NO20013380D0 - 2-aminobenzoksazinonderivater for behandling av fedme - Google Patents

2-aminobenzoksazinonderivater for behandling av fedme

Info

Publication number
NO20013380D0
NO20013380D0 NO20013380A NO20013380A NO20013380D0 NO 20013380 D0 NO20013380 D0 NO 20013380D0 NO 20013380 A NO20013380 A NO 20013380A NO 20013380 A NO20013380 A NO 20013380A NO 20013380 D0 NO20013380 D0 NO 20013380D0
Authority
NO
Norway
Prior art keywords
aminobenzoxazinone
obesity
derivatives
treatment
aminobenzoxazinone derivatives
Prior art date
Application number
NO20013380A
Other languages
English (en)
Other versions
NO321058B1 (no
NO20013380L (no
Inventor
Harold Francis Hodson
Robert Downham
Timothy John Mitchell
Beverley Jane Carr
Christopher Robert Dunk
Richard Michael John Palmer
Original Assignee
Alizyme Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alizyme Therapeutics Ltd filed Critical Alizyme Therapeutics Ltd
Publication of NO20013380D0 publication Critical patent/NO20013380D0/no
Publication of NO20013380L publication Critical patent/NO20013380L/no
Publication of NO321058B1 publication Critical patent/NO321058B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
    • C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/26—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring
    • C07C271/28—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring to a carbon atom of a non-condensed six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/40—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/58—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20013380A 1999-01-08 2001-07-06 Anvendelse av 2-aminobenzoksazinonderivater ved fremstilling av et medikament for profylakse eller behandling av overvekt eller en overvektsrelatert forstyrrelse, 2-aminobenzoksazinonderivater, fremgangsmate for fremstilling derav, farmasoytiske preparater og matprodukter som inneholder derivatene, anvendelser av derivatene samt kosmetisk fremgangsmate ved administrering derav. NO321058B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9900416.0A GB9900416D0 (en) 1999-01-08 1999-01-08 Inhibitors
PCT/GB2000/000031 WO2000040569A1 (en) 1999-01-08 2000-01-06 2-amino-benzoxazinone derivatives for the treatment of obesity

Publications (3)

Publication Number Publication Date
NO20013380D0 true NO20013380D0 (no) 2001-07-06
NO20013380L NO20013380L (no) 2001-09-07
NO321058B1 NO321058B1 (no) 2006-03-06

Family

ID=10845777

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013380A NO321058B1 (no) 1999-01-08 2001-07-06 Anvendelse av 2-aminobenzoksazinonderivater ved fremstilling av et medikament for profylakse eller behandling av overvekt eller en overvektsrelatert forstyrrelse, 2-aminobenzoksazinonderivater, fremgangsmate for fremstilling derav, farmasoytiske preparater og matprodukter som inneholder derivatene, anvendelser av derivatene samt kosmetisk fremgangsmate ved administrering derav.

Country Status (22)

Country Link
US (2) US6656934B2 (no)
EP (1) EP1144395B1 (no)
JP (1) JP2002534419A (no)
KR (1) KR100615914B1 (no)
CN (1) CN100480245C (no)
AR (1) AR022203A1 (no)
AT (1) ATE293610T1 (no)
AU (1) AU770342B2 (no)
CA (1) CA2359987C (no)
DE (1) DE60019556T2 (no)
DK (1) DK1144395T3 (no)
ES (1) ES2240051T3 (no)
GB (1) GB9900416D0 (no)
HK (1) HK1047284A1 (no)
HU (1) HUP0104909A3 (no)
MY (1) MY129247A (no)
NO (1) NO321058B1 (no)
NZ (1) NZ512739A (no)
PL (1) PL350412A1 (no)
PT (1) PT1144395E (no)
RU (1) RU2244711C2 (no)
WO (1) WO2000040569A1 (no)

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US20030027786A1 (en) 2001-06-06 2003-02-06 Karsten Maeder Lipase inhibiting composition
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PT1144395E (pt) 2005-08-31
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DE60019556T2 (de) 2006-02-23
CA2359987A1 (en) 2000-07-13
DK1144395T3 (da) 2005-08-15
RU2244711C2 (ru) 2005-01-20
DE60019556D1 (de) 2005-05-25
EP1144395A1 (en) 2001-10-17
HUP0104909A3 (en) 2004-11-29
ATE293610T1 (de) 2005-05-15
WO2000040569A8 (en) 2001-03-15
CA2359987C (en) 2008-03-25
AR022203A1 (es) 2002-09-04
AU1884500A (en) 2000-07-24
US7776853B2 (en) 2010-08-17
AU770342B2 (en) 2004-02-19
US20030191123A1 (en) 2003-10-09
CN100480245C (zh) 2009-04-22
MY129247A (en) 2007-03-30
KR100615914B1 (ko) 2006-08-28
US6656934B2 (en) 2003-12-02
GB9900416D0 (en) 1999-02-24
US20030013707A1 (en) 2003-01-16
CN1354747A (zh) 2002-06-19
HK1047284A1 (en) 2003-02-14
JP2002534419A (ja) 2002-10-15
PL350412A1 (en) 2002-12-02
NO20013380L (no) 2001-09-07
WO2000040569A1 (en) 2000-07-13
EP1144395B1 (en) 2005-04-20
HUP0104909A2 (hu) 2002-04-29
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ES2240051T3 (es) 2005-10-16
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