PL192020A1 - Sposob wytwarzania n-tetrahydrofurfurylo-noroksymorfonow - Google Patents
Sposob wytwarzania n-tetrahydrofurfurylo-noroksymorfonowInfo
- Publication number
- PL192020A1 PL192020A1 PL19202076A PL19202076A PL192020A1 PL 192020 A1 PL192020 A1 PL 192020A1 PL 19202076 A PL19202076 A PL 19202076A PL 19202076 A PL19202076 A PL 19202076A PL 192020 A1 PL192020 A1 PL 192020A1
- Authority
- PL
- Poland
- Prior art keywords
- noroxymorphone
- tetrahydrofurfuryl
- making
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19752538075 DE2538075A1 (de) | 1975-08-27 | 1975-08-27 | N-tetrahydrofurfuryl-noroxymorphone, deren saeureadditionssalze, diese enthaltende arzneimittel sowie verfahren zu ihrer herstellung |
Publications (2)
Publication Number | Publication Date |
---|---|
PL192020A1 true PL192020A1 (pl) | 1979-03-12 |
PL109091B1 PL109091B1 (en) | 1980-05-31 |
Family
ID=5954931
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL1976192020A PL109091B1 (en) | 1975-08-27 | 1976-08-26 | Method of producing new diastereomers of n-tetrahydrofurfuryle-noroxymorphones |
PL1976213963A PL110724B1 (en) | 1975-08-27 | 1976-08-26 | Method of producing new diastereomers of n-tetrahydrofurfurylonoroxymorphones |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL1976213963A PL110724B1 (en) | 1975-08-27 | 1976-08-26 | Method of producing new diastereomers of n-tetrahydrofurfurylonoroxymorphones |
Country Status (33)
Country | Link |
---|---|
US (1) | US4100288A (pl) |
JP (1) | JPS5231100A (pl) |
AT (1) | AT350737B (pl) |
AU (1) | AU499926B2 (pl) |
BE (1) | BE845563A (pl) |
BG (2) | BG27546A4 (pl) |
CA (1) | CA1068266A (pl) |
CH (5) | CH622521A5 (pl) |
CS (2) | CS192564B2 (pl) |
DD (1) | DD127145A5 (pl) |
DE (1) | DE2538075A1 (pl) |
DK (1) | DK143278C (pl) |
ES (5) | ES450897A1 (pl) |
FI (1) | FI762430A (pl) |
FR (1) | FR2321888A1 (pl) |
GB (1) | GB1519719A (pl) |
GR (1) | GR61158B (pl) |
HU (1) | HU176929B (pl) |
IE (1) | IE44069B1 (pl) |
IL (1) | IL50355A (pl) |
LU (1) | LU75667A1 (pl) |
MX (1) | MX4133E (pl) |
NL (1) | NL7609485A (pl) |
NO (1) | NO145793C (pl) |
NZ (1) | NZ181864A (pl) |
PH (1) | PH13780A (pl) |
PL (2) | PL109091B1 (pl) |
PT (1) | PT65521B (pl) |
RO (1) | RO69457A (pl) |
SE (1) | SE7609495L (pl) |
SU (2) | SU612631A3 (pl) |
YU (1) | YU208176A (pl) |
ZA (1) | ZA765120B (pl) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4272541A (en) * | 1978-06-02 | 1981-06-09 | Miles Laboratories, Inc. | 7,8 and 7-8 Substituted 4,5α-epoxymorphinan-6-one compounds, and methods of treating pain and drug dependence with them |
US4272540A (en) * | 1979-04-24 | 1981-06-09 | Sisa, Incorporated | 14-Methoxymorphinan-6-one compounds and therapeutic methods of treating pain and drug dependence with them |
DE3220831A1 (de) * | 1982-06-03 | 1983-12-08 | Boehringer Ingelheim KG, 6507 Ingelheim | N-(2-methoxyethyl)-noroxymorphon, dessen saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung |
JP5586223B2 (ja) * | 2006-04-21 | 2014-09-10 | ネクター セラピューティクス | モルヒノンの立体選択的還元 |
ES2708726T3 (es) * | 2010-07-08 | 2019-04-10 | Alkermes Pharma Ireland Ltd | Proceso para la síntesis de morfinanos sustituidos |
US9211293B2 (en) | 2011-12-15 | 2015-12-15 | Alkermes Pharma Ireland Limited | Opioid agonist antagonist combinations |
EP3003311A2 (en) | 2013-05-24 | 2016-04-13 | Alkermes Pharma Ireland Limited | Methods for treating depressive symptoms |
AU2014268361B2 (en) | 2013-05-24 | 2018-09-06 | Alkermes Pharma Ireland Limited | Morphan and morphinan analogues, and methods of use |
EP3755704A1 (en) * | 2018-02-23 | 2020-12-30 | Rhodes Technologies Inc. | Novel opioid compounds and uses thereof |
EP4243768A1 (en) | 2020-11-12 | 2023-09-20 | Alkermes Pharma Ireland Limited | Immediate release multilayer tablet |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH446370A (de) | 1964-03-05 | 1967-11-15 | Hoffmann La Roche | Verfahren zur Herstellung von Phenanthren-Derivaten |
DE2238839A1 (de) * | 1972-08-07 | 1974-02-14 | Boehringer Sohn Ingelheim | Neue morphinon-derivate, deren saeureadditionssalze, verfahren zu ihrer herstellung sowie ihre verwendung zur herstellung von arzneimitteln |
-
1975
- 1975-08-27 DE DE19752538075 patent/DE2538075A1/de not_active Withdrawn
-
1976
- 1976-07-28 AT AT553976A patent/AT350737B/de not_active IP Right Cessation
- 1976-08-12 PH PH18780A patent/PH13780A/en unknown
- 1976-08-13 US US05/714,045 patent/US4100288A/en not_active Expired - Lifetime
- 1976-08-13 RO RO7687297A patent/RO69457A/ro unknown
- 1976-08-21 ES ES450897A patent/ES450897A1/es not_active Expired
- 1976-08-23 SU SU762389512A patent/SU612631A3/ru active
- 1976-08-24 FI FI762430A patent/FI762430A/fi not_active Application Discontinuation
- 1976-08-25 CH CH1079676A patent/CH622521A5/de not_active IP Right Cessation
- 1976-08-25 CS CS765528A patent/CS192564B2/cs unknown
- 1976-08-25 CS CS778646A patent/CS192599B2/cs unknown
- 1976-08-25 DD DD194461A patent/DD127145A5/xx unknown
- 1976-08-25 BG BG7634743A patent/BG27546A4/xx unknown
- 1976-08-25 IL IL50355A patent/IL50355A/xx unknown
- 1976-08-25 BG BG7634062A patent/BG27545A3/xx unknown
- 1976-08-26 GB GB35603/76A patent/GB1519719A/en not_active Expired
- 1976-08-26 CA CA259,909A patent/CA1068266A/en not_active Expired
- 1976-08-26 YU YU02081/76A patent/YU208176A/xx unknown
- 1976-08-26 NZ NZ181864A patent/NZ181864A/xx unknown
- 1976-08-26 DK DK386876A patent/DK143278C/da active
- 1976-08-26 HU HU76BO1629A patent/HU176929B/hu unknown
- 1976-08-26 ZA ZA00765120A patent/ZA765120B/xx unknown
- 1976-08-26 PL PL1976192020A patent/PL109091B1/pl unknown
- 1976-08-26 IE IE1911/76A patent/IE44069B1/en unknown
- 1976-08-26 SE SE7609495A patent/SE7609495L/xx not_active Application Discontinuation
- 1976-08-26 JP JP51102168A patent/JPS5231100A/ja active Pending
- 1976-08-26 NL NL7609485A patent/NL7609485A/xx not_active Application Discontinuation
- 1976-08-26 NO NO762932A patent/NO145793C/no unknown
- 1976-08-26 GR GR51547A patent/GR61158B/el unknown
- 1976-08-26 LU LU75667A patent/LU75667A1/xx unknown
- 1976-08-26 PT PT65521A patent/PT65521B/pt unknown
- 1976-08-26 AU AU17201/76A patent/AU499926B2/en not_active Expired
- 1976-08-26 PL PL1976213963A patent/PL110724B1/pl unknown
- 1976-08-26 MX MX764858U patent/MX4133E/es unknown
- 1976-08-26 BE BE170118A patent/BE845563A/xx unknown
- 1976-08-27 FR FR7625985A patent/FR2321888A1/fr active Granted
- 1976-12-09 ES ES454087A patent/ES454087A2/es not_active Expired
- 1976-12-09 ES ES454085A patent/ES454085A1/es not_active Expired
- 1976-12-09 ES ES454084A patent/ES454084A1/es not_active Expired
- 1976-12-09 ES ES454086A patent/ES454086A1/es not_active Expired
-
1977
- 1977-05-31 SU SU772485952A patent/SU638262A3/ru active
-
1980
- 1980-09-18 CH CH699580A patent/CH624116A5/de not_active IP Right Cessation
- 1980-09-18 CH CH699480A patent/CH624115A5/de not_active IP Right Cessation
- 1980-09-18 CH CH699380A patent/CH624114A5/de not_active IP Right Cessation
- 1980-09-18 CH CH699680A patent/CH624117A5/de not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PL194291A1 (pl) | Sposob wytwarzania nowych pochodnych glikozoaminy | |
PL192890A1 (pl) | Sposob wytwarzania nowych 1-benzazoliloalkilo-4-podstawowych piperydyn | |
PL193761A1 (pl) | Sposob wytwarzania czteropierscieniowych chinonow | |
PL215007A1 (pl) | Sposob wytwarzania gamma-pironow | |
PL193183A1 (pl) | Sposob wytwarzania nowych pochodnych 11-dezoksy-16-arylo-omega-tetranorprostaglandyny | |
PL199298A1 (pl) | Sposob wytwarzania 2-bromo-6-fluoro-n-2-imidazolidynylideno-benzaminy | |
PL193861A1 (pl) | Sposob wytwarzania alfa-aminoketonow | |
PL192020A1 (pl) | Sposob wytwarzania n-tetrahydrofurfurylo-noroksymorfonow | |
PL199633A1 (pl) | Sposob wytwarzania 5-m-toliloksyuracylu | |
PL191156A1 (pl) | Sposob wytwarzania nowych epoksyandrostanow | |
PL96241B1 (pl) | Sposob wytwarzania 2-/2-podstawionych-4-tiazolilo/-benzimidazoli | |
PL202091A1 (pl) | Sposob wytwarzania gamma-pyronow | |
PL100616B1 (pl) | Sposob wytwarzania nowych eterowych pochodnych oksymu | |
PL193604A1 (pl) | Sposob wytwarzania nowych d-homosteroidow | |
PL100145B1 (pl) | Sposob wytwarzania nowych zwiazkow dwuureidowych | |
PL190303A1 (pl) | Sposob wytwarzania nowych enamin | |
PL202697A1 (pl) | Sposob wytwarzania 2-bromo-alfa-ergokryptyny | |
PL94616B1 (pl) | Sposob wytwarzania metyloheptenonu-2 | |
PL94617B1 (pl) | Sposob wytwarzania metyloheptenonu-2 | |
PL95878B1 (pl) | Sposob wytwarzania 2-acetamidobenzimidazolu | |
PL98457B1 (pl) | Sposob wytwarzania nowych chloroarylofosforanow | |
PL193219A1 (pl) | Sposob wytwarzania nowych aminoglikozydow 2-dezoksystreptaminy | |
SU546665A1 (ru) | Способ получени хлорлигнина | |
PL101164B1 (pl) | Sposob otrzymywania bromkow p-alkoksybenzylowych | |
PL95763B1 (pl) | Sposob otrzymywania bromoarylofosforanow |