NO20002190L - 2-halo-6-O-substituerte ketolidderivater - Google Patents

2-halo-6-O-substituerte ketolidderivater

Info

Publication number
NO20002190L
NO20002190L NO20002190A NO20002190A NO20002190L NO 20002190 L NO20002190 L NO 20002190L NO 20002190 A NO20002190 A NO 20002190A NO 20002190 A NO20002190 A NO 20002190A NO 20002190 L NO20002190 L NO 20002190L
Authority
NO
Norway
Prior art keywords
halo
ketolide derivatives
substituted ketolide
substituted
derivatives
Prior art date
Application number
NO20002190A
Other languages
English (en)
Norwegian (no)
Other versions
NO20002190D0 (no
Inventor
Ly Tam Phan
Yat Sun Or
Daniel T Chu
Jacob J Plattner
Yan Chen
Richard F Clark
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of NO20002190D0 publication Critical patent/NO20002190D0/no
Publication of NO20002190L publication Critical patent/NO20002190L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
NO20002190A 1997-10-29 2000-04-27 2-halo-6-O-substituerte ketolidderivater NO20002190L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US95988197A 1997-10-29 1997-10-29
US15423998A 1998-09-16 1998-09-16
PCT/US1998/022989 WO1999021871A1 (en) 1997-10-29 1998-10-29 2-halo-6-o-substituted ketolide derivatives

Publications (2)

Publication Number Publication Date
NO20002190D0 NO20002190D0 (no) 2000-04-27
NO20002190L true NO20002190L (no) 2000-06-29

Family

ID=26851273

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20002190A NO20002190L (no) 1997-10-29 2000-04-27 2-halo-6-O-substituerte ketolidderivater

Country Status (24)

Country Link
EP (1) EP1027362B1 (cs)
JP (1) JP2001521039A (cs)
KR (1) KR100536420B1 (cs)
CN (1) CN1240707C (cs)
AR (1) AR015994A1 (cs)
AT (1) ATE298760T1 (cs)
AU (1) AU751448B2 (cs)
BG (1) BG64707B1 (cs)
BR (1) BR9813319A (cs)
CA (1) CA2307788C (cs)
CO (1) CO4990960A1 (cs)
CZ (1) CZ300063B6 (cs)
DE (1) DE69830739T2 (cs)
DK (1) DK1027362T3 (cs)
ES (1) ES2244094T3 (cs)
HU (1) HUP0004282A3 (cs)
IL (1) IL135519A0 (cs)
NO (1) NO20002190L (cs)
NZ (1) NZ503822A (cs)
PL (1) PL191453B1 (cs)
PT (1) PT1027362E (cs)
SK (1) SK286397B6 (cs)
TR (1) TR200001142T2 (cs)
WO (1) WO1999021871A1 (cs)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE39743E1 (en) * 1998-10-15 2007-07-24 Aventis Pharma S.A. 2-halogenated derivatives of 5-0 desosaminyl-erythronolide a, their preparation process and their antibiotic use
FR2784682B1 (fr) 1998-10-15 2002-12-06 Hoechst Marion Roussel Inc Nouveaux derives 2-halogene de 5-0-desosaminylerythronolide a, leur procede de preparation et leur application comme medicaments
WO2000063225A2 (en) * 1999-04-16 2000-10-26 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6939861B2 (en) 1999-04-16 2005-09-06 Kosan Biosciences, Inc. Amido macrolides
US6514944B2 (en) 1999-04-16 2003-02-04 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
ES2306674T3 (es) * 1999-12-02 2008-11-16 Abbott Laboratories Derivados cetolidos 6-o-alquil-2-nor-2-sustituidos.
US6569836B2 (en) 1999-12-02 2003-05-27 Abbott Laboratories 6-O-alkyl-2-nor-2-substituted ketolide derivatives
JP2001261694A (ja) * 2000-03-06 2001-09-26 Pfizer Prod Inc ケトライド抗生物質
US6605707B1 (en) * 2000-03-23 2003-08-12 Abbott Laboratories Process for the preparation of 6-O-propargyl erythromycin derivatives
ES2222966T3 (es) 2000-06-30 2005-02-16 Pfizer Products Inc. Macrolidos antibioticos.
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
CA2460947A1 (en) 2001-09-17 2003-03-27 Ortho-Mcneil Pharmaceutical, Inc. 6-o-carbamate-11,12-lacto-ketolide antimicrobials
PL370714A1 (en) 2001-12-05 2005-05-30 Ortho-Mcneil Pharmaceutical, Inc. 6-o-acyl ketolide derivatives of erythromycine useful as antibacterials
JP2005522453A (ja) * 2002-02-13 2005-07-28 アボット・ラボラトリーズ マクロライド抗菌化合物
CA2483220A1 (en) * 2002-04-25 2003-11-06 Abbott Laboratories Oxolide antibacterials
WO2003090761A1 (en) * 2002-04-25 2003-11-06 Abbott Laboratories 9-oxime macrolide antibacterials
JPWO2004078771A1 (ja) * 2003-03-07 2006-06-08 大正製薬株式会社 2−フルオロ−6−o−置換ケトライド誘導体
JP2007254285A (ja) * 2004-03-16 2007-10-04 Taisho Pharmaceut Co Ltd 2−フルオロ−6−o−置換ケトライド誘導体
KR101566053B1 (ko) * 2009-05-27 2015-11-04 욱크하르트 리미티드 항균 활성을 갖는 케톨라이드

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8506380D0 (en) * 1985-03-12 1985-04-11 Beecham Group Plc Chemical compounds
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
DK0638584T3 (da) * 1992-04-22 1996-04-15 Taisho Pharmaceutical Co Ltd 5-O-desosaminyl-erythronolid-A-derivat
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
CZ20001525A3 (cs) 2000-10-11
JP2001521039A (ja) 2001-11-06
BR9813319A (pt) 2000-08-22
KR100536420B1 (ko) 2005-12-16
WO1999021871A1 (en) 1999-05-06
HK1031383A1 (en) 2001-06-15
AU1288199A (en) 1999-05-17
PT1027362E (pt) 2005-08-31
PL340290A1 (en) 2001-01-29
IL135519A0 (en) 2001-05-20
EP1027362A1 (en) 2000-08-16
KR20010015793A (ko) 2001-02-26
TR200001142T2 (tr) 2000-09-21
HUP0004282A2 (hu) 2001-04-28
NO20002190D0 (no) 2000-04-27
ATE298760T1 (de) 2005-07-15
AR015994A1 (es) 2001-05-30
SK6332000A3 (en) 2000-09-12
AU751448B2 (en) 2002-08-15
DK1027362T3 (da) 2005-10-31
SK286397B6 (sk) 2008-09-05
CO4990960A1 (es) 2000-12-26
DE69830739D1 (de) 2005-08-04
CN1283199A (zh) 2001-02-07
BG64707B1 (bg) 2005-12-30
BG104434A (en) 2001-01-31
DE69830739T2 (de) 2006-04-20
ES2244094T3 (es) 2005-12-01
EP1027362B1 (en) 2005-06-29
NZ503822A (en) 2002-12-20
PL191453B1 (pl) 2006-05-31
CN1240707C (zh) 2006-02-08
CZ300063B6 (cs) 2009-01-21
CA2307788C (en) 2008-05-20
HUP0004282A3 (en) 2001-10-29
CA2307788A1 (en) 1999-05-06

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application