NO20043850L - 10-(3-Cyklopropylaminometyl-1-pyrrolidinyl) pyridobenzo ksazinkarboksylsyrerederivater effektive mot medikament-resistente bakterier - Google Patents

10-(3-Cyklopropylaminometyl-1-pyrrolidinyl) pyridobenzo ksazinkarboksylsyrerederivater effektive mot medikament-resistente bakterier

Info

Publication number
NO20043850L
NO20043850L NO20043850A NO20043850A NO20043850L NO 20043850 L NO20043850 L NO 20043850L NO 20043850 A NO20043850 A NO 20043850A NO 20043850 A NO20043850 A NO 20043850A NO 20043850 L NO20043850 L NO 20043850L
Authority
NO
Norway
Prior art keywords
group
hydrogen atom
resistant bacteria
kazazine
pyridobenzo
Prior art date
Application number
NO20043850A
Other languages
English (en)
Norwegian (no)
Inventor
Yoshikazu Asahina
Masaya Takei
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of NO20043850L publication Critical patent/NO20043850L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
NO20043850A 2002-03-18 2004-09-14 10-(3-Cyklopropylaminometyl-1-pyrrolidinyl) pyridobenzo ksazinkarboksylsyrerederivater effektive mot medikament-resistente bakterier NO20043850L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2002074783 2002-03-18
JP2002369205 2002-12-20
PCT/JP2003/002967 WO2003078439A1 (fr) 2002-03-18 2003-03-13 Derive d'acide 10-(3-cyclopropylaminomethyl-1-pyrrolidinyl)pyridobenzoxazinecarboxylique efficace contre les bacteries resistantes

Publications (1)

Publication Number Publication Date
NO20043850L true NO20043850L (no) 2004-09-14

Family

ID=28043757

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20043850A NO20043850L (no) 2002-03-18 2004-09-14 10-(3-Cyklopropylaminometyl-1-pyrrolidinyl) pyridobenzo ksazinkarboksylsyrerederivater effektive mot medikament-resistente bakterier

Country Status (14)

Country Link
US (1) US7153851B2 (fr)
EP (1) EP1486500B1 (fr)
JP (1) JP4468701B2 (fr)
KR (1) KR20040094806A (fr)
CN (1) CN1653071A (fr)
AT (1) ATE443064T1 (fr)
AU (1) AU2003213335B8 (fr)
BR (1) BR0308643A (fr)
CA (1) CA2478763A1 (fr)
DE (1) DE60329280D1 (fr)
MX (1) MXPA04009026A (fr)
NO (1) NO20043850L (fr)
NZ (1) NZ535182A (fr)
WO (1) WO2003078439A1 (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100410249C (zh) * 2003-09-10 2008-08-13 杏林制药株式会社 7-(4-取代-3-环丙基氨基甲基-1-吡咯烷基)喹诺酮羧酸衍生物
NZ533360A (en) 2004-06-04 2007-02-23 Ind Res Ltd Improved method for preparing 3-hydroxy-4-hydroxymethyl-pyrrolidine compounds
JPWO2006009143A1 (ja) * 2004-07-21 2008-05-01 杏林製薬株式会社 (3s)−3−ヒドロキシメチル−7−オキソピリドベンゾオキサジン−6−カルボン酸エステルの製造方法
GB0428250D0 (en) * 2004-12-23 2005-01-26 Novartis Ag Organic compounds
JP5154402B2 (ja) * 2006-03-09 2013-02-27 杏林製薬株式会社 3,4−ジ置換ピロリジン誘導体の製造方法及び製造中間体
SG182370A1 (en) * 2010-01-08 2012-08-30 Kyorin Seiyaku Kk Method for producing 3,4-disubstituted pyrrolidine derivative and production intermediate thereof
MX2012013717A (es) * 2010-05-31 2013-01-28 Kyorin Seiyaku Kk Metodo para producir derivado de 3-sustituida-4-fluoropirrolidina.
WO2012057093A1 (fr) 2010-10-25 2012-05-03 杏林製薬株式会社 Procédé de fabrication d'un dérivé 3, 4, pyrrolidine disubstituée
CN102276628A (zh) * 2011-06-21 2011-12-14 周崇科 氟喹诺酮类化合物及其合成方法
EP2990038B1 (fr) 2013-04-25 2019-11-20 Kyorin Pharmaceutical Co., Ltd. Composition pharmaceutique solide
EA201791995A1 (ru) * 2015-03-13 2017-12-29 Керин Фармасьютикал Ко., Лтд. Средство для лечения респираторной инфекции
GB201708606D0 (en) 2017-05-30 2017-07-12 King's College London Antibiotic resistance breakers
CN112194667B (zh) * 2020-11-06 2021-08-17 湖南科技大学 取代1,4-苯并噁嗪并二氮卓类化合物及其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4822801A (en) * 1984-07-20 1989-04-18 Warner-Lambert Company 4-oxo-1,4-dihydroquinoline-3-carboxylic acid derivative as antibacterial agents
JPS62155282A (ja) * 1985-12-27 1987-07-10 Sankyo Co Ltd ピリドベンゾオキサジンカルボン酸誘導体
TW425394B (en) * 1996-04-24 2001-03-11 Daiichi Seiyaku Co Antimicrobial quinolone derivatives having 3-(N-cycloalkyl) aminomethylpyrrolidine group
JPH10287669A (ja) 1997-04-10 1998-10-27 Dai Ichi Seiyaku Co Ltd 置換アミノメチルピロリジン誘導体

Also Published As

Publication number Publication date
CA2478763A1 (fr) 2003-09-25
WO2003078439A1 (fr) 2003-09-25
JP4468701B2 (ja) 2010-05-26
AU2003213335B8 (en) 2009-04-02
ATE443064T1 (de) 2009-10-15
CN1653071A (zh) 2005-08-10
EP1486500A4 (fr) 2006-02-08
BR0308643A (pt) 2005-02-09
KR20040094806A (ko) 2004-11-10
AU2003213335A1 (en) 2003-09-29
JPWO2003078439A1 (ja) 2005-07-14
NZ535182A (en) 2006-02-24
AU2003213335B2 (en) 2008-09-11
US7153851B2 (en) 2006-12-26
US20050182052A1 (en) 2005-08-18
DE60329280D1 (de) 2009-10-29
MXPA04009026A (es) 2005-01-25
EP1486500B1 (fr) 2009-09-16
EP1486500A1 (fr) 2004-12-15

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