NO20020811L - Sulfonylkarboksamidderivater, fremgangsmåte for deres fremstilling og deres anvendelse som legemidler - Google Patents
Sulfonylkarboksamidderivater, fremgangsmåte for deres fremstilling og deres anvendelse som legemidlerInfo
- Publication number
- NO20020811L NO20020811L NO20020811A NO20020811A NO20020811L NO 20020811 L NO20020811 L NO 20020811L NO 20020811 A NO20020811 A NO 20020811A NO 20020811 A NO20020811 A NO 20020811A NO 20020811 L NO20020811 L NO 20020811L
- Authority
- NO
- Norway
- Prior art keywords
- drugs
- processes
- preparation
- carboxamide derivatives
- sulfonyl
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/26—Sulfur atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Oppfinnelsen vedrører sulfonyl karboksamid derivater, i tillegg til deres fysiologisk tålbare salter og fysiologisk funksjonelle derivater og deres anvendelse ved produksjon av legemidler for forebygging og behandling av hyperlipidemi og arteriosklerotiske sykdommer. Oppfinnelsen vedrører forbindelse med formel I hvori radikalene har de nærmere angitte betydninger og deres fysiologisk tålbare salter og fysiologisk funksjonelle derivater. Forbindelsene er egnet for bruk for eksempel som lipidsenkende substanser.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE1999141540 DE19941540C2 (de) | 1999-09-01 | 1999-09-01 | Sulfonylcarboxamide zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Hyperlipidämie |
DE2000127611 DE10027611A1 (de) | 2000-06-06 | 2000-06-06 | Sulfonylcarboxamidderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
PCT/EP2000/008027 WO2001016094A1 (de) | 1999-09-01 | 2000-08-17 | Sulfonylcarboxamidderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20020811D0 NO20020811D0 (no) | 2002-02-19 |
NO20020811L true NO20020811L (no) | 2002-04-30 |
Family
ID=26005953
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20020811A NO20020811L (no) | 1999-09-01 | 2002-02-19 | Sulfonylkarboksamidderivater, fremgangsmåte for deres fremstilling og deres anvendelse som legemidler |
Country Status (28)
Country | Link |
---|---|
US (2) | US6342512B1 (no) |
EP (1) | EP1218341B1 (no) |
JP (1) | JP4792186B2 (no) |
KR (1) | KR20020033778A (no) |
CN (1) | CN1372541A (no) |
AR (1) | AR025444A1 (no) |
AT (1) | ATE302754T1 (no) |
AU (1) | AU774071B2 (no) |
BR (1) | BR0013727A (no) |
CA (1) | CA2383781A1 (no) |
CO (1) | CO5190698A1 (no) |
CZ (1) | CZ2002767A3 (no) |
DE (1) | DE50011035D1 (no) |
DK (1) | DK1218341T3 (no) |
EE (1) | EE200200095A (no) |
ES (1) | ES2246247T3 (no) |
HK (1) | HK1048984A1 (no) |
HR (1) | HRP20020177A2 (no) |
HU (1) | HUP0202472A3 (no) |
IL (1) | IL148148A0 (no) |
MX (1) | MXPA02001696A (no) |
MY (1) | MY133732A (no) |
NO (1) | NO20020811L (no) |
PL (1) | PL353367A1 (no) |
PT (1) | PT1218341E (no) |
RU (1) | RU2002107998A (no) |
SK (1) | SK2682002A3 (no) |
WO (1) | WO2001016094A1 (no) |
Families Citing this family (78)
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WO2012120057A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
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WO2012120055A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
WO2012120056A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
WO2012120058A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
WO2012120051A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit adamantan- oder noradamantan substituierte benzyl-oxathiazinderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
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JP6103182B2 (ja) * | 2011-10-03 | 2017-03-29 | セイコーエプソン株式会社 | 発電装置、電子機器、移動手段及び発電装置の制御方法 |
FR2997247B1 (fr) * | 2012-10-22 | 2016-12-09 | Commissariat Energie Atomique | Generateur d'electricite et recuperateur d'energie |
CN104502513B (zh) * | 2015-01-14 | 2016-04-06 | 中国矿业大学连云港徐圩新区高新技术研究院 | 一种对羧基苯磺酰胺的高效液相色谱测定方法 |
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GB1353357A (en) * | 1970-09-14 | 1974-05-15 | Pfizer | Substituted 5-sulphamylbenzoic acids |
US4138399A (en) | 1970-09-14 | 1979-02-06 | Pfizer Inc. | Sulfamylbenzoic acid |
DE2517183A1 (de) * | 1975-04-18 | 1976-10-28 | Hoechst Ag | Basisch substituierte 5-sulfamoyl- anthranilsaeurederivate und verfahren zu ihrer herstellung |
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2000
- 2000-08-17 RU RU2002107998/04A patent/RU2002107998A/ru not_active Application Discontinuation
- 2000-08-17 AT AT00953172T patent/ATE302754T1/de not_active IP Right Cessation
- 2000-08-17 MX MXPA02001696A patent/MXPA02001696A/es unknown
- 2000-08-17 PT PT00953172T patent/PT1218341E/pt unknown
- 2000-08-17 HU HU0202472A patent/HUP0202472A3/hu unknown
- 2000-08-17 BR BR0013727-8A patent/BR0013727A/pt not_active IP Right Cessation
- 2000-08-17 EE EEP200200095A patent/EE200200095A/xx unknown
- 2000-08-17 EP EP00953172A patent/EP1218341B1/de not_active Expired - Lifetime
- 2000-08-17 CA CA002383781A patent/CA2383781A1/en not_active Abandoned
- 2000-08-17 IL IL14814800A patent/IL148148A0/xx unknown
- 2000-08-17 CN CN00811269A patent/CN1372541A/zh active Pending
- 2000-08-17 WO PCT/EP2000/008027 patent/WO2001016094A1/de active IP Right Grant
- 2000-08-17 KR KR1020027002650A patent/KR20020033778A/ko not_active Application Discontinuation
- 2000-08-17 PL PL00353367A patent/PL353367A1/xx not_active Application Discontinuation
- 2000-08-17 CZ CZ2002767A patent/CZ2002767A3/cs unknown
- 2000-08-17 SK SK268-2002A patent/SK2682002A3/sk unknown
- 2000-08-17 JP JP2001519664A patent/JP4792186B2/ja not_active Expired - Fee Related
- 2000-08-17 AU AU65712/00A patent/AU774071B2/en not_active Ceased
- 2000-08-17 DK DK00953172T patent/DK1218341T3/da active
- 2000-08-17 ES ES00953172T patent/ES2246247T3/es not_active Expired - Lifetime
- 2000-08-17 DE DE50011035T patent/DE50011035D1/de not_active Expired - Lifetime
- 2000-08-25 CO CO00063853A patent/CO5190698A1/es not_active Application Discontinuation
- 2000-08-29 MY MYPI20003962 patent/MY133732A/en unknown
- 2000-08-30 AR ARP000104517A patent/AR025444A1/es unknown
- 2000-09-01 US US09/654,841 patent/US6342512B1/en not_active Expired - Lifetime
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2001
- 2001-09-27 US US09/963,380 patent/US6552048B2/en not_active Expired - Lifetime
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2002
- 2002-02-19 NO NO20020811A patent/NO20020811L/no not_active Application Discontinuation
- 2002-02-27 HR HR20020177A patent/HRP20020177A2/hr not_active Application Discontinuation
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2003
- 2003-02-18 HK HK03101152.9A patent/HK1048984A1/zh unknown
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