NO172239C - Fremgangsmaate for fremstilling av mevinolinanaloger - Google Patents

Fremgangsmaate for fremstilling av mevinolinanaloger

Info

Publication number
NO172239C
NO172239C NO883062A NO883062A NO172239C NO 172239 C NO172239 C NO 172239C NO 883062 A NO883062 A NO 883062A NO 883062 A NO883062 A NO 883062A NO 172239 C NO172239 C NO 172239C
Authority
NO
Norway
Prior art keywords
analogs
mevinoline
preparing
procedure
mevinolin
Prior art date
Application number
NO883062A
Other languages
English (en)
Norwegian (no)
Other versions
NO172239B (no
NO883062D0 (no
NO883062L (no
Inventor
Thomas R Verhoeven
David Askin
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22105351&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO172239(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of NO883062D0 publication Critical patent/NO883062D0/no
Publication of NO883062L publication Critical patent/NO883062L/no
Publication of NO172239B publication Critical patent/NO172239B/no
Publication of NO172239C publication Critical patent/NO172239C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
NO883062A 1987-07-10 1988-07-08 Fremgangsmaate for fremstilling av mevinolinanaloger NO172239C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/072,066 US4820850A (en) 1987-07-10 1987-07-10 Process for α-C-alkylation of the 8-acyl group on mevinolin and analogs thereof

Publications (4)

Publication Number Publication Date
NO883062D0 NO883062D0 (no) 1988-07-08
NO883062L NO883062L (no) 1989-01-11
NO172239B NO172239B (no) 1993-03-15
NO172239C true NO172239C (no) 1993-06-23

Family

ID=22105351

Family Applications (1)

Application Number Title Priority Date Filing Date
NO883062A NO172239C (no) 1987-07-10 1988-07-08 Fremgangsmaate for fremstilling av mevinolinanaloger

Country Status (22)

Country Link
US (1) US4820850A (zh)
EP (1) EP0299656B1 (zh)
JP (2) JPH0717663B2 (zh)
KR (1) KR950009314B1 (zh)
CN (1) CN1019395B (zh)
AT (1) ATE59036T1 (zh)
AU (1) AU604937B2 (zh)
CA (1) CA1287063C (zh)
CY (1) CY1613A (zh)
DE (1) DE3861270D1 (zh)
DK (1) DK172811B1 (zh)
ES (1) ES2018710B3 (zh)
FI (1) FI88719C (zh)
GR (1) GR3001351T3 (zh)
HK (1) HK98991A (zh)
IE (1) IE61025B1 (zh)
IL (1) IL86968A (zh)
NO (1) NO172239C (zh)
NZ (1) NZ225306A (zh)
PT (1) PT87909B (zh)
SG (1) SG84691G (zh)
ZA (1) ZA884924B (zh)

Families Citing this family (105)

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Also Published As

Publication number Publication date
JPH0717663B2 (ja) 1995-03-01
CN1019395B (zh) 1992-12-09
ATE59036T1 (de) 1990-12-15
KR890002199A (ko) 1989-04-08
AU604937B2 (en) 1991-01-03
IL86968A0 (en) 1988-12-30
FI883184A0 (fi) 1988-07-04
IE61025B1 (en) 1994-09-07
JPH07196641A (ja) 1995-08-01
NO172239B (no) 1993-03-15
FI883184A (fi) 1989-01-11
KR950009314B1 (ko) 1995-08-19
CY1613A (en) 1992-07-10
NZ225306A (en) 1990-06-26
IE882106L (en) 1989-01-10
CN1031086A (zh) 1989-02-15
PT87909B (pt) 1995-03-01
SG84691G (en) 1991-11-22
JPS6470481A (en) 1989-03-15
EP0299656B1 (en) 1990-12-12
HK98991A (en) 1991-12-13
GR3001351T3 (en) 1992-09-11
DK380788A (da) 1989-02-15
CA1287063C (en) 1991-07-30
DK172811B1 (da) 1999-07-26
US4820850A (en) 1989-04-11
NO883062D0 (no) 1988-07-08
AU1885088A (en) 1989-01-12
ZA884924B (en) 1989-01-17
NO883062L (no) 1989-01-11
FI88719C (fi) 1993-06-28
ES2018710B3 (es) 1991-05-01
EP0299656A1 (en) 1989-01-18
DE3861270D1 (de) 1991-01-24
PT87909A (pt) 1989-06-30
JP2527535B2 (ja) 1996-08-28
DK380788D0 (da) 1988-07-08
FI88719B (fi) 1993-03-15
IL86968A (en) 1992-12-01

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