ZA200903614B - New crystalline forms - Google Patents

New crystalline forms

Info

Publication number
ZA200903614B
ZA200903614B ZA200903614A ZA200903614A ZA200903614B ZA 200903614 B ZA200903614 B ZA 200903614B ZA 200903614 A ZA200903614 A ZA 200903614A ZA 200903614 A ZA200903614 A ZA 200903614A ZA 200903614 B ZA200903614 B ZA 200903614B
Authority
ZA
South Africa
Prior art keywords
crystalline forms
new crystalline
new
forms
crystalline
Prior art date
Application number
ZA200903614A
Other languages
English (en)
Inventor
Bengt Leonard Aslund
Stefan Bengtsson
Gudrun Anita Bergman
Ursula Renata Maria Hohlneicher
Bo Ingvar Ymen
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39232767&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200903614(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ZA200903614B publication Critical patent/ZA200903614B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
  • Investigating Or Analyzing Materials Using Thermal Means (AREA)
ZA200903614A 2006-12-06 2009-05-25 New crystalline forms ZA200903614B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US86875206P 2006-12-06 2006-12-06

Publications (1)

Publication Number Publication Date
ZA200903614B true ZA200903614B (en) 2010-03-31

Family

ID=39232767

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200903614A ZA200903614B (en) 2006-12-06 2009-05-25 New crystalline forms

Country Status (24)

Country Link
US (1) US7820645B2 (xx)
EP (1) EP2099750A1 (xx)
JP (1) JP2010511684A (xx)
KR (1) KR20090087107A (xx)
CN (1) CN101553466B (xx)
AR (1) AR064123A1 (xx)
AU (1) AU2007330605B2 (xx)
BR (1) BRPI0719908A2 (xx)
CA (1) CA2670678A1 (xx)
CL (1) CL2007003522A1 (xx)
CO (1) CO6180434A2 (xx)
EC (1) ECSP099389A (xx)
IL (1) IL198864A0 (xx)
MX (1) MX2009006036A (xx)
MY (1) MY147634A (xx)
NO (1) NO20091935L (xx)
NZ (1) NZ577240A (xx)
PE (1) PE20081445A1 (xx)
RU (1) RU2446156C2 (xx)
SA (1) SA07280675B1 (xx)
TW (1) TW200827336A (xx)
UA (1) UA97122C2 (xx)
WO (1) WO2008068475A1 (xx)
ZA (1) ZA200903614B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035216A1 (es) * 2000-12-01 2004-05-05 Astrazeneca Ab Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
AR034517A1 (es) 2001-06-21 2004-02-25 Astrazeneca Ab Formulacion farmaceutica
SE0201661D0 (sv) * 2002-05-31 2002-05-31 Astrazeneca Ab New salts
US7781424B2 (en) * 2003-05-27 2010-08-24 Astrazeneca Ab Modified release pharmaceutical formulation
TW200900033A (en) * 2007-06-21 2009-01-01 Wen-Qing Li Automatic brewing machine
US20090061000A1 (en) * 2007-08-31 2009-03-05 Astrazeneca Ab Pharmaceutical formulation use 030
US9375678B2 (en) * 2012-05-25 2016-06-28 Georgia Tech Research Corporation Metal-organic framework supported on porous polymer
US9994501B2 (en) 2013-05-07 2018-06-12 Georgia Tech Research Corporation High efficiency, high performance metal-organic framework (MOF) membranes in hollow fibers and tubular modules
US9687791B2 (en) 2013-05-07 2017-06-27 Georgia Tech Research Corporation Flow processing and characterization of metal-organic framework (MOF) membranes in hollow fiber and tubular modules

Family Cites Families (68)

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HU192646B (en) 1984-12-21 1987-06-29 Gyogyszerkutato Intezet Process for preparing new n-alkyl-peptide aldehydes
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ZA897515B (en) 1988-10-07 1990-06-27 Merrell Dow Pharma Novel peptidase inhibitors
IT1229491B (it) 1988-12-28 1991-09-03 Roussel Maestretti S P A Ora R Derivati della 1,2,5,6-tetraidropiridina, loro procedimento di preparazione e loro impiego come sostanze medicinali
TW201303B (xx) 1990-07-05 1993-03-01 Hoffmann La Roche
CA2075154A1 (en) 1991-08-06 1993-02-07 Neelakantan Balasubramanian Peptide aldehydes as antithrombotic agents
SE9102462D0 (sv) 1991-08-28 1991-08-28 Astra Ab New isosteric peptides
US5169638A (en) 1991-10-23 1992-12-08 E. R. Squibb & Sons, Inc. Buoyant controlled release powder formulation
NZ245039A (en) 1991-11-12 1994-12-22 Lilly Co Eli N-phenylalanyl and n-phenylglycyl derivatives of the dipeptide of l-azetidine-2-carboxylic acid and l-arginine aldehyde; anti-blood clotting compositions
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CA2131367A1 (en) 1992-03-04 1993-09-16 Sandor Bajusz New anticoagulant peptide derivatives and pharmaceutical compositions containing the same as well as a process for the preparation thereof
TW223629B (xx) 1992-03-06 1994-05-11 Hoffmann La Roche
SE9301912D0 (sv) 1993-06-03 1993-06-03 Ab Astra Process for the production of aminoalkylguandines
US5783563A (en) 1993-06-03 1998-07-21 Astra Aktiebolag Method for treatment or prophylaxis of venous thrombosis
SE9301916D0 (sv) 1993-06-03 1993-06-03 Ab Astra New peptides derivatives
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EP0648780A1 (en) 1993-08-26 1995-04-19 Bristol-Myers Squibb Company Heterocyclic thrombin inhibitors
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US5707966A (en) 1994-03-04 1998-01-13 Eli Lilly And Company Antithrombotic agents
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US5561146A (en) 1994-06-10 1996-10-01 Bristol-Myers Squibb Company Modified guanidino and amidino thrombin inhibitors
DE4421052A1 (de) 1994-06-17 1995-12-21 Basf Ag Neue Thrombininhibitoren, ihre Herstellung und Verwendung
US5498724A (en) 1994-06-28 1996-03-12 Aktiebolaget Astra Pyrazoleamidine compounds
US5510369A (en) 1994-07-22 1996-04-23 Merck & Co., Inc. Pyrrolidine thrombin inhibitors
NZ302649A (en) 1995-02-17 2000-01-28 Basf Ag Dipeptide amidine derivatives, preparation and pharmaceutical compositions thereof
US5710130A (en) 1995-02-27 1998-01-20 Eli Lilly And Company Antithrombotic agents
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SA96170106A (ar) 1995-07-06 2005-12-03 أسترا أكتيبولاج مشتقات حامض أميني جديدة
TWI238827B (en) 1995-12-21 2005-09-01 Astrazeneca Ab Prodrugs of thrombin inhibitors
SE9601556D0 (sv) 1996-04-24 1996-04-24 Astra Ab New pharmaceutical formulation of a thrombin inhibitor for parenteral use
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AR035216A1 (es) * 2000-12-01 2004-05-05 Astrazeneca Ab Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
US6287599B1 (en) 2000-12-20 2001-09-11 Shire Laboratories, Inc. Sustained release pharmaceutical dosage forms with minimized pH dependent dissolution profiles
AR034517A1 (es) 2001-06-21 2004-02-25 Astrazeneca Ab Formulacion farmaceutica
US6811794B2 (en) 2001-12-20 2004-11-02 Shire Laboratories, Inc. Sustained release pharmaceutical dosage forms with minimized pH dependent dissolution profiles
SE0201658D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab Immediate release pharmaceutical formulation
SE0201661D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab New salts
SE0201659D0 (sv) 2002-05-31 2002-05-31 Astrazeneca Ab Modified release pharmaceutical formulation
US7781424B2 (en) 2003-05-27 2010-08-24 Astrazeneca Ab Modified release pharmaceutical formulation
SE0303220D0 (sv) 2003-11-28 2003-11-28 Astrazeneca Ab New process
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GB0510546D0 (en) 2005-05-24 2005-06-29 Astrazeneca Ab New process

Also Published As

Publication number Publication date
AR064123A1 (es) 2009-03-11
RU2009119411A (ru) 2011-01-20
AU2007330605B2 (en) 2011-11-17
IL198864A0 (en) 2010-02-17
US7820645B2 (en) 2010-10-26
PE20081445A1 (es) 2008-12-07
JP2010511684A (ja) 2010-04-15
KR20090087107A (ko) 2009-08-14
SA07280675B1 (ar) 2012-07-10
AU2007330605A1 (en) 2008-06-12
NO20091935L (no) 2009-07-03
CA2670678A1 (en) 2008-06-12
ECSP099389A (es) 2009-07-31
CN101553466A (zh) 2009-10-07
WO2008068475A1 (en) 2008-06-12
EP2099750A1 (en) 2009-09-16
UA97122C2 (ru) 2012-01-10
TW200827336A (en) 2008-07-01
RU2446156C2 (ru) 2012-03-27
CN101553466B (zh) 2012-08-08
MX2009006036A (es) 2009-06-16
US20080287413A1 (en) 2008-11-20
MY147634A (en) 2012-12-31
CL2007003522A1 (es) 2008-08-22
CO6180434A2 (es) 2010-07-19
NZ577240A (en) 2011-11-25
BRPI0719908A2 (pt) 2014-03-04

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