NO20072352L - Forbindelser og sammensetninger som inhibitorer av cannabinoidreceptor 1-aktivitet - Google Patents

Forbindelser og sammensetninger som inhibitorer av cannabinoidreceptor 1-aktivitet

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Publication number
NO20072352L
NO20072352L NO20072352A NO20072352A NO20072352L NO 20072352 L NO20072352 L NO 20072352L NO 20072352 A NO20072352 A NO 20072352A NO 20072352 A NO20072352 A NO 20072352A NO 20072352 L NO20072352 L NO 20072352L
Authority
NO
Norway
Prior art keywords
compounds
activity
inhibitors
compositions
cannabinoid receptor
Prior art date
Application number
NO20072352A
Other languages
English (en)
Norwegian (no)
Inventor
Hong Liu
Xiaohui He
Ha-Soon Choi
Kunyong Yang
David Woodmansee
Zhicheng Wang
David Archer Ellis
Baogen Wu
Yun He
Truc Ngoc Nguyen
Original Assignee
Irm Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Irm Llc filed Critical Irm Llc
Publication of NO20072352L publication Critical patent/NO20072352L/no

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    • C07D473/18Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07D473/28Oxygen atom
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    • C07D473/32Nitrogen atom
    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine
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NO20072352A 2004-10-26 2007-05-07 Forbindelser og sammensetninger som inhibitorer av cannabinoidreceptor 1-aktivitet NO20072352L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62250804P 2004-10-26 2004-10-26
US67267005P 2005-04-18 2005-04-18
PCT/US2005/038361 WO2006047516A2 (en) 2004-10-26 2005-10-26 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity

Publications (1)

Publication Number Publication Date
NO20072352L true NO20072352L (no) 2007-05-31

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NO20072352A NO20072352L (no) 2004-10-26 2007-05-07 Forbindelser og sammensetninger som inhibitorer av cannabinoidreceptor 1-aktivitet

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US (2) US8158634B2 (ko)
EP (1) EP1807429A4 (ko)
JP (2) JP2008518016A (ko)
KR (1) KR100919524B1 (ko)
CN (2) CN101048408B (ko)
AR (1) AR051596A1 (ko)
AU (2) AU2005299421B2 (ko)
BR (1) BRPI0517015A (ko)
CA (2) CA2581225C (ko)
EC (1) ECSP077421A (ko)
IL (1) IL182527A0 (ko)
MA (1) MA28937B1 (ko)
MX (1) MX2007004936A (ko)
NO (1) NO20072352L (ko)
PE (1) PE20060599A1 (ko)
RU (1) RU2431635C2 (ko)
TN (1) TNSN07161A1 (ko)
TW (1) TW200630096A (ko)
WO (1) WO2006047516A2 (ko)

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NZ540612A (en) 2003-01-14 2008-02-29 Arena Pharm Inc 1,2,3-Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
AU2004257267B2 (en) 2003-07-14 2009-12-03 Arena Pharmaceuticals,Inc Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
JP2007519754A (ja) * 2004-01-30 2007-07-19 スミスクライン ビーチャム コーポレーション 化合物
AR051596A1 (es) * 2004-10-26 2007-01-24 Irm Llc Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios
GB0506147D0 (en) * 2005-03-24 2005-05-04 Merck Sharp & Dohme Therapeutic agents
JP2009536608A (ja) * 2005-05-11 2009-10-15 メルク シャープ エンド ドーム リミテッド バニロイド−1受容体(vr1)の機能を調節する2,3−置換縮合二環式ピリミジン4−(3h)−オン
JP2008543968A (ja) * 2005-06-28 2008-12-04 オーキッド リサーチ ラボラトリーズ リミテッド 新規なピラゾロピリミジノン誘導体
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