NO20053557L - Fremgangsmate for produksjon av 3'-nukleosid prolegemidler. - Google Patents

Fremgangsmate for produksjon av 3'-nukleosid prolegemidler.

Info

Publication number
NO20053557L
NO20053557L NO20053557A NO20053557A NO20053557L NO 20053557 L NO20053557 L NO 20053557L NO 20053557 A NO20053557 A NO 20053557A NO 20053557 A NO20053557 A NO 20053557A NO 20053557 L NO20053557 L NO 20053557L
Authority
NO
Norway
Prior art keywords
producing
nucleoside prodrugs
nucleoside
prodrugs
asylation
Prior art date
Application number
NO20053557A
Other languages
English (en)
Norwegian (no)
Inventor
Richard Storer
Adel Moussa
Steven Mathieu
Original Assignee
Idenix Cayman Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix Cayman Ltd filed Critical Idenix Cayman Ltd
Publication of NO20053557L publication Critical patent/NO20053557L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
NO20053557A 2002-12-23 2005-07-20 Fremgangsmate for produksjon av 3'-nukleosid prolegemidler. NO20053557L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43615002P 2002-12-23 2002-12-23
PCT/US2003/041603 WO2004058792A1 (en) 2002-12-23 2003-12-23 Process for the production of 3'-nucleoside prodrugs

Publications (1)

Publication Number Publication Date
NO20053557L true NO20053557L (no) 2005-09-08

Family

ID=32682350

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20053557A NO20053557L (no) 2002-12-23 2005-07-20 Fremgangsmate for produksjon av 3'-nukleosid prolegemidler.

Country Status (16)

Country Link
US (1) US20040181051A1 (es)
EP (1) EP1575971A4 (es)
JP (1) JP2006514038A (es)
KR (1) KR20050110611A (es)
CN (1) CN100335492C (es)
AU (1) AU2003300434A1 (es)
BR (1) BR0316868A (es)
CA (1) CA2511616A1 (es)
IL (1) IL169314A0 (es)
MX (1) MXPA05006865A (es)
NO (1) NO20053557L (es)
NZ (1) NZ540913A (es)
PL (1) PL377608A1 (es)
RU (1) RU2005123395A (es)
WO (1) WO2004058792A1 (es)
ZA (1) ZA200505040B (es)

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MY164523A (en) 2000-05-23 2017-12-29 Univ Degli Studi Cagliari Methods and compositions for treating hepatitis c virus
NZ547204A (en) 2000-05-26 2008-01-31 Idenix Cayman Ltd Methods and compositions for treating flaviviruses and pestiviruses
KR20050088079A (ko) 2002-11-15 2005-09-01 이데닉스 (케이만) 리미티드 2'-분지형 뉴클레오시드 및 플라비비리다에 돌연변이
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EP1830871A1 (en) * 2004-12-23 2007-09-12 Novartis AG Compositions for hcv treatment
US8802840B2 (en) 2005-03-08 2014-08-12 Biota Scientific Management Pty Ltd. Bicyclic nucleosides and nucleotides as therapeutic agents
US7514410B2 (en) * 2005-03-29 2009-04-07 Biocryst Pharmaceuticals, Inc. Hepatitis C therapies
CA2622191A1 (en) * 2005-09-22 2008-03-11 Keshab Sarma Selective o-acylation of nucleosides
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EP2004634A1 (en) 2006-04-04 2008-12-24 F.Hoffmann-La Roche Ag 3',5'-di-o-acylated nucleosides for hcv treatment
WO2010015637A1 (en) * 2008-08-06 2010-02-11 Novartis Ag New antiviral modified nucleosides
CL2009002206A1 (es) 2008-12-23 2011-08-26 Gilead Pharmasset Llc Compuestos derivados de pirrolo -(2-3-d]-pirimidin-7(6h)-tetrahidrofuran-2-il fosfonamidato, composicion farmaceutica; y su uso en el tratamiento de enfermedades virales.
NZ593648A (en) 2008-12-23 2013-09-27 Gilead Pharmasset Llc Nucleoside phosphoramidates
EA201100851A1 (ru) 2008-12-23 2012-04-30 Фармассет, Инк. Аналоги нуклеозидов
PE20120013A1 (es) * 2009-01-09 2012-02-02 Univ Cardiff Fosforamidato derivados de guanosina compuestos nucleosidos para tratamiento de infecciones virales
BR112012024884A2 (pt) 2010-03-31 2016-10-18 Gilead Pharmasset Llc síntese estereosseletiva de ativos contendo fósforo
EA037868B1 (ru) 2016-09-07 2021-05-28 Атеа Фармасьютикалс, Инк. 2'-замещенные-n6-замещенные пуриновые нуклеотиды для лечения вызванных рнк-вирусом заболеваний
US20220033430A1 (en) * 2018-11-25 2022-02-03 Tnt Medical Corporation Orally active prodrug of gemcitabine

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Also Published As

Publication number Publication date
CA2511616A1 (en) 2004-07-15
CN100335492C (zh) 2007-09-05
WO2004058792A1 (en) 2004-07-15
PL377608A1 (pl) 2006-02-06
KR20050110611A (ko) 2005-11-23
AU2003300434A1 (en) 2004-07-22
ZA200505040B (en) 2006-04-26
IL169314A0 (en) 2007-07-04
MXPA05006865A (es) 2005-12-12
EP1575971A1 (en) 2005-09-21
NZ540913A (en) 2008-02-29
US20040181051A1 (en) 2004-09-16
BR0316868A (pt) 2005-10-25
RU2005123395A (ru) 2006-01-27
CN1751058A (zh) 2006-03-22
JP2006514038A (ja) 2006-04-27
EP1575971A4 (en) 2008-03-05

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