NO20034660L - Spiropyrazolforbindelser, farmasoytiske preparater som omfatter en slik forbindelse, og anvendelse av forbindelsene for fremstilling av farmasoytiske preparater - Google Patents

Spiropyrazolforbindelser, farmasoytiske preparater som omfatter en slik forbindelse, og anvendelse av forbindelsene for fremstilling av farmasoytiske preparater

Info

Publication number
NO20034660L
NO20034660L NO20034660A NO20034660A NO20034660L NO 20034660 L NO20034660 L NO 20034660L NO 20034660 A NO20034660 A NO 20034660A NO 20034660 A NO20034660 A NO 20034660A NO 20034660 L NO20034660 L NO 20034660L
Authority
NO
Norway
Prior art keywords
compounds
compound
preparation
spiropyrazole
pharmaceutical
Prior art date
Application number
NO20034660A
Other languages
English (en)
Norwegian (no)
Other versions
NO20034660D0 (no
Inventor
R Richard Goehring
Donald J Kyle
Sam F Victory
Gary Lee
Parviz Gharagozloo
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Publication of NO20034660D0 publication Critical patent/NO20034660D0/no
Publication of NO20034660L publication Critical patent/NO20034660L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10—Spiro-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Dental Preparations (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO20034660A 2001-04-18 2003-10-17 Spiropyrazolforbindelser, farmasoytiske preparater som omfatter en slik forbindelse, og anvendelse av forbindelsene for fremstilling av farmasoytiske preparater NO20034660L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28467501P 2001-04-18 2001-04-18
PCT/US2002/012376 WO2002085355A1 (en) 2001-04-18 2002-04-18 Spiropyrazole compounds

Publications (2)

Publication Number Publication Date
NO20034660D0 NO20034660D0 (no) 2003-10-17
NO20034660L true NO20034660L (no) 2003-12-17

Family

ID=23091099

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20034660A NO20034660L (no) 2001-04-18 2003-10-17 Spiropyrazolforbindelser, farmasoytiske preparater som omfatter en slik forbindelse, og anvendelse av forbindelsene for fremstilling av farmasoytiske preparater

Country Status (28)

Country Link
US (2) US6635653B2 (xx)
EP (1) EP1385515B1 (xx)
JP (1) JP4342181B2 (xx)
KR (1) KR100628292B1 (xx)
CN (1) CN1516584A (xx)
AT (1) ATE403429T1 (xx)
AU (1) AU2002311833B2 (xx)
BR (1) BR0209127A (xx)
CA (1) CA2444634C (xx)
CY (1) CY1108454T1 (xx)
CZ (1) CZ20032849A3 (xx)
DE (1) DE60228071D1 (xx)
DK (1) DK1385515T3 (xx)
ES (1) ES2312584T3 (xx)
HK (1) HK1062885A1 (xx)
HU (1) HUP0401333A3 (xx)
IL (2) IL158485A0 (xx)
MX (1) MXPA03009604A (xx)
NO (1) NO20034660L (xx)
NZ (1) NZ528978A (xx)
PL (1) PL367263A1 (xx)
PT (1) PT1385515E (xx)
RU (1) RU2299883C2 (xx)
SI (1) SI1385515T1 (xx)
UA (1) UA74439C2 (xx)
WO (1) WO2002085355A1 (xx)
YU (1) YU82403A (xx)
ZA (1) ZA200308103B (xx)

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WO2004034983A2 (en) * 2002-10-17 2004-04-29 Euro-Celtique, S.A. Preparation of triazospiro compounds
US20040242583A1 (en) * 2003-01-20 2004-12-02 Aventis Pharma Deutschland Gmbh Pyrimido[5,4-e][1,2,4]triazine-5,7-diones, processes for preparing them and their use
WO2004103305A2 (en) * 2003-05-16 2004-12-02 Euroceltique S.A. Spiropyrazole compound
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US20110008327A1 (en) 2004-03-29 2011-01-13 Cheng Jin Q Compositions including triciribine and epidermal growth factor receptor inhibitor compounds or salts thereof and methods of use thereof
PL2574341T3 (pl) 2004-03-29 2017-09-29 University Of South Florida Efektywne leczenie guzów i raka fosforanem tricyrybiny
US20100009929A1 (en) 2004-03-29 2010-01-14 Cheng Jin Q Compositions including triciribine and bortezomib and derivatives thereof and methods of use thereof
US20100173864A1 (en) 2004-03-29 2010-07-08 Cheng Jin Q Compositions including triciribine and one or more platinum compounds and methods of use thereof
US20100009928A1 (en) * 2004-03-29 2010-01-14 Cheng Jin Q Compositions including triciribine and taxanes and methods of use thereof
US20100028339A1 (en) 2004-03-29 2010-02-04 Cheng Jin Q Compositions including triciribine and trastuzumab and methods of use thereof
BRPI0608847A2 (pt) 2005-03-08 2010-02-02 Janssen Pharmaceutica Nv derivados de diaza-espiro-[4,4]-nonano substituìdos e seu uso como antagonistas de neurocinina
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US20080051380A1 (en) 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
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SI2076506T1 (sl) 2007-01-16 2011-01-31 Purdue Pharma Lp Heterociklično substituirani piperidini kot ORL-1 ligandi
CA2683598C (en) 2007-04-09 2015-11-17 Janssen Pharmaceutica Nv 1,3,8-trisubstituted-1,3,8-triaza-spiro[4.5]decan-4-one derivatives as ligands of the orl-i receptor for the treatment of anxiety and depression
EP3101018B1 (en) 2007-08-31 2019-03-06 Purdue Pharma L.P. Substituted-quinoxaline-type-piperidine compounds and the uses thereof
EP2324013B3 (en) 2008-07-21 2014-10-22 Purdue Pharma LP Substituted-quinoxaline-type bridged-piperidine compounds and the uses thereof
UA107943C2 (xx) * 2009-11-16 2015-03-10 Lilly Co Eli Сполуки спіропіперидину як антагоністи рецептора orl-1
US9598447B2 (en) 2010-12-22 2017-03-21 Purdue Pharma L.P. Phosphorus-substituted quinoxaline-type piperidine compounds and uses thereof
JP2014533744A (ja) 2011-12-01 2014-12-15 パーデュー、ファーマ、リミテッド、パートナーシップ アゼチジン置換キノキサリンタイプピペリジン化合物とその使用
US9085561B2 (en) 2012-07-30 2015-07-21 Purdue Pharma L.P. Cyclic urea- or lactam-substituted quinoxaline-type piperidines as ORL-1 modulators
US9090618B2 (en) 2012-12-27 2015-07-28 Purdue Pharma L.P. Substituted benzimidazole-type piperidine compounds and uses thereof
US9951038B2 (en) 2012-12-27 2018-04-24 Purdue Pharma L.P. Quinazolin-4(3H)-one-type piperidine compounds and uses thereof
WO2014102590A1 (en) 2012-12-27 2014-07-03 Purdue Pharma L.P. Substituted piperidin-4-amino-type compounds and uses thereof
US9040533B2 (en) 2012-12-27 2015-05-26 Purdue Pharma L.P. Oxime-substituted-quinoxaline-type piperidine compounds as ORL-1 modulators
US9963458B2 (en) 2012-12-27 2018-05-08 Purdue Pharma L.P. Indole and indoline-type piperidine compounds and uses thereof
CA3031705A1 (en) 2016-07-29 2018-02-01 Janssen Pharmaceutica Nv Treatment of prostate cancer with niraparib
CN111825681A (zh) * 2020-07-07 2020-10-27 扬州大学 一种合成(e)-亚苄基螺吡唑吡咯嗪酮类化合物的方法

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CN1516584A (zh) * 2001-04-18 2004-07-28 ŷ�����ǹɷ����޹�˾ 螺吡唑化合物

Also Published As

Publication number Publication date
BR0209127A (pt) 2006-03-21
RU2003133455A (ru) 2005-05-10
YU82403A (sh) 2006-08-17
CY1108454T1 (el) 2014-04-09
HK1062885A1 (en) 2004-12-03
ATE403429T1 (de) 2008-08-15
PL367263A1 (en) 2005-02-21
ZA200308103B (en) 2004-10-18
PT1385515E (pt) 2008-09-15
CZ20032849A3 (en) 2004-03-17
AU2002311833B2 (en) 2005-04-28
MXPA03009604A (es) 2004-04-02
JP4342181B2 (ja) 2009-10-14
WO2002085355A1 (en) 2002-10-31
ES2312584T3 (es) 2009-03-01
NO20034660D0 (no) 2003-10-17
DE60228071D1 (de) 2008-09-18
EP1385515A1 (en) 2004-02-04
CN1516584A (zh) 2004-07-28
US6635653B2 (en) 2003-10-21
CA2444634A1 (en) 2002-10-31
RU2299883C2 (ru) 2007-05-27
IL158485A (en) 2009-09-01
EP1385515A4 (en) 2004-06-30
US20030027834A1 (en) 2003-02-06
US20040087641A1 (en) 2004-05-06
HUP0401333A2 (hu) 2004-10-28
CA2444634C (en) 2011-06-07
IL158485A0 (en) 2004-05-12
DK1385515T3 (da) 2008-10-27
UA74439C2 (uk) 2005-12-15
KR100628292B1 (ko) 2006-09-27
SI1385515T1 (sl) 2008-12-31
EP1385515B1 (en) 2008-08-06
JP2004531531A (ja) 2004-10-14
HUP0401333A3 (en) 2004-11-29
NZ528978A (en) 2004-06-25
KR20040008159A (ko) 2004-01-28

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