NO20001557L - Tetrahydrofuranfosfat- og hydroksyestere som prolegemidler for det tilsvarende antifungale middel - Google Patents
Tetrahydrofuranfosfat- og hydroksyestere som prolegemidler for det tilsvarende antifungale middelInfo
- Publication number
- NO20001557L NO20001557L NO20001557A NO20001557A NO20001557L NO 20001557 L NO20001557 L NO 20001557L NO 20001557 A NO20001557 A NO 20001557A NO 20001557 A NO20001557 A NO 20001557A NO 20001557 L NO20001557 L NO 20001557L
- Authority
- NO
- Norway
- Prior art keywords
- prodrugs
- tetrahydrofuran
- phosphate
- antifungal agent
- hydroxy esters
- Prior art date
Links
- 229940121375 antifungal agent Drugs 0.000 title 1
- 239000003429 antifungal agent Substances 0.000 title 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 title 1
- MSZYQCNHWFXSAK-UHFFFAOYSA-N oxolane;phosphoric acid Chemical compound C1CCOC1.OP(O)(O)=O MSZYQCNHWFXSAK-UHFFFAOYSA-N 0.000 title 1
- 229940002612 prodrug Drugs 0.000 title 1
- 239000000651 prodrug Substances 0.000 title 1
- 206010017533 Fungal infection Diseases 0.000 abstract 1
- 208000031888 Mycoses Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
- C07F9/6518—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US93782797A | 1997-09-25 | 1997-09-25 | |
| PCT/US1998/018508 WO1999015522A1 (en) | 1997-09-25 | 1998-09-22 | Tetrahydrofuran phosphate- and hydroxy esters, as prodrugs for the corresponding antifungal agent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20001557D0 NO20001557D0 (no) | 2000-03-24 |
| NO20001557L true NO20001557L (no) | 2000-03-24 |
Family
ID=25470461
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20001557A NO20001557L (no) | 1997-09-25 | 2000-03-24 | Tetrahydrofuranfosfat- og hydroksyestere som prolegemidler for det tilsvarende antifungale middel |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP1027349B1 (de) |
| JP (1) | JP3473949B2 (de) |
| KR (1) | KR20010024297A (de) |
| CN (1) | CN1125066C (de) |
| AR (1) | AR015458A1 (de) |
| AT (1) | ATE286502T1 (de) |
| AU (1) | AU1698199A (de) |
| BR (1) | BR9812671A (de) |
| CA (1) | CA2304624C (de) |
| CO (1) | CO5011088A1 (de) |
| DE (1) | DE69828524T2 (de) |
| ES (1) | ES2232974T3 (de) |
| HK (1) | HK1025960A1 (de) |
| HU (1) | HUP0004616A3 (de) |
| ID (1) | ID28294A (de) |
| IL (1) | IL134469A0 (de) |
| MY (1) | MY133775A (de) |
| NO (1) | NO20001557L (de) |
| NZ (1) | NZ502709A (de) |
| PE (1) | PE120799A1 (de) |
| PL (1) | PL339488A1 (de) |
| PT (1) | PT1027349E (de) |
| SK (1) | SK3912000A3 (de) |
| TR (1) | TR200000753T2 (de) |
| WO (1) | WO1999015522A1 (de) |
| ZA (1) | ZA988688B (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU1915500A (en) | 1998-11-20 | 2000-06-13 | Bristol-Myers Squibb Company | Water soluble prodrugs of azole compounds |
| CA2798002C (en) * | 2010-05-19 | 2019-12-03 | Sandoz Ag | Process for the preparation of chiral triazolones |
| CN111138421A (zh) * | 2019-12-26 | 2020-05-12 | 上海英诺富成生物科技有限公司 | 抗真菌水溶性化合物及其制备方法与应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5693626A (en) * | 1993-12-21 | 1997-12-02 | Schering Corporation | Tetrahydrofuran antifungals |
| DE69428125T2 (de) * | 1993-12-21 | 2002-05-02 | Schering Corp., Kenilworth | Fungizide tetrahydrofurane |
-
1998
- 1998-09-22 DE DE69828524T patent/DE69828524T2/de not_active Expired - Lifetime
- 1998-09-22 PT PT98961721T patent/PT1027349E/pt unknown
- 1998-09-22 CN CN98809550A patent/CN1125066C/zh not_active Expired - Fee Related
- 1998-09-22 ZA ZA988688A patent/ZA988688B/xx unknown
- 1998-09-22 ES ES98961721T patent/ES2232974T3/es not_active Expired - Lifetime
- 1998-09-22 HU HU0004616A patent/HUP0004616A3/hu unknown
- 1998-09-22 AR ARP980104741A patent/AR015458A1/es unknown
- 1998-09-22 MY MYPI98004343A patent/MY133775A/en unknown
- 1998-09-22 SK SK391-2000A patent/SK3912000A3/sk unknown
- 1998-09-22 NZ NZ502709A patent/NZ502709A/en unknown
- 1998-09-22 EP EP98961721A patent/EP1027349B1/de not_active Expired - Lifetime
- 1998-09-22 BR BR9812671-7A patent/BR9812671A/pt not_active IP Right Cessation
- 1998-09-22 IL IL13446998A patent/IL134469A0/xx unknown
- 1998-09-22 CA CA002304624A patent/CA2304624C/en not_active Expired - Fee Related
- 1998-09-22 JP JP2000512827A patent/JP3473949B2/ja not_active Expired - Fee Related
- 1998-09-22 TR TR2000/00753T patent/TR200000753T2/xx unknown
- 1998-09-22 PE PE1998000905A patent/PE120799A1/es not_active Application Discontinuation
- 1998-09-22 ID IDW20000551A patent/ID28294A/id unknown
- 1998-09-22 AU AU16981/99A patent/AU1698199A/en not_active Abandoned
- 1998-09-22 AT AT98961721T patent/ATE286502T1/de not_active IP Right Cessation
- 1998-09-22 KR KR1020007003196A patent/KR20010024297A/ko not_active Application Discontinuation
- 1998-09-22 WO PCT/US1998/018508 patent/WO1999015522A1/en not_active Application Discontinuation
- 1998-09-22 PL PL98339488A patent/PL339488A1/xx unknown
- 1998-09-23 CO CO98055163A patent/CO5011088A1/es unknown
-
2000
- 2000-03-24 NO NO20001557A patent/NO20001557L/no not_active Application Discontinuation
- 2000-08-17 HK HK00105167A patent/HK1025960A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1271356A (zh) | 2000-10-25 |
| AR015458A1 (es) | 2001-05-02 |
| CA2304624C (en) | 2007-06-19 |
| ATE286502T1 (de) | 2005-01-15 |
| PL339488A1 (en) | 2000-12-18 |
| EP1027349B1 (de) | 2005-01-05 |
| EP1027349A1 (de) | 2000-08-16 |
| CA2304624A1 (en) | 1999-04-01 |
| JP3473949B2 (ja) | 2003-12-08 |
| JP2001517665A (ja) | 2001-10-09 |
| TR200000753T2 (tr) | 2001-01-22 |
| DE69828524T2 (de) | 2005-12-29 |
| PE120799A1 (es) | 1999-12-01 |
| ZA988688B (en) | 1999-03-23 |
| AU1698199A (en) | 1999-04-12 |
| PT1027349E (pt) | 2005-05-31 |
| IL134469A0 (en) | 2001-04-30 |
| CN1125066C (zh) | 2003-10-22 |
| WO1999015522A1 (en) | 1999-04-01 |
| DE69828524D1 (de) | 2005-02-10 |
| NO20001557D0 (no) | 2000-03-24 |
| MY133775A (en) | 2007-11-30 |
| CO5011088A1 (es) | 2001-02-28 |
| KR20010024297A (ko) | 2001-03-26 |
| SK3912000A3 (en) | 2000-08-14 |
| HUP0004616A3 (en) | 2002-04-29 |
| BR9812671A (pt) | 2000-08-22 |
| HK1025960A1 (en) | 2000-12-01 |
| ES2232974T3 (es) | 2005-06-01 |
| NZ502709A (en) | 2001-11-30 |
| HUP0004616A2 (hu) | 2002-03-28 |
| ID28294A (id) | 2001-05-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |