NO145793C - Analogifremgangsmaate for fremstilling av den fysiologisk aktive forbindelse n-(r-tetrahydrofurfuryl)-noroksymorfon - Google Patents

Analogifremgangsmaate for fremstilling av den fysiologisk aktive forbindelse n-(r-tetrahydrofurfuryl)-noroksymorfon

Info

Publication number
NO145793C
NO145793C NO762932A NO762932A NO145793C NO 145793 C NO145793 C NO 145793C NO 762932 A NO762932 A NO 762932A NO 762932 A NO762932 A NO 762932A NO 145793 C NO145793 C NO 145793C
Authority
NO
Norway
Prior art keywords
noroxymorphone
tetrahydrofurfuryl
preparing
active compound
physiologically active
Prior art date
Application number
NO762932A
Other languages
English (en)
Norwegian (no)
Other versions
NO145793B (no
NO762932L (pt
Inventor
Herbert Merz
Gerhard Walther
Adolf Langbein
Klaus Stockhaus
Helmut Wick
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of NO762932L publication Critical patent/NO762932L/no
Publication of NO145793B publication Critical patent/NO145793B/no
Publication of NO145793C publication Critical patent/NO145793C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/06Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
    • C07D489/08Oxygen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO762932A 1975-08-27 1976-08-26 Analogifremgangsmaate for fremstilling av den fysiologisk aktive forbindelse n-(r-tetrahydrofurfuryl)-noroksymorfon NO145793C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19752538075 DE2538075A1 (de) 1975-08-27 1975-08-27 N-tetrahydrofurfuryl-noroxymorphone, deren saeureadditionssalze, diese enthaltende arzneimittel sowie verfahren zu ihrer herstellung

Publications (3)

Publication Number Publication Date
NO762932L NO762932L (pt) 1977-03-01
NO145793B NO145793B (no) 1982-02-22
NO145793C true NO145793C (no) 1982-06-02

Family

ID=5954931

Family Applications (1)

Application Number Title Priority Date Filing Date
NO762932A NO145793C (no) 1975-08-27 1976-08-26 Analogifremgangsmaate for fremstilling av den fysiologisk aktive forbindelse n-(r-tetrahydrofurfuryl)-noroksymorfon

Country Status (33)

Country Link
US (1) US4100288A (pt)
JP (1) JPS5231100A (pt)
AT (1) AT350737B (pt)
AU (1) AU499926B2 (pt)
BE (1) BE845563A (pt)
BG (2) BG27546A4 (pt)
CA (1) CA1068266A (pt)
CH (5) CH622521A5 (pt)
CS (2) CS192564B2 (pt)
DD (1) DD127145A5 (pt)
DE (1) DE2538075A1 (pt)
DK (1) DK143278C (pt)
ES (5) ES450897A1 (pt)
FI (1) FI762430A (pt)
FR (1) FR2321888A1 (pt)
GB (1) GB1519719A (pt)
GR (1) GR61158B (pt)
HU (1) HU176929B (pt)
IE (1) IE44069B1 (pt)
IL (1) IL50355A (pt)
LU (1) LU75667A1 (pt)
MX (1) MX4133E (pt)
NL (1) NL7609485A (pt)
NO (1) NO145793C (pt)
NZ (1) NZ181864A (pt)
PH (1) PH13780A (pt)
PL (2) PL109091B1 (pt)
PT (1) PT65521B (pt)
RO (1) RO69457A (pt)
SE (1) SE7609495L (pt)
SU (2) SU612631A3 (pt)
YU (1) YU208176A (pt)
ZA (1) ZA765120B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272541A (en) * 1978-06-02 1981-06-09 Miles Laboratories, Inc. 7,8 and 7-8 Substituted 4,5α-epoxymorphinan-6-one compounds, and methods of treating pain and drug dependence with them
US4272540A (en) * 1979-04-24 1981-06-09 Sisa, Incorporated 14-Methoxymorphinan-6-one compounds and therapeutic methods of treating pain and drug dependence with them
DE3220831A1 (de) * 1982-06-03 1983-12-08 Boehringer Ingelheim KG, 6507 Ingelheim N-(2-methoxyethyl)-noroxymorphon, dessen saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung
JP5586223B2 (ja) * 2006-04-21 2014-09-10 ネクター セラピューティクス モルヒノンの立体選択的還元
ES2708726T3 (es) * 2010-07-08 2019-04-10 Alkermes Pharma Ireland Ltd Proceso para la síntesis de morfinanos sustituidos
US9211293B2 (en) 2011-12-15 2015-12-15 Alkermes Pharma Ireland Limited Opioid agonist antagonist combinations
EP3003311A2 (en) 2013-05-24 2016-04-13 Alkermes Pharma Ireland Limited Methods for treating depressive symptoms
AU2014268361B2 (en) 2013-05-24 2018-09-06 Alkermes Pharma Ireland Limited Morphan and morphinan analogues, and methods of use
EP3755704A1 (en) * 2018-02-23 2020-12-30 Rhodes Technologies Inc. Novel opioid compounds and uses thereof
EP4243768A1 (en) 2020-11-12 2023-09-20 Alkermes Pharma Ireland Limited Immediate release multilayer tablet

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH446370A (de) 1964-03-05 1967-11-15 Hoffmann La Roche Verfahren zur Herstellung von Phenanthren-Derivaten
DE2238839A1 (de) * 1972-08-07 1974-02-14 Boehringer Sohn Ingelheim Neue morphinon-derivate, deren saeureadditionssalze, verfahren zu ihrer herstellung sowie ihre verwendung zur herstellung von arzneimitteln

Also Published As

Publication number Publication date
NO145793B (no) 1982-02-22
BG27545A3 (en) 1979-11-12
PT65521A (de) 1976-09-01
CH624115A5 (pt) 1981-07-15
DK143278C (da) 1981-12-07
PT65521B (de) 1978-07-04
NZ181864A (en) 1978-06-20
ES454084A1 (es) 1977-11-16
US4100288A (en) 1978-07-11
BE845563A (fr) 1977-02-28
CH624114A5 (pt) 1981-07-15
ZA765120B (en) 1978-05-30
RO69457A (ro) 1981-04-30
LU75667A1 (pt) 1977-09-13
CH624116A5 (pt) 1981-07-15
DD127145A5 (pt) 1977-09-07
SU638262A3 (ru) 1978-12-15
CA1068266A (en) 1979-12-18
MX4133E (es) 1982-01-06
IL50355A0 (en) 1976-10-31
CH624117A5 (pt) 1981-07-15
ATA553976A (de) 1978-11-15
AT350737B (de) 1979-06-11
AU1720176A (en) 1978-03-02
FR2321888B1 (pt) 1980-01-11
GB1519719A (en) 1978-08-02
CS192564B2 (en) 1979-08-31
PL110724B1 (en) 1980-07-31
ES454086A1 (es) 1977-11-16
ES450897A1 (es) 1977-12-01
DE2538075A1 (de) 1977-03-17
IL50355A (en) 1979-11-30
DK386876A (da) 1977-02-28
GR61158B (en) 1978-09-30
AU499926B2 (en) 1979-05-03
YU208176A (en) 1982-08-31
NO762932L (pt) 1977-03-01
SU612631A3 (ru) 1978-06-25
NL7609485A (nl) 1977-03-01
CH622521A5 (pt) 1981-04-15
ES454085A1 (es) 1977-11-16
JPS5231100A (en) 1977-03-09
HU176929B (hu) 1981-06-28
FR2321888A1 (fr) 1977-03-25
PH13780A (en) 1980-09-26
IE44069L (en) 1977-02-27
BG27546A4 (en) 1979-11-12
CS192599B2 (en) 1979-08-31
IE44069B1 (en) 1981-08-12
PL192020A1 (pl) 1979-03-12
PL109091B1 (en) 1980-05-31
ES454087A2 (es) 1977-11-16
SE7609495L (sv) 1977-02-28
DK143278B (da) 1981-08-03
FI762430A (pt) 1977-02-28

Similar Documents

Publication Publication Date Title
NO145199C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive nortropinestere.
NO143576C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive heterocykliske forbindelser
NO149106C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive benzcykloamider
NO141800C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive benzomorfaner.
NO143460C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive benzomorfaner.
NO142173C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme, 1,1-diaryl-1-oksadiazolalkylaminderivater
NO149428C (no) Fremgangsmaate for fremstilling av fysiologisk aktive prostaglandinderivater.
SE7604475L (sv) Forfarande for framstellning av 1,1,1-triaryl-alkylaminer
NO142838C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive isokinolinderivater
NO145198C (no) Analogifremgangsmaate til fremstilling av terapeutisk aktivt 1,2-benzisotia-zolinon-3
NO145793C (no) Analogifremgangsmaate for fremstilling av den fysiologisk aktive forbindelse n-(r-tetrahydrofurfuryl)-noroksymorfon
NO146199C (no) Fremgangsmaate for fremstilling av alfa-6-deoksy-5-hydroksytetracyklin-hydroklorid
NO141894C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive pyridobenzodiazepinoner
SE428686B (sv) Forfarande for framstellning av antiinflammatoriskt aktiva imidazoler
NO144108C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive n-(1-benzylpiperid-4-yl)-benzamider
NO144928C (no) Analogifremgangsmaate for fremstilling av fysiologisk aktive zantinderivater.
NO144457C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive dihydro-1,4-pyridiner
NO145383C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive substituerte indoler.
SE417509B (sv) Forfarande for framstellning av anthelmintiskt aktiva 2-karbalkoxiamino-5 (6)-fenyl-sulfonyloxi-bensimidazoler
NO145238C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive dihydrokarbostyril-derivater
SE428922B (sv) Forfarande for framstellning av 13, 14-dihydro-11-dioxi-prostaglandiner
NO146672C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive cinnolinderivater
NO147601C (no) Analogifremgangsmaate for fremstilling av den terapeutisk aktive forbindelse l-pyroglutamyl-l-histidyl-glycin
NO142403C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive isokinoliner.
NO773344L (no) Analogifremgangsmaate for fremstilling av fysiologisk aktive pyridobenzodiazepinoner