NO174551C - Analogifremgangsmåte for fremstilling av terapeutisk aktive aminomethyl-oxooxazolidinyl-aroylbenzen-derivater - Google Patents
Analogifremgangsmåte for fremstilling av terapeutisk aktive aminomethyl-oxooxazolidinyl-aroylbenzen-derivaterInfo
- Publication number
- NO174551C NO174551C NO884594A NO884594A NO174551C NO 174551 C NO174551 C NO 174551C NO 884594 A NO884594 A NO 884594A NO 884594 A NO884594 A NO 884594A NO 174551 C NO174551 C NO 174551C
- Authority
- NO
- Norway
- Prior art keywords
- aroylbenzene
- derivatives
- oxooxazolidinyl
- aminomethyl
- therapeutically active
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10903287A | 1987-10-16 | 1987-10-16 |
Publications (4)
Publication Number | Publication Date |
---|---|
NO884594D0 NO884594D0 (no) | 1988-10-14 |
NO884594L NO884594L (no) | 1989-04-17 |
NO174551B NO174551B (no) | 1994-02-14 |
NO174551C true NO174551C (no) | 1994-05-25 |
Family
ID=22325458
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO884594A NO174551C (no) | 1987-10-16 | 1988-10-14 | Analogifremgangsmåte for fremstilling av terapeutisk aktive aminomethyl-oxooxazolidinyl-aroylbenzen-derivater |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP0312000B1 (de) |
JP (1) | JPH01132570A (de) |
KR (1) | KR890006602A (de) |
AT (1) | ATE73783T1 (de) |
AU (1) | AU617366B2 (de) |
CA (1) | CA1320730C (de) |
DE (1) | DE3869310D1 (de) |
DK (1) | DK573988A (de) |
ES (1) | ES2033394T3 (de) |
FI (1) | FI884755A (de) |
GR (1) | GR3004973T3 (de) |
HU (1) | HU199810B (de) |
IE (1) | IE60426B1 (de) |
IL (1) | IL88047A (de) |
MY (1) | MY103784A (de) |
NO (1) | NO174551C (de) |
NZ (1) | NZ226582A (de) |
PT (1) | PT88765B (de) |
SU (1) | SU1616517A3 (de) |
ZA (1) | ZA887683B (de) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
US5231188A (en) * | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
EP0610265B1 (de) * | 1991-11-01 | 1996-12-27 | PHARMACIA & UPJOHN COMPANY | Substituierte aryl- und heteroaryl-phenyloxazolidinone |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
HUT74099A (en) * | 1992-12-08 | 1996-11-28 | Upjohn Co | Tropone-substituted phenyloxazolidinone antibacterial agents and pharmaceutical compositions containing the same |
US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
EP0730591B1 (de) * | 1993-11-22 | 1999-07-14 | PHARMACIA & UPJOHN COMPANY | Substituierte hydroxyacetyl piperazine phenyl oxazolidinonsäureester |
DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
DE4425609A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | Benzofuranyl- und Benzothienyloxazolidinone |
DE4425612A1 (de) * | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
DE19514313A1 (de) | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
RU2128660C1 (ru) * | 1994-11-15 | 1999-04-10 | Фармация Энд Апджон Компани | Бициклические оксазин- или тиазин-оксазолидиноны или их фармацевтически приемлемые соли и способы лечения микробных инфекций |
PL185872B1 (pl) * | 1995-02-03 | 2003-08-29 | Upjohn Co | Nowe podstawione fenylooksazolidynonyNowe podstawione fenylooksazolidynony |
HRP960159A2 (en) * | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
DE69614847T2 (de) * | 1995-05-11 | 2002-04-04 | Pharmacia & Upjohn Co., Kalamazoo | Spirocyclische und bicyclische diazinyl- und carbazinyloxazolidinone |
US5883093A (en) * | 1995-09-12 | 1999-03-16 | Pharmacia & Upjohn Company | Phenyloxazolidinone antimicrobials |
DE19601265A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone |
GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
DE19604223A1 (de) | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
HRP970049A2 (en) | 1996-02-06 | 1998-04-30 | Bayer Ag | New heteroaryl oxazolidinones |
GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
GB9609919D0 (en) | 1996-05-11 | 1996-07-17 | Zeneca Ltd | Chemical compounds |
GB9717804D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
EP1007525A1 (de) * | 1997-08-29 | 2000-06-14 | Zeneca Limited | Oxooxazolidinylbenzolderivate |
EP1030852B1 (de) * | 1997-11-12 | 2003-09-17 | PHARMACIA & UPJOHN COMPANY | Oxazolidinone derivate und pharmazeutische zusammensetzungen |
GB9725244D0 (en) | 1997-11-29 | 1998-01-28 | Zeneca Ltd | Chemical compounds |
NZ505902A (en) * | 1998-01-23 | 2003-08-29 | Upjohn Co | Oxazolidinone compounds useful as antimicrobial agents and combinatorial libraries |
US7002020B1 (en) | 1998-01-23 | 2006-02-21 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
US6562844B2 (en) | 1998-01-23 | 2003-05-13 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
AU1379900A (en) * | 1998-11-17 | 2000-06-05 | Bayer Aktiengesellschaft | Novel substituted phenyloxazolidone derivatives |
NZ523700A (en) | 2000-07-17 | 2004-11-26 | Ranbaxy Lab Ltd | Oxazolidinone derivatives as antimicrobials |
US6956040B2 (en) | 2001-07-16 | 2005-10-18 | Ranbaxy Laboratories Limited | Oxazolidinone piperazinyl derivatives as potential antimicrobials |
KR100854211B1 (ko) | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
CN101220002B (zh) * | 2007-12-28 | 2011-07-13 | 天津药物研究院 | 作为抗菌剂的噁唑烷酮类化合物 |
KR101023174B1 (ko) * | 2008-09-24 | 2011-03-18 | 주식회사 레고켐 바이오사이언스 | 사이클릭 아미독심 또는 사이클릭 아미드라존 기를 가지는 신규한 옥사졸리디논 유도체 및 이를 함유하는 의약 조성물 |
ES2744907T3 (es) | 2008-10-10 | 2020-02-26 | Merck Sharp & Dohme | Compuestos usados en la síntesis de oxazolidinonas |
EP2393808B1 (de) | 2009-02-03 | 2019-05-08 | Merck Sharp & Dohme Corp. | Kristalline form von r)-3-(4-(2-(2-methyltetrazol-5-yl)pyridin-5-yl)-3-fluorophenyl)-5-hydroxymethyloxazolidin-2-on-dihydrogenphosphat |
US8580767B2 (en) | 2009-05-28 | 2013-11-12 | Trius Therapeutics, Inc. | Oxazolidinone containing dimer compounds, compositions and methods to make and use |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1222708A (en) * | 1968-10-22 | 1971-02-17 | Delalande Sa | Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation |
FR2500450A1 (fr) * | 1981-02-25 | 1982-08-27 | Delalande Sa | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique |
ES533097A0 (es) * | 1983-06-07 | 1985-08-01 | Du Pont | Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno. |
CA1260948A (en) * | 1984-12-05 | 1989-09-26 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
-
1988
- 1988-10-11 CA CA000579796A patent/CA1320730C/en not_active Expired - Fee Related
- 1988-10-12 ES ES198888116903T patent/ES2033394T3/es not_active Expired - Lifetime
- 1988-10-12 AT AT88116903T patent/ATE73783T1/de not_active IP Right Cessation
- 1988-10-12 DE DE8888116903T patent/DE3869310D1/de not_active Expired - Fee Related
- 1988-10-12 EP EP88116903A patent/EP0312000B1/de not_active Expired - Lifetime
- 1988-10-14 MY MYPI88001159A patent/MY103784A/en unknown
- 1988-10-14 NZ NZ226582A patent/NZ226582A/xx unknown
- 1988-10-14 HU HU885297A patent/HU199810B/hu not_active IP Right Cessation
- 1988-10-14 PT PT88765A patent/PT88765B/pt not_active IP Right Cessation
- 1988-10-14 FI FI884755A patent/FI884755A/fi not_active Application Discontinuation
- 1988-10-14 DK DK573988A patent/DK573988A/da not_active Application Discontinuation
- 1988-10-14 KR KR1019880013394A patent/KR890006602A/ko not_active Application Discontinuation
- 1988-10-14 NO NO884594A patent/NO174551C/no unknown
- 1988-10-14 IE IE311988A patent/IE60426B1/en not_active IP Right Cessation
- 1988-10-14 IL IL88047A patent/IL88047A/xx unknown
- 1988-10-14 JP JP63257417A patent/JPH01132570A/ja active Pending
- 1988-10-14 ZA ZA887683A patent/ZA887683B/xx unknown
- 1988-10-14 SU SU884356643A patent/SU1616517A3/ru active
- 1988-10-17 AU AU23962/88A patent/AU617366B2/en not_active Ceased
-
1992
- 1992-06-18 GR GR920401308T patent/GR3004973T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
FI884755A (fi) | 1989-04-17 |
GR3004973T3 (de) | 1993-04-28 |
MY103784A (en) | 1993-09-30 |
AU2396288A (en) | 1989-04-20 |
ZA887683B (en) | 1990-06-27 |
NO884594L (no) | 1989-04-17 |
PT88765B (pt) | 1992-12-31 |
JPH01132570A (ja) | 1989-05-25 |
DK573988D0 (da) | 1988-10-14 |
CA1320730C (en) | 1993-07-27 |
DK573988A (da) | 1989-04-17 |
NZ226582A (en) | 1990-06-26 |
NO174551B (no) | 1994-02-14 |
ES2033394T3 (es) | 1993-03-16 |
IL88047A (en) | 1992-11-15 |
FI884755A0 (fi) | 1988-10-14 |
EP0312000A1 (de) | 1989-04-19 |
SU1616517A3 (ru) | 1990-12-23 |
IE883119L (en) | 1989-04-16 |
IL88047A0 (en) | 1989-06-30 |
ATE73783T1 (de) | 1992-04-15 |
IE60426B1 (en) | 1994-07-13 |
AU617366B2 (en) | 1991-11-28 |
EP0312000B1 (de) | 1992-03-18 |
KR890006602A (ko) | 1989-06-14 |
DE3869310D1 (de) | 1992-04-23 |
HU199810B (en) | 1990-03-28 |
NO884594D0 (no) | 1988-10-14 |
HUT49864A (en) | 1989-11-28 |
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