NO20003111D0 - Ortho-anthranilamidderivater som antikoagulanter - Google Patents

Ortho-anthranilamidderivater som antikoagulanter

Info

Publication number
NO20003111D0
NO20003111D0 NO20003111A NO20003111A NO20003111D0 NO 20003111 D0 NO20003111 D0 NO 20003111D0 NO 20003111 A NO20003111 A NO 20003111A NO 20003111 A NO20003111 A NO 20003111A NO 20003111 D0 NO20003111 D0 NO 20003111D0
Authority
NO
Norway
Prior art keywords
anticoagulants
ortho
anthranilamide derivatives
anthranilamide
derivatives
Prior art date
Application number
NO20003111A
Other languages
English (en)
Other versions
NO20003111L (no
Inventor
Damian O Arnaiz
Yuo-Ling Chou
Rushad E Karanjawala
Monica J Kochanny
Wheeseong Lee
Amy Mei Liang
Michael M Morrissey
Gary B Phillips
Karna Lyn Sacchi
Stephen T Sakata
Kenneth J Shaw
R Michael Snider
Shung C Wu
Bin Ye
Zuchun Zhao
Brian D Griedel
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/187,459 external-priority patent/US6140351A/en
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO20003111D0 publication Critical patent/NO20003111D0/no
Publication of NO20003111L publication Critical patent/NO20003111L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D333/70Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
NO20003111A 1997-12-19 2000-06-16 Orto-antranilamidderivater som antikoagulanter NO20003111L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US99428497A 1997-12-19 1997-12-19
US09/187,459 US6140351A (en) 1997-12-19 1998-11-05 Ortho-anthranilamide derivatives as anti-coagulants
PCT/EP1998/007650 WO1999032477A1 (en) 1997-12-19 1998-11-27 Ortho-anthranilamide derivatives as anti-coagulants

Publications (2)

Publication Number Publication Date
NO20003111D0 true NO20003111D0 (no) 2000-06-16
NO20003111L NO20003111L (no) 2000-08-18

Family

ID=26883056

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20003111A NO20003111L (no) 1997-12-19 2000-06-16 Orto-antranilamidderivater som antikoagulanter

Country Status (19)

Country Link
US (2) US6498185B1 (no)
EP (1) EP1040108B1 (no)
JP (1) JP3811006B2 (no)
CN (1) CN1143855C (no)
AT (1) ATE260103T1 (no)
AU (1) AU751856B2 (no)
CA (1) CA2315070A1 (no)
DE (1) DE69821985T2 (no)
DK (1) DK1040108T3 (no)
ES (1) ES2215337T3 (no)
HU (1) HUP0101172A3 (no)
IL (1) IL135536A0 (no)
NO (1) NO20003111L (no)
NZ (1) NZ503809A (no)
PL (1) PL341044A1 (no)
PT (1) PT1040108E (no)
RU (1) RU2226529C2 (no)
SK (1) SK9432000A3 (no)
WO (1) WO1999032477A1 (no)

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Also Published As

Publication number Publication date
EP1040108A1 (en) 2000-10-04
IL135536A0 (en) 2001-05-20
CN1143855C (zh) 2004-03-31
EP1040108B1 (en) 2004-02-25
NO20003111L (no) 2000-08-18
JP3811006B2 (ja) 2006-08-16
ATE260103T1 (de) 2004-03-15
CN1282329A (zh) 2001-01-31
DK1040108T3 (da) 2004-05-24
JP2001526283A (ja) 2001-12-18
SK9432000A3 (en) 2001-02-12
HUP0101172A1 (hu) 2002-05-29
PT1040108E (pt) 2004-06-30
ES2215337T3 (es) 2004-10-01
DE69821985D1 (de) 2004-04-01
HUP0101172A3 (en) 2002-12-28
PL341044A1 (en) 2001-03-26
WO1999032477A1 (en) 1999-07-01
CA2315070A1 (en) 1999-07-01
AU1875999A (en) 1999-07-12
US6380221B1 (en) 2002-04-30
DE69821985T2 (de) 2005-05-04
RU2226529C2 (ru) 2004-04-10
WO1999032477B1 (en) 1999-09-10
AU751856B2 (en) 2002-08-29
NZ503809A (en) 2002-04-26
US6498185B1 (en) 2002-12-24

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