NO20081086L - Makrosykliske peptider som HCV NS3-proteaseinhibitorer - Google Patents
Makrosykliske peptider som HCV NS3-proteaseinhibitorerInfo
- Publication number
- NO20081086L NO20081086L NO20081086A NO20081086A NO20081086L NO 20081086 L NO20081086 L NO 20081086L NO 20081086 A NO20081086 A NO 20081086A NO 20081086 A NO20081086 A NO 20081086A NO 20081086 L NO20081086 L NO 20081086L
- Authority
- NO
- Norway
- Prior art keywords
- hcv
- protease inhibitors
- macrocyclic peptides
- protease
- macrocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/12—Cyclic peptides with only normal peptide bonds in the ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/06—Tripeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70425605P | 2005-08-01 | 2005-08-01 | |
US72450905P | 2005-10-07 | 2005-10-07 | |
PCT/US2006/029635 WO2007016441A1 (fr) | 2005-08-01 | 2006-07-28 | Peptides macrocycliques en tant qu’inhibiteurs de la protéase ns3 du vhc |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20081086L true NO20081086L (no) | 2008-04-30 |
Family
ID=37404447
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20081086A NO20081086L (no) | 2005-08-01 | 2008-02-29 | Makrosykliske peptider som HCV NS3-proteaseinhibitorer |
Country Status (16)
Country | Link |
---|---|
US (1) | US8278322B2 (fr) |
EP (1) | EP1913016B1 (fr) |
JP (1) | JP4705984B2 (fr) |
KR (1) | KR20080036598A (fr) |
AU (1) | AU2006275605B2 (fr) |
BR (1) | BRPI0614205A2 (fr) |
CA (1) | CA2615896C (fr) |
CR (1) | CR9731A (fr) |
EC (1) | ECSP088157A (fr) |
IL (1) | IL189166A0 (fr) |
MA (1) | MA29757B1 (fr) |
MX (1) | MX2008001588A (fr) |
NO (1) | NO20081086L (fr) |
NZ (1) | NZ565269A (fr) |
RU (1) | RU2008107972A (fr) |
WO (1) | WO2007016441A1 (fr) |
Families Citing this family (88)
Publication number | Priority date | Publication date | Assignee | Title |
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MY140680A (en) | 2002-05-20 | 2010-01-15 | Bristol Myers Squibb Co | Hepatitis c virus inhibitors |
WO2006119061A2 (fr) | 2005-05-02 | 2006-11-09 | Merck & Co., Inc. | Inhibiteurs de la protease ns3 du vhc |
KR101269568B1 (ko) * | 2005-07-04 | 2013-06-04 | 자난 사이텍 컴퍼니 리미티드 | 루테늄 착물 리간드, 루테늄 착물, 고정 루테늄 착물 촉매및 그의 제조방법과 용도 |
RU2008107972A (ru) | 2005-08-01 | 2009-09-10 | Мерк энд Ко., Инк. (US) | Макроциклические пептиды в качестве ингибиторов ns3-протеазы hcv |
US7741281B2 (en) | 2005-11-03 | 2010-06-22 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
GB0609492D0 (en) * | 2006-05-15 | 2006-06-21 | Angeletti P Ist Richerche Bio | Therapeutic agents |
GB0612423D0 (en) * | 2006-06-23 | 2006-08-02 | Angeletti P Ist Richerche Bio | Therapeutic agents |
US7935670B2 (en) | 2006-07-11 | 2011-05-03 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
US8138164B2 (en) | 2006-10-24 | 2012-03-20 | Merck Sharp & Dohme Corp. | HCV NS3 protease inhibitors |
AU2007309546A1 (en) | 2006-10-24 | 2008-05-02 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. | HCV NS3 protease inhibitors |
US8309540B2 (en) | 2006-10-24 | 2012-11-13 | Merck Sharp & Dohme Corp. | HCV NS3 protease inhibitors |
WO2008057209A1 (fr) * | 2006-10-27 | 2008-05-15 | Merck & Co., Inc. | Inhibiteurs de protéase ns3 du vhc |
WO2008057208A2 (fr) * | 2006-10-27 | 2008-05-15 | Merck & Co., Inc. | Inhibiteurs de protéase ns3 du vhc |
US8343477B2 (en) | 2006-11-01 | 2013-01-01 | Bristol-Myers Squibb Company | Inhibitors of hepatitis C virus |
US7772180B2 (en) | 2006-11-09 | 2010-08-10 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
US7763584B2 (en) | 2006-11-16 | 2010-07-27 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
US8003604B2 (en) | 2006-11-16 | 2011-08-23 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
US7888464B2 (en) | 2006-11-16 | 2011-02-15 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
GB0625349D0 (en) | 2006-12-20 | 2007-01-31 | Angeletti P Ist Richerche Bio | Therapeutic compounds |
AU2007335962B2 (en) | 2006-12-20 | 2012-09-06 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa | Antiviral indoles |
GB0625345D0 (en) | 2006-12-20 | 2007-01-31 | Angeletti P Ist Richerche Bio | Therapeutic compounds |
US20100143886A1 (en) | 2007-03-09 | 2010-06-10 | Ludmerer Steven W | In vivo hcv resistance to anti-viral inhibitors |
CA2693537C (fr) | 2007-07-17 | 2013-06-25 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa | Derives macrocycliques d'indole pour le traitement des infections d'hepatite c |
CA2699891C (fr) * | 2007-07-19 | 2013-10-22 | Nigel Liverton | Composes macrocycliques servant d'agents antiviraux |
US8383583B2 (en) | 2007-10-26 | 2013-02-26 | Enanta Pharmaceuticals, Inc. | Macrocyclic, pyridazinone-containing hepatitis C serine protease inhibitors |
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2006
- 2006-07-28 RU RU2008107972/04A patent/RU2008107972A/ru not_active Application Discontinuation
- 2006-07-28 WO PCT/US2006/029635 patent/WO2007016441A1/fr active Application Filing
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- 2006-07-28 EP EP06800513A patent/EP1913016B1/fr active Active
- 2006-07-28 KR KR1020087002861A patent/KR20080036598A/ko not_active Application Discontinuation
- 2006-07-28 JP JP2008525069A patent/JP4705984B2/ja not_active Expired - Fee Related
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- 2006-07-28 CA CA2615896A patent/CA2615896C/fr not_active Expired - Fee Related
- 2006-07-28 US US11/989,886 patent/US8278322B2/en active Active
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Also Published As
Publication number | Publication date |
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WO2007016441A1 (fr) | 2007-02-08 |
CA2615896C (fr) | 2012-11-13 |
US20110028494A1 (en) | 2011-02-03 |
CR9731A (es) | 2008-04-10 |
AU2006275605A1 (en) | 2007-02-08 |
ECSP088157A (es) | 2008-02-20 |
EP1913016B1 (fr) | 2013-01-16 |
CA2615896A1 (fr) | 2007-02-08 |
NZ565269A (en) | 2010-03-26 |
EP1913016A1 (fr) | 2008-04-23 |
BRPI0614205A2 (pt) | 2016-11-22 |
JP2009503080A (ja) | 2009-01-29 |
MX2008001588A (es) | 2008-02-19 |
IL189166A0 (en) | 2008-08-07 |
US8278322B2 (en) | 2012-10-02 |
MA29757B1 (fr) | 2008-09-01 |
RU2008107972A (ru) | 2009-09-10 |
KR20080036598A (ko) | 2008-04-28 |
JP4705984B2 (ja) | 2011-06-22 |
AU2006275605B2 (en) | 2011-01-06 |
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