AR064123A1 - Derivados cristalinos de azetidina. procesos de obtencion y usos. - Google Patents

Derivados cristalinos de azetidina. procesos de obtencion y usos.

Info

Publication number
AR064123A1
AR064123A1 ARP070105412A ARP070105412A AR064123A1 AR 064123 A1 AR064123 A1 AR 064123A1 AR P070105412 A ARP070105412 A AR P070105412A AR P070105412 A ARP070105412 A AR P070105412A AR 064123 A1 AR064123 A1 AR 064123A1
Authority
AR
Argentina
Prior art keywords
obtaining
processes
azetidine
derivatives
crystal
Prior art date
Application number
ARP070105412A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39232767&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR064123(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AR064123A1 publication Critical patent/AR064123A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
  • Investigating Or Analyzing Materials Using Thermal Means (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Procesos de obtencion, composiciones farmacéuticas que los contienen y uso como inhibidores de trombina. Reivindicacion 1: Una forma cristalina de un compuesto seleccionado de Ph(3-Cl)(5-OCHF2)-(R)CH(OH)C(O)-Aze-Pab(OMe) o Ph(3-Cl)(5-OCHF2)- (R)CH(OH)C(O)-Aze-Pab(OH).
ARP070105412A 2006-12-06 2007-12-04 Derivados cristalinos de azetidina. procesos de obtencion y usos. AR064123A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US86875206P 2006-12-06 2006-12-06

Publications (1)

Publication Number Publication Date
AR064123A1 true AR064123A1 (es) 2009-03-11

Family

ID=39232767

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070105412A AR064123A1 (es) 2006-12-06 2007-12-04 Derivados cristalinos de azetidina. procesos de obtencion y usos.

Country Status (24)

Country Link
US (1) US7820645B2 (es)
EP (1) EP2099750A1 (es)
JP (1) JP2010511684A (es)
KR (1) KR20090087107A (es)
CN (1) CN101553466B (es)
AR (1) AR064123A1 (es)
AU (1) AU2007330605B2 (es)
BR (1) BRPI0719908A2 (es)
CA (1) CA2670678A1 (es)
CL (1) CL2007003522A1 (es)
CO (1) CO6180434A2 (es)
EC (1) ECSP099389A (es)
IL (1) IL198864A0 (es)
MX (1) MX2009006036A (es)
MY (1) MY147634A (es)
NO (1) NO20091935L (es)
NZ (1) NZ577240A (es)
PE (1) PE20081445A1 (es)
RU (1) RU2446156C2 (es)
SA (1) SA07280675B1 (es)
TW (1) TW200827336A (es)
UA (1) UA97122C2 (es)
WO (1) WO2008068475A1 (es)
ZA (1) ZA200903614B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035216A1 (es) 2000-12-01 2004-05-05 Astrazeneca Ab Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
AR034517A1 (es) 2001-06-21 2004-02-25 Astrazeneca Ab Formulacion farmaceutica
SE0201661D0 (sv) * 2002-05-31 2002-05-31 Astrazeneca Ab New salts
US7781424B2 (en) * 2003-05-27 2010-08-24 Astrazeneca Ab Modified release pharmaceutical formulation
TW200900033A (en) * 2007-06-21 2009-01-01 Wen-Qing Li Automatic brewing machine
US20090061000A1 (en) * 2007-08-31 2009-03-05 Astrazeneca Ab Pharmaceutical formulation use 030
US9375678B2 (en) * 2012-05-25 2016-06-28 Georgia Tech Research Corporation Metal-organic framework supported on porous polymer
US9687791B2 (en) 2013-05-07 2017-06-27 Georgia Tech Research Corporation Flow processing and characterization of metal-organic framework (MOF) membranes in hollow fiber and tubular modules
US9994501B2 (en) 2013-05-07 2018-06-12 Georgia Tech Research Corporation High efficiency, high performance metal-organic framework (MOF) membranes in hollow fibers and tubular modules

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HU192646B (en) 1984-12-21 1987-06-29 Gyogyszerkutato Intezet Process for preparing new n-alkyl-peptide aldehydes
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Also Published As

Publication number Publication date
RU2009119411A (ru) 2011-01-20
PE20081445A1 (es) 2008-12-07
EP2099750A1 (en) 2009-09-16
SA07280675B1 (ar) 2012-07-10
WO2008068475A1 (en) 2008-06-12
ZA200903614B (en) 2010-03-31
US7820645B2 (en) 2010-10-26
AU2007330605A1 (en) 2008-06-12
MY147634A (en) 2012-12-31
UA97122C2 (ru) 2012-01-10
TW200827336A (en) 2008-07-01
ECSP099389A (es) 2009-07-31
US20080287413A1 (en) 2008-11-20
CA2670678A1 (en) 2008-06-12
CO6180434A2 (es) 2010-07-19
RU2446156C2 (ru) 2012-03-27
CN101553466A (zh) 2009-10-07
NZ577240A (en) 2011-11-25
JP2010511684A (ja) 2010-04-15
CN101553466B (zh) 2012-08-08
KR20090087107A (ko) 2009-08-14
MX2009006036A (es) 2009-06-16
IL198864A0 (en) 2010-02-17
BRPI0719908A2 (pt) 2014-03-04
CL2007003522A1 (es) 2008-08-22
AU2007330605B2 (en) 2011-11-17
NO20091935L (no) 2009-07-03

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