NO20071095L - Hittil ukjente tiofenderivater - Google Patents

Hittil ukjente tiofenderivater

Info

Publication number
NO20071095L
NO20071095L NO20071095A NO20071095A NO20071095L NO 20071095 L NO20071095 L NO 20071095L NO 20071095 A NO20071095 A NO 20071095A NO 20071095 A NO20071095 A NO 20071095A NO 20071095 L NO20071095 L NO 20071095L
Authority
NO
Norway
Prior art keywords
thiophene derivatives
hitherto unknown
derivatives
hitherto
unknown
Prior art date
Application number
NO20071095A
Other languages
English (en)
Norwegian (no)
Inventor
Martin Bolli
Thomas Weller
Walter Fischli
Martine Clozel
Oliver Nayler
Daniel Bur
Claus Mueller
Michael Scherz
David Lehmann
Boris Mathys
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of NO20071095L publication Critical patent/NO20071095L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/78Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/14Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Transplantation (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO20071095A 2004-07-29 2007-02-27 Hittil ukjente tiofenderivater NO20071095L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/EP2004/008501 WO2006010379A1 (en) 2004-07-29 2004-07-29 Novel thiophene derivatives as immunosuppressive agents
PCT/EP2005/007892 WO2006010544A2 (en) 2004-07-29 2005-07-20 1, 1a, 5, 5a-tetrahydro-3-thia-cyclopropa’a! pentalenes: tricyclic thiophene derivatives as s1p1/edg1 receptor agonists

Publications (1)

Publication Number Publication Date
NO20071095L true NO20071095L (no) 2007-02-27

Family

ID=34958296

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071095A NO20071095L (no) 2004-07-29 2007-02-27 Hittil ukjente tiofenderivater

Country Status (23)

Country Link
US (1) US7750040B2 (de)
EP (1) EP1805163B1 (de)
JP (1) JP4807884B2 (de)
KR (1) KR20070046849A (de)
CN (1) CN1993346B (de)
AR (1) AR050273A1 (de)
AT (1) ATE409697T1 (de)
AU (1) AU2005266529A1 (de)
BR (1) BRPI0513841A (de)
CA (1) CA2574305A1 (de)
DE (1) DE602005010109D1 (de)
DK (1) DK1805163T3 (de)
ES (1) ES2313391T3 (de)
IL (1) IL180962A0 (de)
MX (1) MX2007000972A (de)
NO (1) NO20071095L (de)
PL (1) PL1805163T3 (de)
PT (1) PT1805163E (de)
RU (1) RU2386626C2 (de)
SI (1) SI1805163T1 (de)
TW (1) TW200616994A (de)
WO (2) WO2006010379A1 (de)
ZA (1) ZA200700535B (de)

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AU2006226022A1 (en) 2005-03-23 2006-09-28 Actelion Pharmaceuticals Ltd. Novel thiophene derivatives as sphingosine-1-phosphate-1 receptor agonists
WO2006100633A1 (en) 2005-03-23 2006-09-28 Actelion Pharmaceuticals Ltd NOVEL THIOPHENE DERIVATIVES AS SPHINGOSINE-l-PHOSPHATE-1 RECEPTOR AGONISTS
EP1863787B1 (de) * 2005-03-23 2011-05-25 Actelion Pharmaceuticals Ltd. Hydrierte benzo[c]thiophenderivate als immunmodulatoren
BRPI0611631A2 (pt) * 2005-06-24 2010-09-21 Actelion Pharmaceuticals Ltd composto, composição farmacêutica, e, uso de um composto
AR057894A1 (es) * 2005-11-23 2007-12-26 Actelion Pharmaceuticals Ltd Derivados de tiofeno
TWI404706B (zh) * 2006-01-11 2013-08-11 Actelion Pharmaceuticals Ltd 新穎噻吩衍生物
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EP2069335B1 (de) * 2006-09-08 2012-12-26 Actelion Pharmaceuticals Ltd. Pyridin-3-yl-derivate als immunmodulatoren
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EP2262799B1 (de) * 2008-03-06 2012-07-04 Actelion Pharmaceuticals Ltd. Pyridinverbindungen
US8575200B2 (en) * 2008-03-07 2013-11-05 Actelion Pharmaceuticals Ltd Pyridin-2-yl derivatives as immunomodulating agents
SI2278960T2 (sl) 2008-03-17 2020-02-28 Actelion Pharmaceuticals Ltd. Režim odmerjanja za selektivni agonist receptorja sip1
JP5449346B2 (ja) 2008-07-15 2014-03-19 サノフイ Edg−1受容体アゴニストとしてのオキサゾロピリミジン類
CN104311472B9 (zh) 2008-07-23 2020-03-17 艾尼纳制药公司 经取代的1,2,3,4-四氢环戊并[b]吲哚-3-基乙酸衍生物
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DE202014011050U1 (de) 2014-11-05 2017-07-26 Carl Zeiss Meditec Ag Vorrichtung für das Untersuchen eines Patientenauges
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Also Published As

Publication number Publication date
PT1805163E (pt) 2008-12-05
WO2006010544A3 (en) 2006-03-30
BRPI0513841A (pt) 2008-05-20
US7750040B2 (en) 2010-07-06
PL1805163T3 (pl) 2009-04-30
EP1805163A2 (de) 2007-07-11
WO2006010379A1 (en) 2006-02-02
DK1805163T3 (da) 2008-12-15
AU2005266529A1 (en) 2006-02-02
JP2008508210A (ja) 2008-03-21
ATE409697T1 (de) 2008-10-15
DE602005010109D1 (de) 2008-11-13
CN1993346A (zh) 2007-07-04
US20080064740A1 (en) 2008-03-13
KR20070046849A (ko) 2007-05-03
MX2007000972A (es) 2007-04-10
AR050273A1 (es) 2006-10-11
CN1993346B (zh) 2011-04-27
EP1805163B1 (de) 2008-10-01
JP4807884B2 (ja) 2011-11-02
SI1805163T1 (sl) 2009-02-28
IL180962A0 (en) 2007-07-04
TW200616994A (en) 2006-06-01
CA2574305A1 (en) 2006-02-02
WO2006010544A2 (en) 2006-02-02
ZA200700535B (en) 2008-10-29
ES2313391T3 (es) 2009-03-01
RU2007107164A (ru) 2008-09-10
RU2386626C2 (ru) 2010-04-20

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