NO177099C - Analogifremgangsmåte for fremstilling av nye, terapeutisk aktive steroidderivater - Google Patents

Analogifremgangsmåte for fremstilling av nye, terapeutisk aktive steroidderivater

Info

Publication number
NO177099C
NO177099C NO901102A NO901102A NO177099C NO 177099 C NO177099 C NO 177099C NO 901102 A NO901102 A NO 901102A NO 901102 A NO901102 A NO 901102A NO 177099 C NO177099 C NO 177099C
Authority
NO
Norway
Prior art keywords
therapeutically active
analogous process
steroid derivatives
preparing new
active steroid
Prior art date
Application number
NO901102A
Other languages
English (en)
Other versions
NO177099B (no
NO901102L (no
NO901102D0 (no
Inventor
Csaba Molnar
Gyorgy Hajos
Laszlo Szporny
Jozsef Toth
Arpad Kiraly
Anna Boor
Janos Csorgei
Krisztina Szekely
Lilla Forgacs
Gyorgy Fekete
Bulcsu Herenyi
Sandor Holy
Josef Szunyog
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of NO901102D0 publication Critical patent/NO901102D0/no
Publication of NO901102L publication Critical patent/NO901102L/no
Publication of NO177099B publication Critical patent/NO177099B/no
Publication of NO177099C publication Critical patent/NO177099C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/0026Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031Oxygen-containing hetero ring cyclic ketals at positions 16, 17
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J7/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C07J7/008Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO901102A 1989-03-09 1990-03-08 Analogifremgangsmåte for fremstilling av nye, terapeutisk aktive steroidderivater NO177099C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU891155A HU203769B (en) 1989-03-09 1989-03-09 Process for producing new steroide derivatives and pharmaceutical compositions containing them

Publications (4)

Publication Number Publication Date
NO901102D0 NO901102D0 (no) 1990-03-08
NO901102L NO901102L (no) 1990-09-10
NO177099B NO177099B (no) 1995-04-10
NO177099C true NO177099C (no) 1995-07-19

Family

ID=10953084

Family Applications (1)

Application Number Title Priority Date Filing Date
NO901102A NO177099C (no) 1989-03-09 1990-03-08 Analogifremgangsmåte for fremstilling av nye, terapeutisk aktive steroidderivater

Country Status (19)

Country Link
US (1) US5053404A (no)
EP (1) EP0387090A3 (no)
JP (1) JPH075629B2 (no)
KR (1) KR930009446B1 (no)
CN (1) CN1045397A (no)
AR (1) AR245452A1 (no)
AU (1) AU617929B2 (no)
BG (1) BG60440B2 (no)
CA (1) CA2011280A1 (no)
EG (1) EG19166A (no)
FI (1) FI901200A0 (no)
HU (1) HU203769B (no)
IL (1) IL93477A (no)
IN (1) IN169862B (no)
NO (1) NO177099C (no)
PH (1) PH26685A (no)
PT (1) PT93374A (no)
TW (1) TW208020B (no)
ZA (1) ZA901753B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9100341D0 (sv) * 1991-02-04 1991-02-04 Astra Ab Novel steroids
FR2675146A1 (fr) * 1991-04-10 1992-10-16 Roussel Uclaf Nouveaux derives sterouides de la pregna-1,4-diene-3,20-dione, leur preparation, leur application a la preparation de derives 16,17-methylene dioxy substitues et nouveaux intermediaires.
DE69942578D1 (de) 1998-05-22 2010-08-26 Univ R Bifunktionelle moleküle sowie darauf basierende therapien.
EP3827747A1 (en) 2005-04-28 2021-06-02 Otsuka Pharmaceutical Co., Ltd. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
NZ616673A (en) 2009-02-20 2014-08-29 To Bbb Holding B V Glutathione-based drug delivery system
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
CN110078785A (zh) * 2019-06-04 2019-08-02 博诺康源(北京)药业科技有限公司 一种布地奈德杂质ep-ze的合成方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3167545A (en) * 1959-02-07 1965-01-26 Syntex Corp 16beta-methyl-16alpha, 17 alpha-dihydroxy pregnenes and the 16alpha, 17alpha-cyclic ketals and acetals thereof
US3345362A (en) * 1961-07-27 1967-10-03 Lilly Co Eli Novel pregnenolone acetonides
US3798216A (en) * 1969-03-07 1974-03-19 Fabrication Des Antibiotique S 9-fluoro-11beta,21-dihydroxy-16alpha,17-(2-propenylidenedioxy)-pregna-1,4-diene-3,20-dione and derivatives thereof
SE378109B (no) * 1972-05-19 1975-08-18 Bofors Ab
US3992534A (en) * 1972-05-19 1976-11-16 Ab Bofors Compositions and method of treating with component B of stereoisomeric mixtures of 2'-unsymmetrical 16,17-methylenedioxy steriods
SE8008524L (sv) * 1980-12-04 1982-06-05 Draco Ab 4-pregnen-derivat, ett forfarande for deras framstellning, beredning och metod for behandling av inflammatoriska tillstand
DE3133631A1 (de) * 1981-08-21 1983-03-03 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue kortikoide ihre herstellung und verwendung
HU182775B (en) * 1981-10-15 1984-03-28 Richter Gedeon Vegyeszet Process for preparing new 3-chloro-pregnane derivatives
SE8501693D0 (sv) * 1985-04-04 1985-04-04 Draco Ab Novel 16,17-acetalsubstituted androstane-17beta-carboxylic acid esters
SE8506015D0 (sv) * 1985-12-19 1985-12-19 Draco Ab Novel 16,17-acetalsubstituted pregnane 21-oic acid derivatives

Also Published As

Publication number Publication date
AU5079890A (en) 1990-09-20
TW208020B (no) 1993-06-21
HU203769B (en) 1991-09-30
KR930009446B1 (ko) 1993-10-04
EG19166A (en) 1994-11-30
IL93477A (en) 1994-07-31
FI901200A0 (fi) 1990-03-09
ZA901753B (en) 1990-12-28
BG60440B2 (bg) 1995-03-31
JPH02279697A (ja) 1990-11-15
PT93374A (pt) 1990-11-07
PH26685A (en) 1992-09-15
KR900014423A (ko) 1990-10-23
IL93477A0 (en) 1990-11-29
CA2011280A1 (en) 1990-09-09
NO177099B (no) 1995-04-10
NO901102L (no) 1990-09-10
EP0387090A3 (en) 1992-05-06
JPH075629B2 (ja) 1995-01-25
IN169862B (no) 1992-01-04
US5053404A (en) 1991-10-01
EP0387090A2 (en) 1990-09-12
AU617929B2 (en) 1991-12-05
AR245452A1 (es) 1994-01-31
NO901102D0 (no) 1990-03-08
CN1045397A (zh) 1990-09-19

Similar Documents

Publication Publication Date Title
NO176759C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive 3-substituerte-2-oksindol-derivater
NO179639C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive, substituerte piperidinforbindelser
NO177387C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive imidazo-kondenserte, 6-leddede, heterocykliske forbindelser
NO174385C (no) Analogifremgangsmåte ved fremstilling av terapeutisk aktive spiro-substituerte glutamid-derivater
NO180749C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive benzimidazolsubstituerte derivater
NO174467C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive kromanderivater
NO891191D0 (no) Fremgangsmaate for fremstilling av nye, terapeutisk virksomme catecholderivater.
NO174959C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive N-aminobutyl-N-fenyl-arylamidderivater
NO178967C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive pyridazin-derivater
NO177096C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive, substituerte isokinoliner
NO176477C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive 2-alkoksymetylsubstituerte kromanderivater
NO173784C (no) Anaslogifremgangsmaate for fremstilling av terapeutisk aktive tieno-tri-azolo-diazepinderivater
NO178374C (no) Analogifremgangsmåte for fremstilling av nye terapeutisk aktive acetylcholinesteraseinhibitorer
NO175976C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-(1,6-dihydro-6-okso-pyridazinyl-3-oksy)-3-kromanolderivater
NO174391C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive kromanderivater
NO176100C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive oksodihydropyridyl- og oksodihydropyridazinylkromanderivater
NO870998L (no) FremgangsmŸte for fremstilling av nye, terapeutisk aktive acetamid-derivater.
NO175781C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive tetracykliske forbindelser
NO174892C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive, substituerte dihydropyrrolizinforbindelser
NO177099C (no) Analogifremgangsmåte for fremstilling av nye, terapeutisk aktive steroidderivater
NO173607C (no) Analogifremgangsmaate for fremstilling av nye terapeutisk aktive tienotriazolo-diazepin-derivater
NO174422C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive kromanderivater
NO174200C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive 2-imino-6-polyfluoralkoksybenzotiazol-forbindelser
FI903077A0 (fi) Menetelmä valmistaa terapeuttisesti aktiivisia R(-)-3-kinuklidinolijohdannaisia
NO173332C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive tetrahydrofuranderivater