NO174772C - Analogifremgangsmåte ved fremstilling av terapeutisk aktive piperazinylderivater - Google Patents

Analogifremgangsmåte ved fremstilling av terapeutisk aktive piperazinylderivater

Info

Publication number
NO174772C
NO174772C NO895281A NO895281A NO174772C NO 174772 C NO174772 C NO 174772C NO 895281 A NO895281 A NO 895281A NO 895281 A NO895281 A NO 895281A NO 174772 C NO174772 C NO 174772C
Authority
NO
Norway
Prior art keywords
preparation
compounds
therapeutically active
analogous procedure
piperazinyl derivatives
Prior art date
Application number
NO895281A
Other languages
English (en)
Other versions
NO174772B (no
NO895281D0 (no
NO895281L (no
Inventor
Jens Perregaard
John Willie Stenberg
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of NO895281D0 publication Critical patent/NO895281D0/no
Publication of NO895281L publication Critical patent/NO895281L/no
Publication of NO174772B publication Critical patent/NO174772B/no
Publication of NO174772C publication Critical patent/NO174772C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO895281A 1988-12-28 1989-12-27 Analogifremgangsmåte ved fremstilling av terapeutisk aktive piperazinylderivater NO174772C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888830312A GB8830312D0 (en) 1988-12-28 1988-12-28 Heterocyclic compounds

Publications (4)

Publication Number Publication Date
NO895281D0 NO895281D0 (no) 1989-12-27
NO895281L NO895281L (no) 1990-06-29
NO174772B NO174772B (no) 1994-03-28
NO174772C true NO174772C (no) 1994-07-06

Family

ID=10649223

Family Applications (1)

Application Number Title Priority Date Filing Date
NO895281A NO174772C (no) 1988-12-28 1989-12-27 Analogifremgangsmåte ved fremstilling av terapeutisk aktive piperazinylderivater

Country Status (17)

Country Link
US (1) US5002948A (no)
EP (1) EP0376607B1 (no)
JP (1) JP2895121B2 (no)
AT (1) ATE102184T1 (no)
AU (1) AU637991B2 (no)
CA (1) CA2006356C (no)
DE (1) DE68913487T2 (no)
DK (1) DK169266B1 (no)
ES (1) ES2062050T3 (no)
FI (1) FI93005C (no)
GB (1) GB8830312D0 (no)
IE (1) IE62668B1 (no)
IL (1) IL92990A (no)
NO (1) NO174772C (no)
NZ (1) NZ231855A (no)
PT (1) PT92728B (no)
ZA (1) ZA899960B (no)

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DE4101686A1 (de) * 1991-01-22 1992-07-23 Merck Patent Gmbh Indolderivate
NZ243065A (en) * 1991-06-13 1995-07-26 Lundbeck & Co As H Piperidine derivatives and pharmaceutical compositions
DE4127849A1 (de) * 1991-08-22 1993-02-25 Merck Patent Gmbh Benzodioxanderivate
CA2084531A1 (en) * 1991-12-19 1993-06-20 David W. Smith Antimigraine 4-pyrimidinyl and pyridinyl derivatives of indol-3yl-alkyl piperazines
DK55192D0 (da) * 1992-04-28 1992-04-28 Lundbeck & Co As H 1-piperazino-1,2-dihydroindenderivater
DK78692D0 (da) * 1992-06-12 1992-06-12 Lundbeck & Co As H Dimere piperidin- og piperazinderivater
FR2692264B1 (fr) * 1992-06-12 1994-08-05 Adir Nouvelles piperazines 1,4-disubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant.
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CA2297825C (en) 1997-07-25 2006-03-14 H. Lundbeck A/S Indole and 2,3-dihydroindole derivatives, their preparation and use
DE69902766T2 (de) * 1998-04-08 2003-02-06 Wyeth, Madison N-aryloxyethylaminderivate zur behandlung der depression
AR022303A1 (es) 1999-01-22 2002-09-04 Lundbeck & Co As H Derivados de piperidina, tetrahidropiridina y piperazina, su preparacion y utilizacion
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JP5220746B2 (ja) 2006-08-25 2013-06-26 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 制御放出システム及びその製造方法
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EP2459533A4 (en) 2009-07-30 2013-01-16 Univ Singapore SMALL MOLECULE INHIBITORS OF ISOPRENYLCYSTEIN CARBOXYL METHYLTRANERASE WITH POTENTIAL ANTICANCING ACTIVITY
CA2770724A1 (en) * 2009-08-10 2011-02-17 Galenea Corporation 5-ht inhibiting indole compounds
CN102993186B (zh) * 2012-12-20 2015-11-18 北京海步国际医药科技发展有限公司 一种新型的哌嗪衍生物
EP3027607B1 (en) 2013-07-29 2020-08-26 Sunshine Lake Pharma Co., Ltd. Substituted heteroaryl compounds and methods of use thereof
WO2015090235A1 (en) 2013-12-20 2015-06-25 Sunshine Lake Pharma Co., Ltd. Substituted piperazine compounds and methods of use thereof
CN106065018B (zh) * 2015-04-23 2020-04-21 广东东阳光药业有限公司 取代的吲哚化合物及其使用方法和用途
WO2016192657A1 (en) 2015-06-03 2016-12-08 Sunshine Lake Pharma Co., Ltd. Substituted piperazine compounds and methods of use and use thereof

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Also Published As

Publication number Publication date
NZ231855A (en) 1992-02-25
AU4719889A (en) 1990-07-05
IE893976L (en) 1990-06-13
DK169266B1 (da) 1994-09-26
FI93005B (fi) 1994-10-31
FI896300A0 (fi) 1989-12-28
EP0376607A1 (en) 1990-07-04
US5002948A (en) 1991-03-26
IL92990A0 (en) 1990-09-17
AU637991B2 (en) 1993-06-17
DK645689A (da) 1990-06-29
EP0376607B1 (en) 1994-03-02
ATE102184T1 (de) 1994-03-15
IE62668B1 (en) 1995-02-22
IL92990A (en) 1995-01-24
DE68913487D1 (de) 1994-04-07
DE68913487T2 (de) 1994-08-04
JPH02225460A (ja) 1990-09-07
FI93005C (fi) 1995-02-10
PT92728B (pt) 1995-12-29
NO174772B (no) 1994-03-28
NO895281D0 (no) 1989-12-27
GB8830312D0 (en) 1989-02-22
NO895281L (no) 1990-06-29
CA2006356C (en) 1999-09-14
JP2895121B2 (ja) 1999-05-24
DK645689D0 (da) 1989-12-19
ZA899960B (en) 1990-11-28
PT92728A (pt) 1990-06-29
ES2062050T3 (es) 1994-12-16
CA2006356A1 (en) 1990-06-28

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