-01
ZA200903614B (en) 2010-03-31
EP2099750A1 (en) 2009-09-16
SA07280675B1 (ar) 2012-07-10
US20080287413A1 (en) 2008-11-20
RU2446156C2 (ru) 2012-03-27
PE20081445A1 (es) 2008-12-07
US7820645B2 (en) 2010-10-26
ECSP099389A (es) 2009-07-31
RU2009119411A (ru) 2011-01-20
CO6180434A2 (es) 2010-07-19
AU2007330605B2 (en) 2011-11-17
UA97122C2 (ru) 2012-01-10
CL2007003522A1 (es) 2008-08-22
WO2008068475A1 (en) 2008-06-12
KR20090087107A (ko) 2009-08-14
BRPI0719908A2 (pt) 2014-03-04
NZ577240A (en) 2011-11-25
CA2670678A1 (en) 2008-06-12
MX2009006036A (es) 2009-06-16
IL198864A0 (en) 2010-02-17
AU2007330605A1 (en) 2008-06-12
AR064123A1 (es) 2009-03-11
MY147634A (en) 2012-12-31
CN101553466A (zh) 2009-10-07

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application